Torthaí cuardaigh - Rima Al‐awar
- 1 - 20 toradh as 35 á dtaispeáint
- Téigh chuig an gcéad leathanach eile
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1
Asymmetric Synthesis of All the Known Phlegmarine Alkaloids de réir Bradley Wolfe, Adam H. Libby, Rima Al‐awar, Christopher J. Foti, Daniel L. Comins
Foilsithe / Cruthaithe 2010Artigo -
2
Small Molecule Kinase Inhibitor Screen Identifies Polo-Like Kinase 1 as a Target for Neuroblastoma Tumor-Initiating Cells de réir Natalie Grinshtein, Alessandro Datti, Mayumi Fujitani, David Uehling, Michaël Prakesch, Methvin Isaac, Meredith S. Irwin, Jeffrey L. Wrana, Rima Al‐awar, David R. Kaplan
Foilsithe / Cruthaithe 2011Artigo -
3
Metformin Pharmacokinetics in Mouse Tumors: Implications for Human Therapy de réir Ryan J.O. Dowling, Sonya H.L. Lam, C. Bassi, Samar Mouaaz, Ahmed Aman, Taira Kiyota, Rima Al‐awar, Pamela J. Goodwin, Vuk Stambolic
Foilsithe / Cruthaithe 2016Carta -
4
PI3K/AKT/mTOR inhibition in combination with doxorubicin is an effective therapy for leiomyosarcoma de réir Yael Babichev, Leah Kabaroff, Alessandro Datti, David Uehling, Methvin Isaac, Rima Al‐awar, Michaël Prakesch, Ren Sun, Paul C. Boutros, Rosemarie E. Venier, Brendan C. Dickson, Rebecca Gladdy
Foilsithe / Cruthaithe 2016Artigo -
5
Bromo-deaza-SAH: A potent and selective DOT1L inhibitor de réir Wenyu Yu, David Smil, Fengling Li, W. Tempel, O. Fedorov, Kong T. Nguyen, Yuri Bolshan, Rima Al‐awar, Stefan Knapp, C.H. Arrowsmith, Masoud Vedadi, Peter J. Brown, Matthieu Schapira
Foilsithe / Cruthaithe 2013Artigo -
6
Discovery of a Selective Inhibitor for the YEATS Domains of ENL/AF9 de réir Thomas Christott, James M. Bennett, Carmen H. Coxon, Octovia Monteiro, Charline Giroud, Viktor Beke, Suet Ling Felce, Vicki Gamble, C. Gileadi, Gennady Poda, Rima Al‐awar, Gillian Farnie, Oleg Fedorov
Foilsithe / Cruthaithe 2018Artigo -
7
A genome-wide CRISPR/Cas9 screen in acute myeloid leukemia cells identifies regulators of TAK-243 sensitivity de réir Samir H. Barghout, Ahmed Aman, Kazem Nouri, Zachary Blatman, Karen Arevalo, Geethu Emily Thomas, Neil MacLean, Rose Hurren, Troy Ketela, Mehakpreet Saini, Moustafa Abohawya, Taira Kiyota, Rima Al‐awar, Aaron D. Schimmer
Foilsithe / Cruthaithe 2021Artigo -
8
Gain-of-function p53 mutants co-opt chromatin pathways to drive cancer growth de réir Jiajun Zhu, Morgan A. Sammons, Greg Donahue, Zhixun Dou, Masoud Vedadi, Matthäus Getlik, Dalia Baršytė-Lovejoy, Rima Al‐awar, Bryson W. Katona, Ali Shilatifard, Jing Huang, Xianxin Hua, C.H. Arrowsmith, Shelley L. Berger
Foilsithe / Cruthaithe 2015Artigo -
9
Combined deletion of <scp>P</scp>ten and p53 in mammary epithelium accelerates triple‐negative breast cancer with dependency on e<scp>EF</scp>2<scp>K</scp> de réir Jeff C. Liu, Véronique Voisin, Sharon Wang, Dong‐Yu Wang, Robert A. Jones, Alessandro Datti, David Uehling, Rima Al‐awar, Sean E. Egan, Gary D. Bader, Ming‐Sound Tsao, Tak W. Mak, Eldad Zacksenhaus
