Výsledky vyhledávání - Jakka Raghavaiah
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1
Indole Chloropyridinyl Ester-Derived SARS-CoV-2 3CLpro Inhibitors: Enzyme Inhibition, Antiviral Efficacy, Structure–Activity Relationship, and X-ray Structural Studies Autor Arun K. Ghosh, Jakka Raghavaiah, Dana Shahabi, Monika Yadav, Brandon J. Anson, Emma K. Lendy, Shin-ichiro Hattori, Nobuyo Higashi‐Kuwata, Hiroaki Mitsuya, Andrew D. Mesecar
Vydáno 2021Artigo -
2
GRL-0920, an Indole Chloropyridinyl Ester, Completely Blocks SARS-CoV-2 Infection Autor Shin-ichiro Hattori, Nobuyo Higshi-Kuwata, Jakka Raghavaiah, Debananda Das, Haydar Bulut, David A. Davis, Yuki Takamatsu, Kouki Matsuda, Nobutoki Takamune, Naoki Kishimoto, Tadashi Okamura, Shogo Misumi, Robert Yarchoan, Kenji Maeda, Arun K. Ghosh, Hiroaki Mitsuya
Vydáno 2020Artigo -
3
A small molecule compound with an indole moiety inhibits the main protease of SARS-CoV-2 and blocks virus replication Autor Shin-ichiro Hattori, Nobuyo Higashi‐Kuwata, Hironori Hayashi, Srinivasa Rao Allu, Jakka Raghavaiah, Haydar Bulut, Debananda Das, Brandon J. Anson, Emma K. Lendy, Yuki Takamatsu, Nobutoki Takamune, Naoki Kishimoto, Kazutaka Murayama, Kazuya Hasegawa, Mi Li, David A. Davis, Eiichi Kodama, Robert Yarchoan, Alexander Wlodawer, Shogo Misumi, Andrew D. Mesecar, Arun K. Ghosh, Hiroaki Mitsuya
Vydáno 2021Artigo
Vyhledávací nástroje:
Související témata
Biochemistry
Chemistry
Enzyme
In vitro
Indole test
Biology
Protease
Stereochemistry
Vero cell
Virology
Virus
Antiretroviral therapy
Coronavirus disease 2019 (COVID-19)
Cytotoxicity
Disease
Enzyme inhibitor
IC50
Immunology
Infectious disease (medical specialty)
Infectivity
Lopinavir
Medicine
Moiety
Nitazoxanide
Pathology
Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2)
Small molecule
Structure–activity relationship
Viral load
Viral replication