Risultati della ricerca - Marcel Scheepstra
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1
Bivalent Ligands for Protein Degradation in Drug Discovery di Marcel Scheepstra, Koen F. W. Hekking, Luc Van Hijfte, R.H.A. Folmer
Pubblicazione 2019Revisão -
2
Identification of an allosteric binding site for RORγt inhibition di Marcel Scheepstra, S. Leysen, Geert C. van Almen, J. Richard Miller, Jennifer Piesvaux, Victoria Kutilek, Hans van Eenennaam, Hongjun Zhang, Kenneth Barr, Sunil Nagpal, S.M. Soisson, Maria Kornienko, Kristen Wiley, Nathaniel L. Elsen, Sujata Sharma, Craig C. Correll, B. Wesley Trotter, Mario van der Stelt, Arthur Oubrie, Christian Ottmann, Gopal Parthasarathy, Luc Brunsveld
Pubblicazione 2015Artigo
Strumenti per la ricerca:
Soggetti correlati
Biochemistry
Biology
Cell biology
Chemistry
Computational biology
Drug discovery
Gene
Allosteric regulation
Binding site
Cereblon
Chemical biology
Computer science
Enzyme
Function (biology)
Ligand (biochemistry)
Linker
Nuclear receptor
Operating system
Proteasome
Protein degradation
Proteolysis
Proteome
RAR-related orphan receptor gamma
Receptor
Small molecule
Target protein
Transcription factor
Ubiquitin
Ubiquitin ligase