Search Results - Martin Empting
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Single-domain antibodies for biomedical applications by Simon Krah, Christian Schröter, Stefan Zielonka, Martin Empting, Bernhard Valldorf, Harald Kolmar
Published 2015Revisão -
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Exploring the chemical space of ureidothiophene-2-carboxylic acids as inhibitors of the quorum sensing enzyme PqsD from Pseudomonas aeruginosa by J. Henning Sahner, Martin Empting, Ahmed A. M. Kamal, Elisabeth Weidel, Matthias F. Groh, Carsten Börger, Rolf W. Hartmann
Published 2015Artigo -
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Tracheal brush cells release acetylcholine in response to bitter tastants for paracrine and autocrine signaling by Monika I. Hollenhorst, Innokentij Jurastow, Rajender Nandigama, Silke Appenzeller, Lei Li, Jörg Vogel, Stephanie Wiederhold, Mike Althaus, Martin Empting, Janine Altmüller, Anna K. H. Hirsch, Veit Flockerzi, Brendan J. Canning, Antoine‐Emmanuel Saliba, Gabriela Krasteva‐Christ
Published 2019Artigo -
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Squalenyl Hydrogen Sulfate Nanoparticles for Simultaneous Delivery of Tobramycin and an Alkylquinolone Quorum Sensing Inhibitor Enable the Eradication of <i>P. aeruginosa</i> Biofi... by Duy‐Khiet Ho, Xabier Murgia, Chiara Rossi, Rebekka Christmann, Antonio G. Hüfner de Mello Martins, Marcus Koch, Anastasia Andreas, Jennifer Herrmann, Rolf Müller, Martin Empting, Rolf W. Hartmann, Didier Desmaële, Brigitta Loretz, Patrick Couvreur, Claus‐Michael Lehr
Published 2020Artigo -
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Towards Translation of PqsR Inverse Agonists: From In Vitro Efficacy Optimization to In Vivo Proof‐of‐Principle by Mostafa M. Hamed, Ahmed S. Abdelsamie, Katharina Rox, Christian Schütz, Andreas M. Kany, Teresa Röhrig, Stefan Schmelz, Wulf Blankenfeldt, Alejandro Arce‐Rodríguez, José Manuel Borrero‐de Acuña, Dieter Jahn, Jessica Rademacher, Felix C. Ringshausen, Nina Cramer, Burkhard Tümmler, Anna K. H. Hirsch, Rolf W. Hartmann, Martin Empting
Published 2023Artigo -
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A New PqsR Inverse Agonist Potentiates Tobramycin Efficacy to Eradicate <i>Pseudomonas aeruginosa</i> Biofilms by Christian Schütz, Duy‐Khiet Ho, Mostafa M. Hamed, Ahmed S. Abdelsamie, Teresa Röhrig, Christian Herr, Andreas M. Kany, Katharina Rox, Stefan Schmelz, Lorenz Siebenbürger, Marius Wirth, Carsten Börger, Samir Yahiaoui, Robert Bals, Andrea Scrima, Wulf Blankenfeldt, Justus C. Horstmann, Rebekka Christmann, Xabier Murgia, Marcus Koch, Aylin Berwanger, Brigitta Loretz, Anna K. H. Hirsch, Rolf W. Hartmann, Claus‐Michael Lehr, Martin Empting
Published 2021Artigo -
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Drug repurposing screen identifies lonafarnib as respiratory syncytial virus fusion protein inhibitor by Svenja M. Sake, Xiaoyu Zhang, Manoj Kumar Rajak, Melanie Urbanek‐Quaing, Arnaud Carpentier, Antonia P. Gunesch, Christina Grethe, Alina Matthaei, Jessica Rückert, Marie Galloux, Thibaut Larcher, Ronan Le Goffic, Fortune Hontonnou, Arnab K. Chatterjee, Kristen Johnson, Kaycie Morwood, Katharina Rox, Walid A. M. Elgaher, Jiabin Huang, Martin Wetzke, Gesine Hansen, Nicole Fischer, Jean-François Éléouët, Marie‐Anne Rameix‐Welti, Anna K. H. Hirsch, Elisabeth Herold, Martin Empting, Chris Lauber, Thomas F. Schulz, Thomas Krey, Sibylle Haid, Thomas Pietschmann
Published 2024Artigo -
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Identification of targetable vulnerabilities of PLK1-overexpressing cancers by synthetic dosage lethality by Chelsea E. Cunningham, Frederick S. Vizeacoumar, Yue Zhang, Liliia Kyrylenko, Simon Both, Vincent Maranda, He Dong, Jared D.W. Price, Peng Gao, Konrad Wagner, Yingwen Wu, Mary Lazell-Wright, Ashtalakshmi Ganapathysamy, Rithik Hari, Kalpana K. Bhanumathy, Connor Denomy, Anjali Saxena, Jeff P Vizeacoumar, Alain Morejon Morales, Faizaan Khan, Shayla R. Mosley, A. Chen, Tetiana Katrii, Ben G. E. Zoller, Karthic Rajamanickam, Prachi Walke, Lihui Gong, Hardikkumar Patel, Hussain Elhasasna, Renuka Dahiya, Omar Abuhussein, Anton E. Dmitriev, Tanya Freywald, Érika Prando Munhoz, Eytan Ruppin, Joo Sang Lee, Katharina Rox, Martin Köebel, Laura Hopkins, Cheng‐Han Lee, Sunil Yadav, Gilles Gasparoni, Walter Jörn, Anand Krishnan, Raju Datla, Behzad M. Toosi, Kristi Baker, Jalna Meens, David W. Cescon, Laurie Ailles, Scot C. Leary, Yuliang Wu, Martin Empting, Alexandra K. Kiemer, Andrew Freywald, Franco J. Vizeacoumar
Published 2025Artigo
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Biology
Biochemistry
Chemistry
Genetics
Gene
Bacteria
Microbiology
Pseudomonas aeruginosa
Quorum sensing
Biofilm
Virulence
Computational biology
Antibiotics
Pharmacology
Tobramycin
Antibody
Cell biology
Drug discovery
Enzyme
Gentamicin
Immunology
In vitro
Pyocyanin
Small molecule
Acetylcholine
Alternative splicing
Autocrine signalling
Autoinducer
Biosynthesis
Biotechnology