検索結果 - Jianwei Che
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Covalent drugs targeting histidine – an unexploited opportunity? 著者: Jianwei Che, Lyn H. Jones
出版事項 2022Editorial -
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Targeting<i>MET</i>Dysregulation in Cancer 著者: Gonzalo Recondo, Jianwei Che, Pasi A. Jänne, Mark M. Awad
出版事項 2020Revisão -
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Expanding the Diversity of Allosteric Bcr-Abl Inhibitors 著者: Xianming Deng, Okram Barun, Qiang Ding, Jianming Zhang, Yongmun Choi, Francisco Adrián, Amy Wojciechowski, Guobao Zhang, Jianwei Che, Badry Bursulaya, Sandra W. Cowan‐Jacob, Gabriele Rummel, Taebo Sim, Nathanael S. Gray
出版事項 2010Artigo -
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Pharmacological blockade of TEAD–YAP reveals its therapeutic limitation in cancer cells 著者: Yang Sun, Lu Hu, Zhipeng Tao, Gopala K. Jarugumilli, Hannah Erb, Alka Singh, Qi Li, Jennifer L. Cotton, Patricia Greninger, Regina K. Egan, Y. Tony Ip, Cyril H. Benes, Jianwei Che, Junhao Mao, Xu Wu
出版事項 2022Artigo -
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Discovery of BAF312 (Siponimod), a Potent and Selective S1P Receptor Modulator 著者: Shifeng Pan, Nathanael S. Gray, Wenqi Gao, Yuan Mi, Yi Fan, Xing Wang, Tove Tuntland, Jianwei Che, Sophie Lefebvre, Yu Chen, Alan Chu, Klaus Hinterding, Anne Gardin, Peter End, Peter Heining, Christian Bruns, Nigel G. Cooke, Barbara Nuesslein‐Hildesheim
出版事項 2013Artigo -
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Discovery and resistance mechanism of a selective CDK12 degrader 著者: Baishan Jiang, Yang Gao, Jianwei Che, Wenchao Lu, Ines H. Kaltheuner, Ruben Dries, Marian Kalocsay, Matthew J. Berberich, Jie Jiang, Inchul You, Nicholas Kwiatkowski, Kristin M. Riching, Danette L. Daniels, Peter K. Sorger, Matthias Geyer, Tinghu Zhang, Nathanael S. Gray
出版事項 2021Artigo -
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Cereblon covalent modulation through structure-based design of histidine targeting chemical probes 著者: Justin T. Cruite, Geoffrey P. Dann, Jianwei Che, Katherine A. Donovan, Silas Ferrao, Scott B. Ficarro, Eric S. Fischer, Nathanael S. Gray, Fidel Huerta, Nikki R. Kong, Hu Liu, Jarrod A. Marto, Rebecca J. Metivier, Radosław P. Nowak, Breanna L. Zerfas, Lyn H. Jones
出版事項 2022Artigo -
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Exploring the target scope of KEAP1 E3 ligase-based PROTACs 著者: Guangyan Du, Jie Jiang, Nathaniel J. Henning, Nozhat Safaee, Eriko Koide, Radosław P. Nowak, Katherine A. Donovan, Hojong Yoon, Inchul You, Hong Yue, Nicholas A. Eleuteri, Zhixiang He, Zhengnian Li, Hubert T. Huang, Jianwei Che, Behnam Nabet, Tinghu Zhang, Eric S. Fischer, Nathanael S. Gray
出版事項 2022Artigo -
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Depletion of creatine phosphagen energetics with a covalent creatine kinase inhibitor 著者: Narek Darabedian, Wenzhi Ji, Mengyang Fan, Shan Lin, Hyuk‐Soo Seo, Ekaterina V. Vinogradova, Tomer M. Yaron, Evanna L. Mills, Haopeng Xiao, Kristine Senkane, Emily M. Huntsman, Jared L. Johnson, Jianwei Che, Lewis C. Cantley, Benjamin F. Cravatt, Sirano Dhe‐Paganon, Kimberly Stegmaier, Tinghu Zhang, Nathanael S. Gray, Edward T. Chouchani
出版事項 2023Artigo -
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Structure-Based Design of Y-Shaped Covalent TEAD Inhibitors 著者: Wenchao Lu, Mengyang Fan, Wenzhi Ji, Jason Tse, Inchul You, Scott B. Ficarro, Isidoro Tavares, Jianwei Che, Audrey Y. Kim, Xijun Zhu, Andrew S. Boghossian, Matthew G. Rees, Melissa M. Ronan, Jennifer A. Roth, Stephen M. Hinshaw, Behnam Nabet, Steven M. Corsello, Nicholas Kwiatkowski, Jarrod A. Marto, Tinghu Zhang, Nathanael S. Gray
出版事項 2023Artigo -
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The human zinc-binding cysteine proteome 著者: Nils Burger, Melanie J. Mittenbühler, Haopeng Xiao, Sang-Hee Shin, Shelley M Wei, Erik Henze, Sebastian Schindler, Sepideh Mehravar, David M. Wood, Jonathan J. Petrocelli, Yizhi Sun, Hans‐Georg Sprenger, Pedro Latorre‐Muro, Amanda L. Smythers, Luiz H. M. Bozi, Narek Darabedian, Yingde Zhu, Hyuk‐Soo Seo, Sirano Dhe‐Paganon, Jianwei Che, Edward T. Chouchani
出版事項 2024Artigo -
