Bilaketaren emaitzak - P.M. Collins
- Erakusten 1 - 6 emaitzak -- 6
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Synthesis and Demonstration of the Biological Relevance of sp<sup>3</sup>‐rich Scaffolds Distantly Related to Natural Product Frameworks nork Daniel J. Foley, Philip G. E. Craven, P.M. Collins, Richard G. Doveston, A. Aimon, R. Talon, Ian Churcher, F. von Delft, Stephen Marsden, Adam Nelson
Argitaratua 2017Artigo -
3
A poised fragment library enables rapid synthetic expansion yielding the first reported inhibitors of PHIP(2), an atypical bromodomain nork Oakley B. Cox, T. Krojer, P.M. Collins, Octovia Monteiro, R. Talon, A.R. Bradley, O. Fedorov, Jahangir Amin, Brian D. Marsden, John Spencer, F. von Delft, Paul E. Brennan
Argitaratua 2015Artigo -
4
Characterization of Three Druggable Hot-Spots in the Aurora-A/TPX2 Interaction Using Biochemical, Biophysical, and Fragment-Based Approaches nork Patrick J. McIntyre, P.M. Collins, Lukáš Vrzal, Kristian Birchall, Laurence Arnold, Chido Mpamhanga, P.J. Coombs, Selena G. Burgess, Mark W. Richards, Anja Winter, Václav Veverka, F. von Delft, Andy Merritt, Richard Bayliss
Argitaratua 2017Artigo -
5
Crystallographic approach to fragment-based hit discovery against <i>Schistosoma mansoni</i> purine nucleoside phosphorylase nork Muhammad Faheem, Napoleão Fonseca Valadares, J. Brandão-Neto, Dom Bellini, P.M. Collins, Nicholas M. Pearce, Louise E. Bird, J.R. Torini, Raymond J. Owens, H.M. Pereira, F. von Delft, J.A.R.G. Barbosa
Argitaratua 2021Artigo -
6
Galectin‐3‐Binding Glycomimetics that Strongly Reduce Bleomycin‐Induced Lung Fibrosis and Modulate Intracellular Glycan Recognition nork Tamara Delaine, P.M. Collins, Alison C. MacKinnon, Gunjan Sharma, John Stegmayr, Vishal Kumar Rajput, Santanu Mandal, Ian Cumpstey, A. Larumbe, Bader A. Salameh, Barbro Kahl‐Knutsson, Hilde van Hattum, Monique van Scherpenzeel, Roland J. Pieters, Tariq Sethi, Hans Schambye, Stina Oredsson, Hakon Leffler, Helen Blanchard, Ulf J. Nilsson
Argitaratua 2016Artigo
Bilaketa egiteko lanabesak:
Antzeko gaiak
Biochemistry
Biology
Chemistry
Computational biology
Drug discovery
Gene
Combinatorial chemistry
Immunology
Internal medicine
Medicine
Stereochemistry
Algorithm
Aurora inhibitor
Aurora kinase
Bromodomain
Cell
Cell biology
Cell cycle
Chemical biology
Chemical space
Chromosome
Computer science
Druggability
Enzyme
Epigenetics
Fragment (logic)
Galectin
Galectin-3
Geometry
Glycan