Canlyniadau Chwilio - Frederik Rombouts
- Dangos 1 - 6 canlyniadau o 6
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Pyrido[4,3-<i>e</i>][1,2,4]triazolo[4,3-<i>a</i>]pyrazines as Selective, Brain Penetrant Phosphodiesterase 2 (PDE2) Inhibitors gan Frederik Rombouts, Gary Tresadern, Peter Buijnsters, Xavier Langlois, Fulgencio Tovar, Thomas Steinbrecher, Greet Vanhoof, Marijke Somers, José-Ignacio Andrés, Andrés A. Trabanco
Cyhoeddwyd 2015Artigo -
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Structure-Based Design of a Potent, Selective, and Brain Penetrating PDE2 Inhibitor with Demonstrated Target Engagement gan Peter Buijnsters, Meri De Angelis, Xavier Langlois, Frederik Rombouts, Wendy E. Sanderson, Gary Tresadern, Alison Ritchie, Andrés A. Trabanco, Greet Vanhoof, Yves Van Roosbroeck, José-Ignacio Andrés
Cyhoeddwyd 2014Artigo -
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Preclinical Evaluation of<sup>18</sup>F-JNJ64349311, a Novel PET Tracer for Tau Imaging gan Lieven Declercq, Frederik Rombouts, Michel Koole, Katleen Fierens, Jonas Mariën, Xavier Langlois, José Ignacio Andrés, Mark E. Schmidt, Gregor J. Macdonald, Diederik Moechars, Wim Vanduffel, Thomas Tousseyn, Rik Vandenberghe, Koen Van Laere, Alfons Verbruggen, Guy Bormans
Cyhoeddwyd 2017Artigo -
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1,4-Oxazine β-Secretase 1 (BACE1) Inhibitors: From Hit Generation to Orally Bioavailable Brain Penetrant Leads gan Frederik Rombouts, Gary Tresadern, Óscar Delgado, Carolina Martínez‐Lamenca, Michiel Van Gool, Aránzazu García-Molina, Sergio A. Alonso de Diego, Daniel Oehlrich, Hana Prokopcová, José M. Martı́n-Alonso, Nigel Austin, Herman Borghys, Sven Van Brandt, Michel Surkyn, Michel De Cleyn, Ann Vos, Richard S. Alexander, Gregor J. Macdonald, Dieder Moechars, Harrie J. M. Gijsen, Andrés A. Trabanco
Cyhoeddwyd 2015Artigo
Offerynnau Chwilio:
Pynciau Perthynol
Chemistry
Medicine
Pharmacology
Biochemistry
Biology
Organic chemistry
Alzheimer's disease
Biotechnology
Combinatorial chemistry
Disease
Enzyme
In vitro
In vivo
Internal medicine
Neuroscience
Pathology
Penetrant (biochemical)
Phosphodiesterase
Alkyl
Amyloid precursor protein
Amyloid precursor protein secretase
Atrophy
Benzazepines
Bioavailability
Biodistribution
Cell biology
Central nervous system
Copper
Efflux
Erectile dysfunction