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Molecular Mechanisms of Acquired Resistance to MET Tyrosine Kinase Inhibitors in Patients with MET Exon 14–Mutant NSCLC 著者: Gonzalo Recondo, Magda Bahcall, Liam F. Spurr, Jianwei Che, Biagio Ricciuti, Giulia C. Leonardi, Ying‐Chun Lo, Yvonne Y. Li, Giuseppe Lamberti, Tom Nguyen, Marina S.D. Milan, Deepti Venkatraman, Renato Umeton, Cloud P. Paweletz, Adem Albayrak, Andrew D. Cherniack, Kristin S. Price, Stephen R. Fairclough, Mizuki Nishino, Lynette M. Sholl, Geoffrey R. Oxnard, Pasi A. Jänne, Mark M. Awad
出版事項 2020Artigo -
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Covalent disruptor of YAP-TEAD association suppresses defective Hippo signaling 著者: Mengyang Fan, Wenchao Lu, Jianwei Che, Nicholas Kwiatkowski, Yang Gao, Hyuk‐Soo Seo, Scott B. Ficarro, Prafulla C. Gokhale, Yao Liu, Ezekiel A. Geffken, Jimit Lakhani, Kijun Song, Miljan Kuljanin, Wenzhi Ji, Jie Jiang, Zhixiang He, Jason Tse, Andrew S. Boghossian, Matthew G. Rees, Melissa M. Ronan, Jennifer A. Roth, Joseph D. Mancias, Jarrod A. Marto, Sirano Dhe‐Paganon, Tinghu Zhang, Nathanael S. Gray
出版事項 2022Artigo -
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(<i>R</i>)-2-Phenylpyrrolidine Substituted Imidazopyridazines: A New Class of Potent and Selective Pan-TRK Inhibitors 著者: Ha-Soon Choi, Paul V. Rucker, Zhicheng Wang, Yi Fan, Pamela Albaugh, Greg Chopiuk, F. Gessier, Fangxian Sun, Francisco Adrián, Guoxun Liu, Tami Hood, Nanxin Li, Yong Jia, Jianwei Che, Susan McCormack, Allen Li, Jie Li, Auzon Steffy, AnneMarie Culazzo, Celine Tompkins, Van Phung, Andreas Kreusch, Min Lu, Bin Hu, Apurva Chaudhary, Mahavir Prashad, Tove Tuntland, Bo Liu, Jennifer L. Harris, H. Martin Seidel, Jon C. Loren, Valentina Molteni
出版事項 2015Artigo -
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Mapping the Degradable Kinome Provides a Resource for Expedited Degrader Development 著者: Katherine A. Donovan, Fleur M. Ferguson, Jonathan W. Bushman, Nicholas A. Eleuteri, Debabrata Bhunia, SeongShick Ryu, Li Tan, Kun Shi, Hong Yue, Xiaoxi Liu, Dennis Dobrovolsky, Baishan Jiang, Jinhua Wang, Mingfeng Hao, Inchul You, Mingxing Teng, Yanke Liang, John M. Hatcher, Zhengnian Li, Theresa Manz, Brian J. Groendyke, Wanyi Hu, Yunju Nam, Sandip Sengupta, Hanna Cho, Injae Shin, Michael P. Agius, Irene M. Ghobrial, W Michelle, Jianwei Che, Sara J. Buhrlage, Taebo Sim, Nathanael S. Gray, Eric S. Fischer
出版事項 2020Artigo -
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Imaging of <i>Plasmodium</i> Liver Stages to Drive Next-Generation Antimalarial Drug Discovery 著者: Stephan Meister, David Plouffe, Kelli Kuhen, Ghislain M. C. Bonamy, Tao Wu, S. Whitney Barnes, Selina Bopp, Rachel Borboa, A. Taylor Bright, Jianwei Che, Steve Cohen, Neekesh V. Dharia, Kerstin Gagaring, Montip Gettayacamin, Perry Gordon, Todd Groessl, Nobutaka Kato, Lee M, Case W. McNamara, David A. Fidock, A. S. Nagle, Tae‐gyu Nam, Wendy Richmond, Jason Roland, Matthias Rottmann, Bin Zhou, Patrick Froissard, Richard Glynne, Dominique Mazier, Jetsumon Sattabongkot, Peter G. Schultz, Tove Tuntland, John R. Walker, Yingyao Zhou, Arnab K. Chatterjee, Thierry T. Diagana, Elizabeth A. Winzeler
出版事項 2011Artigo -
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Targeting Wnt-driven cancer through the inhibition of Porcupine by LGK974 著者: Jun Liu, Shifeng Pan, Mindy H. Hsieh, Nicholas Ng, Fangxian Sun, Tao Wang, Shailaja Kasibhatla, Alwin G. Schuller, Allen G. Li, Cheng Dai, Jie Li, Celin Tompkins, AnneMarie Pferdekamper, Auzon Steffy, Jane Cheng, Colleen Kowal, Van Phung, Gui-Rong Guo, Yan Wang, Martin P. Graham, Shannon Flynn, J. Chad Brenner, Chun Li, Maria Cristina Villarroel, Peter G. Schultz, Xu Wu, Peter McNamara, William R. Sellers, Lilli Petruzzelli, Anthony Boral, H. Martin Seidel, Margaret E. McLaughlin, Jianwei Che, Thomas E. Carey, Gary Vanasse, Jennifer L. Harris
出版事項 2013Artigo
関連主題
Biology
Gene
Biochemistry
Computational biology
Cancer research
Chemistry
Cell biology
Genetics
Pharmacology
Cancer
Drug discovery
Enzyme
Medicine
Signal transduction
Ubiquitin
Bioinformatics
Cysteine
Kinase
Small molecule
Transcription factor
Ubiquitin ligase
Cereblon
Covalent bond
Drug
Drug development
Ecology
Internal medicine
Organic chemistry
Proteomics
Receptor