Ngā hua rapu - Lena M. Berger
- E whakaatu ana i te 1 - 4 hua o te 4
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1
Development of Potent Dual BET/HDAC Inhibitors via Pharmacophore Merging and Structure-Guided Optimization mā Nicolas Bauer, Dimitrios-Ilias Balourdas, Joel R. Schneider, Xin Zhang, Lena M. Berger, Benedict‐Tilman Berger, Martin P. Schwalm, N. Klopp, Jens T. Siveke, Stefan Knapp, Andreas C. Joerger
I whakaputaina 2024Artigo -
2
Design, Synthesis, and Evaluation of WD-Repeat-Containing Protein 5 (WDR5) Degraders mā Anja Dölle, Bikash Adhikari, Andreas Krämer, Janik Weckesser, Nicola Berner, Lena M. Berger, Mathias Diebold, Magdalena M. Szewczyk, Dalia Baršytė-Lovejoy, C.H. Arrowsmith, Jakob Gebel, Frank Löhr, Volker Dötsch, Martin Eilers, Stephanie Heinzlmeir, Bernhard Küster, Christoph Sotriffer, Elmar Wolf, Stefan Knapp
I whakaputaina 2021Artigo -
3
Design of a “Two-in-One” Mutant-Selective Epidermal Growth Factor Receptor Inhibitor That Spans the Orthosteric and Allosteric Sites mā Florian Wittlinger, David E. Heppner, Ciric To, Marcel Günther, Bo Hee Shin, Jaimin K. Rana, Anna M. Schmoker, Tyler S. Beyett, Lena M. Berger, Benedict‐Tilman Berger, Nicolas Bauer, James D. Vasta, Cesear Corona, Matthew B. Robers, Stefan Knapp, Pasi A. Jänne, Michael J. Eck, Stefan Laufer
I whakaputaina 2021Artigo -
4
Inhibition of DYRK1B BY C81 impedes inflammatory processes in leukocytes by reducing STAT3 activity mā Sarah Ciurus, Mohammed A.F. Elewa, Megan A. Palmer, Anne Wolf, Mandy Hector, Dominik C. Fuhrmann, Dominique Thomas, Robert Gurke, Martin P. Schwalm, Lena M. Berger, Thomas Zech, Luisa D. Burgers, Rolf Marschalek, Gerd Geißlinger, Stefan Knapp, Thomas Langmann, Franz Bracher, Andreas Weigert, Robert Fürst
I whakaputaina 2025Artigo
Ngā utauta rapu:
Ngā marau whai pānga
Biology
Chemistry
Biochemistry
Cancer research
Gene
Acetylation
Cancer
Computational biology
Genetics
Histone
Allosteric regulation
BRD4
Bromodomain
Cell biology
Cetuximab
Colorectal cancer
Computer science
EGFR inhibitors
Epidermal growth factor receptor
Epigenetics
Erlotinib
Gefitinib
HDAC1
Histone deacetylase
Immunology
Inflammation
Linker
Methylation
Methyltransferase
Mutant