Foilsithe / Cruthaithe 2014Artigo -
10
Synthesis, Optimization, and Evaluation of Novel Small Molecules as Antagonists of WDR5-MLL Interaction de réir Yuri Bolshan, Matthäus Getlik, Ekaterina Kuznetsova, Gregory A. Wasney, Taraneh Hajian, Gennadiy Poda, Kong T. Nguyen, Hong Wu, L. Dombrovski, Aiping Dong, Guillermo Senisterra, Matthieu Schapira, C.H. Arrowsmith, Peter J. Brown, Rima Al‐awar, Masoud Vedadi, David Smil
Foilsithe / Cruthaithe 2013Artigo -
11
Potent Targeting of the STAT3 Protein in Brain Cancer Stem Cells: A Promising Route for Treating Glioblastoma de réir Sina Haftchenary, H. Artee Luchman, Andriana O. Jouk, Anthony J. Veloso, Brent D. G. Page, Xin Cheng, Sean S.H. Dawson, Natalie Grinshtein, Vijay Shahani, Kağan Kerman, David R. Kaplan, Carly Griffin, Ahmed Aman, Rima Al‐awar, Samuel Weiss, Patrick T. Gunning
Foilsithe / Cruthaithe 2013Artigo -
12
Virus-Tumor Interactome Screen Reveals ER Stress Response Can Reprogram Resistant Cancers for Oncolytic Virus-Triggered Caspase-2 Cell Death de réir Douglas J. Mahoney, Charles Lefebvre, Kristina J. Allan, J Brun, Cina A. Sanaei, Stephen Baird, Nelson Pearce, S. A.‐M. Grönberg, Brian C. Wilson, Mikael Prakesh, Ahmed Aman, Methvin Isaac, Ahmed Mamai, David Uehling, Rima Al‐awar, Theresa Falls, Tommy Alain, David F. Stojdl
Foilsithe / Cruthaithe 2011Artigo -
13
Small molecule epigenetic screen identifies novel EZH2 and HDAC inhibitors that target glioblastoma brain tumor-initiating cells de réir Natalie Grinshtein, Constanza Rioseco, Richard Marcellus, David Uehling, Ahmed Aman, Xueqing Lun, Osamu Muto, Lauren Podmore, Jake Lever, Yaoqing Shen, Michael Blough, G. Cairncross, Stephen M. Robbins, Steven J.M. Jones, Marco A. Marra, Rima Al‐awar, Donna L. Senger, David R. Kaplan
Foilsithe / Cruthaithe 2016Artigo -
14
MYC Interacts with the G9a Histone Methyltransferase to Drive Transcriptional Repression and Tumorigenesis de réir William B. Tu, Yu-Jia Shiah, Corey Lourenco, Peter J. Mullen, Dharmendra Dingar, Cornelia Redel, Aaliya Tamachi, Wail Ba-Alawi, Ahmed Aman, Rima Al‐awar, David W. Cescon, Benjamin Haibe‐Kains, C.H. Arrowsmith, Brian Raught, Paul C. Boutros, Linda Z. Penn
Foilsithe / Cruthaithe 2018Artigo -
15
Interrogation of Functional Cell-Surface Markers Identifies CD151 Dependency in High-Grade Serous Ovarian Cancer de réir Mauricio Medrano, Laudine Communal, Kevin R. Brown, Marcin Iwanicki, Josée Normand, Joshua Paterson, Fabrice Sircoulomb, Paul M. Krzyzanowski, Marián Novak, Sasha A. Doodnauth, Fernando Suárez, Jane Cullis, Rima Al‐awar, Benjamin G. Neel, John D. McPherson, Ronny Drapkin, Laurie Ailles, Anne‐Marie Mes‐Masson, Robert Rottapel
