Хайлтын үр дүнгүүд - Pascal Furet
- 24-н 1 - 20 үр дүнгүүдийг харуулж байна
- Дараагийн хуудас руу очих
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Catalytic inhibition of topoisomerase II by a novel rationally designed ATP-competitive purine analogue -н Patrick Chêne, Joëlle Rudloff, Joseph Schoepfer, Pascal Furet, Peter Meier, Zhiyan Qian, Jean‐Marc Schlaeppi, Rita Schmitz, Thomas Radimerski
Хэвлэсэн 2009Artigo -
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Crystal Structures of Human MdmX (HdmX) in Complex with p53 Peptide Analogues Reveal Surprising Conformational Changes -н Joerg Kallen, A. Goepfert, Anke Blechschmidt, Aude Izaac, Martin Geiser, Gisele Tavares, Paul Ramage, Pascal Furet, Keiichi Masuya, Joanna Lisztwan
Хэвлэсэн 2009Artigo -
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The small molecule specific EphB4 kinase inhibitor NVP-BHG712 inhibits VEGF driven angiogenesis -н Georg Martiny‐Baron, Philipp Holzer, Éric Billy, Christian Schnell, Joseph Brueggen, Mireille Ferretti, Niko Schmiedeberg, Jeanette M. Wood, Pascal Furet, Patricia Imbach
Хэвлэсэн 2010Artigo -
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2-Formylpyridyl Ureas as Highly Selective Reversible-Covalent Inhibitors of Fibroblast Growth Factor Receptor 4 -н Thomas Knoepfel, Pascal Furet, Robert Mah, Nicole Buschmann, Catherine Leblanc, Sebastien Ripoche, Diana Graus-Porta, Markus Wartmann, Inga Galuba, Robin A. Fairhurst
Хэвлэсэн 2018Artigo -
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Structural biology contributions to the discovery of drugs to treat chronic myelogenous leukaemia -н Sandra W. Cowan‐Jacob, Gabriele Fendrich, Andreas Floersheimer, Pascal Furet, Janis Liebetanz, Gabriele Rummel, Paul Rheinberger, Mario Centeleghe, Doriano Fabbro, Paul W. Manley
Хэвлэсэн 2006Artigo -
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Different Susceptibility of Protein Kinases to Staurosporine Inhibition -н Flavio Meggio, Arianna Donella Deana, Maria Ruzzene, Anna Maria Brunati, Luca Cesaro, Bárbara Guerra, Thomas Meyer, Helmut Mett, Doriano Fabbro, Pascal Furet, Grażyna Dobrowolska, Lorenzo A. Pinna
Хэвлэсэн 1995Artigo -
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p53 dynamics vary between tissues and are linked with radiation sensitivity -н Jacob Stewart-Ornstein, Yoshiko Iwamoto, Miles A. Miller, Mark Prytyskach, Stéphane Ferretti, Philipp Holzer, Joerg Kallen, Pascal Furet, Ashwini Jambhekar, William C. Forrester, Ralph Weissleder, Galit Lahav
Хэвлэсэн 2021Artigo -
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Biochemical and three-dimensional-structural study of the specific inhibition of protein kinase CK2 by [5-oxo-5,6-dihydroindolo-(1,2-a)quinazolin-7-yl]acetic acid (IQA) -н Stefania Sarno, E. De Moliner, Maria Ruzzene, Mario A. Pagano, Roberto Battistutta, Jenny Bain, Doriano Fabbro, Joseph Schoepfer, Matthew Elliott, Pascal Furet, Flavio Meggio, Giuseppe Zanotti, Lorenzo A. Pinna
Хэвлэсэн 2003Artigo -
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Capmatinib (INC280) Is Active Against Models of Non–Small Cell Lung Cancer and Other Cancer Types with Defined Mechanisms of MET Activation -н Sabrina Baltschukat, Barbara Schacher Engstler, Alan Huang, Huai-Xiang Hao, Angela Tam, Hui Qin Wang, Jinsheng Liang, Matthew T. DiMare, Hyo-Eun Carrie Bhang, Youzhen Wang, Pascal Furet, William R. Sellers, Francesco Hofmann, Joseph Schoepfer, Ralph Tiedt
Хэвлэсэн 2019Artigo -
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Potent, Selective, and Orally Bioavailable Inhibitors of VPS34 Provide Chemical Tools to Modulate Autophagy <i>in Vivo</i> -н Ayako Honda, Edmund Harrington, Iván Cornella‐Taracido, Pascal Furet, Mark Knapp, Meir Glick, Ellen Triantafellow, William E. Dowdle, Dmitri Wiedershain, Wieslawa Maniara, Christine Moore, Peter M. Finan, Lawrence G. Hamann, Brant Firestone, Leon O. Murphy, Erin P. Keaney
