Search Results - Haydar Bulut
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1
Single atom changes in newly synthesized HIV protease inhibitors reveal structural basis for extreme affinity, high genetic barrier, and adaptation to the HIV protease plasticity by Haydar Bulut, Shin‐ichiro Hattori, Hiromi Aoki-Ogata, Hironori Hayashi, Debananda Das, Manabu Aoki, David A. Davis, Kalapala Venkateswara Rao, Prasanth R. Nyalapatla, Arun K. Ghosh, Hiroaki Mitsuya
Published 2020Artigo -
2
Design and Development of Highly Potent HIV-1 Protease Inhibitors with a Crown-Like Oxotricyclic Core as the P2-Ligand To Combat Multidrug-Resistant HIV Variants by Arun K. Ghosh, Kalapala Venkateswara Rao, Prasanth R. Nyalapatla, Heather L. Osswald, Cuthbert D. Martyr, Manabu Aoki, Hironori Hayashi, Johnson Agniswamy, Yuan-Fang Wang, Haydar Bulut, Debananda Das, Irene T. Weber, Hiroaki Mitsuya
Published 2017Artigo -
3
GRL-0920, an Indole Chloropyridinyl Ester, Completely Blocks SARS-CoV-2 Infection by Shin-ichiro Hattori, Nobuyo Higshi-Kuwata, Jakka Raghavaiah, Debananda Das, Haydar Bulut, David A. Davis, Yuki Takamatsu, Kouki Matsuda, Nobutoki Takamune, Naoki Kishimoto, Tadashi Okamura, Shogo Misumi, Robert Yarchoan, Kenji Maeda, Arun K. Ghosh, Hiroaki Mitsuya
Published 2020Artigo -
4
Disruption of adaptor protein 2μ ( <scp>AP</scp> ‐2μ) in cochlear hair cells impairs vesicle reloading of synaptic release sites and hearing by Sangyong Jung, Tanja Maritzen, Carolin Wichmann, Zhizi Jing, Andreas Neef, Natalia H. Revelo, Hanan Al‐Moyed, Sandra Meese, Sonja M. Wojcik, Iliana Panou, Haydar Bulut, Peter Schu, Ralf Ficner, Ellen Reisinger, Silvio O. Rizzoli, Jakob Neef, Nicola Strenzke, Volker Haucke, Tobias Moser
Published 2015Artigo -
5
Role of the Clathrin Terminal Domain in Regulating Coated Pit Dynamics Revealed by Small Molecule Inhibition by Lisa von Kleist, Wiebke Stahlschmidt, Haydar Bulut, Kira V. Gromova, Dmytro Puchkov, Mark J. Robertson, Kylie A. MacGregor, N.V. Tomilin, Arndt Pechstein, Ngoc Chau, Megan Chircop, Jennette A. Sakoff, Jens Peter von Kries, Wolfram Saenger, Hans‐Georg Kräusslich, Oleg Shupliakov, Phillip J. Robinson, Adam McCluskey, Volker Haucke
Published 2011Artigo -
6
A novel central nervous system-penetrating protease inhibitor overcomes human immunodeficiency virus 1 resistance with unprecedented aM to pM potency by Manabu Aoki, Hironori Hayashi, Kalapala Venkateswara Rao, Debananda Das, Nobuyo Higashi‐Kuwata, Haydar Bulut, Hiromi Aoki-Ogata, Yuki Takamatsu, Ravikiran S. Yedidi, David A. Davis, Shin-ichiro Hattori, Noriko Nishida, Kazuya Hasegawa, Nobutoki Takamune, Prasanth R. Nyalapatla, Heather L. Osswald, Hirofumi Jono, Hideyuki Saito, Robert Yarchoan, Shogo Misumi, Arun K. Ghosh, Hiroaki Mitsuya
Published 2017Artigo -
7
Disruption of endocytosis through chemical inhibition of clathrin heavy chain function by Wim Dejonghe, Isha Sharma, Bram Denoo, Steven De Munck, Qing Lu, Kiril Mishev, Haydar Bulut, Evelien Mylle, Riet De Rycke, Mina Vasileva, Daniel V. Savatin, Wim Nerinckx, An Staes, Andrzej Drozdzecki, Dominique Audenaert, Klaas Yperman, Annemieke Madder, Jiřı́ Friml, Daniël Van Damme, Kris Gevaert, Volker Haucke, Savvas N. Savvides, Johan M. Winne, Eugenia Russinova
Published 2019Artigo -
8
A small molecule compound with an indole moiety inhibits the main protease of SARS-CoV-2 and blocks virus replication by Shin-ichiro Hattori, Nobuyo Higashi‐Kuwata, Hironori Hayashi, Srinivasa Rao Allu, Jakka Raghavaiah, Haydar Bulut, Debananda Das, Brandon J. Anson, Emma K. Lendy, Yuki Takamatsu, Nobutoki Takamune, Naoki Kishimoto, Kazutaka Murayama, Kazuya Hasegawa, Mi Li, David A. Davis, Eiichi Kodama, Robert Yarchoan, Alexander Wlodawer, Shogo Misumi, Andrew D. Mesecar, Arun K. Ghosh, Hiroaki Mitsuya
Published 2021Artigo
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Biochemistry
Biology
Chemistry
Enzyme
Protease
Virology
Antiretroviral therapy
Viral load
Human immunodeficiency virus (HIV)
In vitro
Receptor
Stereochemistry
Cell biology
Clathrin
Darunavir
Endocytosis
HIV-1 protease
Indole test
Medicine
Pathology
Protease inhibitor (pharmacology)
Small molecule
Vero cell
Virus
Amphiphysin
Art
Art history
Biophysics
Bulk endocytosis
Chemical biology