Foilsithe / Cruthaithe 2017Artigo -
16
Small-molecule inhibition of MLL activity by disruption of its interaction with WDR5 de réir Guillermo Senisterra, Hong Wu, Abdellah Allali‐Hassani, Gregory A. Wasney, Dalia Baršytė-Lovejoy, L. Dombrovski, Aiping Dong, Kong T. Nguyen, David Smil, Yuri Bolshan, Taraneh Hajian, Hao He, Alma Seitova, Irene Chau, Fengling Li, Gennadiy Poda, Jean‐François Couture, Peter J. Brown, Rima Al‐awar, Matthieu Schapira, C.H. Arrowsmith, Masoud Vedadi
Foilsithe / Cruthaithe 2012Artigo -
17
Wnt Inhibitor Screen Reveals Iron Dependence of β-Catenin Signaling in Cancers de réir Siyuan Song, Tania Christova, Stephen Perusini, Solmaz Alizadeh, Ren-Yue Bao, Bryan W. Miller, Rose Hurren, Yulia Jitkova, Marcela Gronda, Methvin Isaac, Babu Joseph, Ratheesh Subramaniam, Ahmed Aman, Anh Chau, Donna E. Hogge, Scott J. Weir, James M. Kasper, Aaron D. Schimmer, Rima Al‐awar, Jeffrey L. Wrana, Liliana Attisano
Foilsithe / Cruthaithe 2011Artigo -
18
Discovery of Small-Molecule Antagonists of the PWWP Domain of NSD2 de réir Renato Ferreira de Freitas, Yanli Liu, Magdalena M. Szewczyk, Naimee Mehta, Fengling Li, David McLeod, Carlos Zepeda‐Velázquez, David Dilworth, Ronan P. Hanley, Elisa Gibson, Peter J. Brown, Rima Al‐awar, Lindsey I. James, C.H. Arrowsmith, Dalia Baršytė-Lovejoy, Jinrong Min, Masoud Vedadi, Matthieu Schapira, Abdellah Allali‐Hassani
Foilsithe / Cruthaithe 2020Pré-impressão -
19
Discovery of Small-Molecule Antagonists of the PWWP Domain of NSD2 de réir Renato Ferreira de Freitas, Yanli Liu, Magdalena M. Szewczyk, Naimee Mehta, Fengling Li, David McLeod, Carlos Zepeda‐Velázquez, David Dilworth, Ronan P. Hanley, Elisa Gibson, Peter J. Brown, Rima Al‐awar, Lindsey I. James, C.H. Arrowsmith, Dalia Baršytė-Lovejoy, Jinrong Min, Masoud Vedadi, Matthieu Schapira, Abdellah Allali‐Hassani
Foilsithe / Cruthaithe 2021Artigo -
20
Structure and mechanism of action of the hydroxy–aryl–aldehyde class of IRE1 endoribonuclease inhibitors de réir Mário Sanches, Nicole M. Duffy, Manisha Talukdar, N. Thevakumaran, David Chiovitti, Marella D. Canny, Kenneth Lee, Igor Kurinov, David Uehling, Rima Al‐awar, Gennadiy Poda, Michaël Prakesch, Brian J. Wilson, Victor Tam, Colleen Schweitzer, András Toró, Julie L. Lucas, D Vuga, Lynn Lehmann, Daniel Durocher, Qingping Zeng, John B. Patterson, Frank Sicheri
Foilsithe / Cruthaithe 2014Artigo
Uirlisí cuardaigh:
Ábhair a bhaineann le hábhar
Biology
Gene
Biochemistry
Cell biology
Chemistry
Cancer research
Genetics
Computational biology
Methylation
Methyltransferase
Cancer
Epigenetics
Histone
Small molecule
Medicine
Receptor
Enzyme
Gene expression
Histone methyltransferase
In vitro
Signal transduction
Amino acid
Cell culture
Drug discovery
Internal medicine
Molecular biology
Mutant
Pharmacology
RNA
Antagonist