Хэвлэсэн 2015Artigo -
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In vivo antitumor activity of NVP-AEW541—A novel, potent, and selective inhibitor of the IGF-IR kinase -н Carlos Garcı́a-Echeverrı́a, Mark Pearson, Andreas Marti, Thomas Meyer, Juergen Mestan, Johann Zimmermann, Jiaping Gao, Josef Brueggen, Hans‐Georg Capraro, Robert Cozens, Dean B. Evans, Doriano Fabbro, Pascal Furet, Diana Graus Porta, Janis Liebetanz, Georg Martiny‐Baron, Stephan Ruetz, Francesco Hofmann
Хэвлэсэн 2004Artigo -
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A Drug Resistance Screen Using a Selective MET Inhibitor Reveals a Spectrum of Mutations That Partially Overlap with Activating Mutations Found in Cancer Patients -н Ralph Tiedt, Elisa Degenkolbe, Pascal Furet, B.A. Appleton, Sabrina Wagner, Joseph Schoepfer, Emily Buck, David A. Ruddy, John E. Monahan, Michael D. Jones, Jutta Blank, Dorothea Haasen, Peter Drueckes, Markus Wartmann, Clive McCarthy, William R. Sellers, Francesco Hofmann
Хэвлэсэн 2011Artigo -
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Identification and characterization of NVP-BEZ235, a new orally available dual phosphatidylinositol 3-kinase/mammalian target of rapamycin inhibitor with potent <i>in vivo</i> anti... -н Sauveur-Michel Maira, Frédéric Stauffer, Josef Brueggen, Pascal Furet, Christian Schnell, Christine Fritsch, Saskia M. Brachmann, Patrick Chêne, Alain De Pover, Kevin Schoemaker, Doriano Fabbro, Daniela Gabriel, Marjo Simonen, Leon O. Murphy, Peter M. Finan, William R. Sellers, Carlos García-Echeverría
Хэвлэсэн 2008Artigo -
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Potent and Selective Inhibition of Polycythemia by the Quinoxaline JAK2 Inhibitor NVP-BSK805 -н Fabienne Baffert, Catherine H. Régnier, Alain De Pover, Carole Pissot‐Soldermann, Gisele Tavares, Francesca Blasco, Josef Brueggen, Patrick Chêne, Peter Drueckes, Dirk Erdmann, Pascal Furet, Marc Gerspacher, Marc Lang, David Ledieu, Lynda Nolan, Stephan Ruetz, Joerg Trappe, Eric Vangrevelinghe, Markus Wartmann, Lorenza Wyder, Francesco Hofmann, Thomas Radimerski
Хэвлэсэн 2010Artigo -
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A distinct p53 target gene set predicts for response to the selective p53–HDM2 inhibitor NVP-CGM097 -н Sébastien Jeay, Swann Gaulis, Stéphane Ferretti, Hans Bitter, Moriko Ito, Therese‐Marie Stachyra, Masato Murakami, Stephan Ruetz, Daniel Guthy, Caroline Rynn, Michael Rugaard Jensen, Marion Wiesmann, Joerg Kallen, Pascal Furet, F. Gessier, Philipp Holzer, Keiichi Masuya, Jens Würthner, Ensar Halilovic, Francesco Hofmann, William R. Sellers, Diana Graus Porta
Хэвлэсэн 2015Artigo -
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FGF401, A First-In-Class Highly Selective and Potent FGFR4 Inhibitor for the Treatment of FGF19-Driven Hepatocellular Cancer -н Andreas Weiss, Flavia Adler, Alexandra Buhles, Christelle Stamm, Robin A. Fairhurst, Michael Kiffe, Dario Sterker, Mario Centeleghe, Markus Wartmann, Jacqueline Kinyamu-Akunda, Heiko S. Schadt, Philippe Couttet, Wolf Armin, Youzhen Wang, Patrizia Barzaghi-Rinaudo, Masato Murakami, Audrey Kauffmann, Thomas Knoepfel, Nicole Buschmann, Catherine Leblanc, Robert Mah, Pascal Furet, Jutta Blank, Francesco Hofmann, William R. Sellers, Diana Graus Porta
Хэвлэсэн 2019Artigo
Хайх хэрэгслүүд:
Холбогдох сэдвүүд
Biology
Cancer research
Biochemistry
Genetics
Chemistry
Kinase
Medicine
Cancer
Pharmacology
Gene
Signal transduction
In vivo
Internal medicine
Cell biology
Immunology
Tyrosine kinase
Protein kinase A
Receptor
ABL
Biotechnology
Colorectal cancer
Computational biology
Fibroblast growth factor
Fibroblast growth factor receptor
Mutation
Myeloid leukemia
Small molecule
Apoptosis
Cancer cell
Drug discovery