תוצאות חיפוש - Anang A. Shelat
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Nanomolar Affinity Small Molecule Correctors of Defective ΔF508-CFTR Chloride Channel Gating מאת Hong Yang, Anang A. Shelat, R. Kiplin Guy, Vadiraj S. Gopinath, Tonghui Ma, Kai Du, Gergely L. Lukács, Alessandro Taddei, Chiara Folli, Nicoletta Pedemonte, Luis J. V. Galietta, A. S. Verkman
יצא לאור 2003Artigo -
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Discovery of Trypanocidal Compounds by Whole Cell HTS of <i>Trypanosoma brucei</i> מאת Zachary B. Mackey, Arthur M. Baca, Jeremy P. Mallari, Beth Apsel, Anang A. Shelat, Elizabeth Hansell, Peter K. Chiang, Brian Wolff, Kiplin R. Guy, Janice A. Williams, James H. McKerrow
יצא לאור 2006Artigo -
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Discovery of Small Molecule Inhibitors of the Interaction of the Thyroid Hormone Receptor with Transcriptional Coregulators מאת Leggy A. Arnold, Eva Estébanez‐Perpiñá, Marie Togashi, Natalia Jouravel, Anang A. Shelat, Andrea C. McReynolds, Ellena Mar, Phuong Nguyen, John D. Baxter, Robert J. Fletterick, Paul Webb, R. Kiplin Guy
יצא לאור 2005Artigo -
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ABCG2 requires a single aromatic amino acid to “clamp” substrates and inhibitors into the binding pocket מאת Tomoka Gose, Talha Shafi, Yu Fukuda, Sourav Das, Yao Wang, Alice Allcock, Ailsa Gavan McHarg, J.A. Lynch, Taosheng Chen, Ikumi Tamai, Anang A. Shelat, Robert C. Ford, John D. Schuetz
יצא לאור 2020Artigo -
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Targeting Metabolic Reprogramming by Influenza Infection for Therapeutic Intervention מאת Heather S. Smallwood, Susu Duan, Marie Morfouace, Svetlana Rezinciuc, Barry L. Shulkin, Anang A. Shelat, Erika Zink, Sandra Milasta, Resha Bajracharya, Ajayi J. Oluwaseum, Martine F. Roussel, Douglas R. Green, Ljiljana Paša‐Tolić, Paul G. Thomas
יצא לאור 2017Artigo -
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Nuclear ULK1 promotes cell death in response to oxidative stress through PARP1 מאת Aashish Joshi, Rekha Iyengar, Joung Hyuck Joo, XiuJie Li-Harms, C. David Wright, Roberta Marino, Brett J Winborn, Aaron H. Phillips, Jamshid Temirov, Sebastiano Sciarretta, Richard W. Kriwacki, Junmin Peng, Anang A. Shelat, Mondira Kundu
יצא לאור 2015Artigo -
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Identification and Characterization of the First Small Molecule Inhibitor of MDMX מאת Damon R. Reed, Ying Shen, Anang A. Shelat, Leggy A. Arnold, Antonio M. Ferreira, Fangyi Zhu, Nicholas L. Mills, David C. Smithson, C.A. Regni, Donald Bashford, Samantha A. Cicero, Brenda A. Schulman, Aart G. Jochemsen, R. Kiplin Guy, Michael A. Dyer
יצא לאור 2010Artigo -
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Pemetrexed and Gemcitabine as Combination Therapy for the Treatment of Group3 Medulloblastoma מאת Marie Morfouace, Anang A. Shelat, Megan O. Jacus, Burgess B. Freeman, David C. Turner, Sarah Robinson, Frédérique Zindy, Yong‐Dong Wang, David Finkelstein, Olivier Ayrault, Laure Bihannic, Stéphanie Puget, Xiao‐Nan Li, James M. Olson, Giles Robinson, R. Kiplin Guy, Clinton F. Stewart, Amar Gajjar, Martine F. Roussel
יצא לאור 2014Artigo -
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Systematic Screening Identifies Dual PI3K and mTOR Inhibition as a Conserved Therapeutic Vulnerability in Osteosarcoma מאת Ankita Gupte, Emma K. Baker, Soo-San Wan, Elizabeth Stewart, Amos Hong Pheng Loh, Anang A. Shelat, Cathryn M. Gould, Alistair M. Chalk, Scott Taylor, Kurt Lackovic, Åsa Karlström, Anthony J. Mutsaers, Jayesh Desai, Piyush B. Madhamshettiwar, Andrew C.W. Zannettino, Christopher J. Burns, David C.S. Huang, Michael A. Dyer, Kaylene J. Simpson, Carl R. Walkley
יצא לאור 2015Artigo -
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Orthotopic patient-derived xenografts of paediatric solid tumours מאת Elizabeth Stewart, Sara M. Federico, Xiang Chen, Anang A. Shelat, Cori Bradley, Brittney Gordon, Åsa Karlström, Nathaniel Twarog, Michael R. Clay, Armita Bahrami, Burgess B. Freeman, Beisi Xu, Xin Zhou, Jianrong Wu, Victoria Honnell, Monica Ocarz, Kaley Blankenship, Jason Dapper, Elaine R. Mardis, Richard K. Wilson, James R. Downing, Jinghui Zhang, John Easton, Alberto S. Pappo, Michael A. Dyer
יצא לאור 2017Artigo -
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Targeting the DNA Repair Pathway in Ewing Sarcoma מאת Elizabeth Stewart, Ross Goshorn, Cori Bradley, Lyra Griffiths, Claudia A. Benavente, Nathaniel Twarog, Gregory M. Miller, William Caufield, Burgess B. Freeman, Armita Bahrami, Alberto S. Pappo, Jianrong Wu, Amos Hong Pheng Loh, Åsa Karlström, Chris Calabrese, Brittney Gordon, Lyudmila Tsurkan, M. Jason Hatfield, Philip M. Potter, Scott E. Snyder, Suresh Thiagarajan, Abbas Shirinifard, András Sablauer, Anang A. Shelat, Michael A. Dyer
יצא לאור 2014Artigo -
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Modeling and targeting of erythroleukemia by hematopoietic genome editing מאת Ilaria Iacobucci, Chunxu Qu, Elena Varotto, Laura J. Janke, Yang Xu, Aman Seth, Anang A. Shelat, Jake D. Friske, Reiji Fukano, Jiyang Yu, Burgess B. Freeman, James A. Kennedy, Adam S. Sperling, Rena Zheng, Yingzhe Wang, Harini Jogiraju, Kirsten Dickerson, Debbie Payne-Turner, Sarah M. Morris, Emily Hollis, Nina J Ghosn, Georgia E. Haggard, R. Coleman Lindsley, Benjamin L. Ebert, Charles G. Mullighan
יצא לאור 2021Artigo -
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Phenyl‐Glutarimides: Alternative Cereblon Binders for the Design of PROTACs מאת Jaeki Min, Anand Mayasundari, Fatemeh Keramatnia, Barbara Jonchère, Seung Wook Yang, Jamie Jarusiewicz, Marisa Actis, Sourav Das, Brandon Young, Jake Slavish, Lei Yang, Yong Li, Xiang Fu, Shalandus H. Garrett, Mi‐Kyung Yun, Zhenmei Li, Stanley Nithianantham, Sergio C. Chai, Taosheng Chen, Anang A. Shelat, Richard Lee, Gisele Nishiguchi, Stephen W. White, Martine F. Roussel, Patrick Ryan Potts, Marcus Fischer, Zoran Ranković
יצא לאור 2021Artigo
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