Search Results - Anang A. Shelat
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Catalysis, Specificity, and ACP Docking Site of Streptomyces coelicolor Malonyl-CoA:ACP Transacylase by Adrian T. Keatinge‐Clay, Anang A. Shelat, David F. Savage, Shiou‐Chuan Tsai, Larry J. W. Miercke, Joseph D. O’Connell, Chaitan Khosla, R. M. Stroud
Published 2003Artigo -
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Nanomolar Affinity Small Molecule Correctors of Defective ΔF508-CFTR Chloride Channel Gating by Hong Yang, Anang A. Shelat, R. Kiplin Guy, Vadiraj S. Gopinath, Tonghui Ma, Kai Du, Gergely L. Lukács, Alessandro Taddei, Chiara Folli, Nicoletta Pedemonte, Luis J. V. Galietta, A. S. Verkman
Published 2003Artigo -
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Discovery of Trypanocidal Compounds by Whole Cell HTS of <i>Trypanosoma brucei</i> by Zachary B. Mackey, Arthur M. Baca, Jeremy P. Mallari, Beth Apsel, Anang A. Shelat, Elizabeth Hansell, Peter K. Chiang, Brian Wolff, Kiplin R. Guy, Janice A. Williams, James H. McKerrow
Published 2006Artigo -
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Discovery of Small Molecule Inhibitors of the Interaction of the Thyroid Hormone Receptor with Transcriptional Coregulators by Leggy A. Arnold, Eva Estébanez‐Perpiñá, Marie Togashi, Natalia Jouravel, Anang A. Shelat, Andrea C. McReynolds, Ellena Mar, Phuong Nguyen, John D. Baxter, Robert J. Fletterick, Paul Webb, R. Kiplin Guy
Published 2005Artigo -
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Targeting Metabolic Reprogramming by Influenza Infection for Therapeutic Intervention by Heather S. Smallwood, Susu Duan, Marie Morfouace, Svetlana Rezinciuc, Barry L. Shulkin, Anang A. Shelat, Erika Zink, Sandra Milasta, Resha Bajracharya, Ajayi J. Oluwaseum, Martine F. Roussel, Douglas R. Green, Ljiljana Paša‐Tolić, Paul G. Thomas
Published 2017Artigo -
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Nuclear ULK1 promotes cell death in response to oxidative stress through PARP1 by Aashish Joshi, Rekha Iyengar, Joung Hyuck Joo, XiuJie Li-Harms, C. David Wright, Roberta Marino, Brett J Winborn, Aaron H. Phillips, Jamshid Temirov, Sebastiano Sciarretta, Richard W. Kriwacki, Junmin Peng, Anang A. Shelat, Mondira Kundu
Published 2015Artigo -
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Identification and Characterization of the First Small Molecule Inhibitor of MDMX by Damon R. Reed, Ying Shen, Anang A. Shelat, Leggy A. Arnold, Antonio M. Ferreira, Fangyi Zhu, Nicholas L. Mills, David C. Smithson, C.A. Regni, Donald Bashford, Samantha A. Cicero, Brenda A. Schulman, Aart G. Jochemsen, R. Kiplin Guy, Michael A. Dyer
Published 2010Artigo -
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Pemetrexed and Gemcitabine as Combination Therapy for the Treatment of Group3 Medulloblastoma by Marie Morfouace, Anang A. Shelat, Megan O. Jacus, Burgess B. Freeman, David C. Turner, Sarah Robinson, Frédérique Zindy, Yong‐Dong Wang, David Finkelstein, Olivier Ayrault, Laure Bihannic, Stéphanie Puget, Xiao‐Nan Li, James M. Olson, Giles Robinson, R. Kiplin Guy, Clinton F. Stewart, Amar Gajjar, Martine F. Roussel
Published 2014Artigo -
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Systematic Screening Identifies Dual PI3K and mTOR Inhibition as a Conserved Therapeutic Vulnerability in Osteosarcoma by Ankita Gupte, Emma K. Baker, Soo-San Wan, Elizabeth Stewart, Amos Hong Pheng Loh, Anang A. Shelat, Cathryn M. Gould, Alistair M. Chalk, Scott Taylor, Kurt Lackovic, Åsa Karlström, Anthony J. Mutsaers, Jayesh Desai, Piyush B. Madhamshettiwar, Andrew C.W. Zannettino, Christopher J. Burns, David C.S. Huang, Michael A. Dyer, Kaylene J. Simpson, Carl R. Walkley
Published 2015Artigo -
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Orthotopic patient-derived xenografts of paediatric solid tumours by Elizabeth Stewart, Sara M. Federico, Xiang Chen, Anang A. Shelat, Cori Bradley, Brittney Gordon, Åsa Karlström, Nathaniel Twarog, Michael R. Clay, Armita Bahrami, Burgess B. Freeman, Beisi Xu, Xin Zhou, Jianrong Wu, Victoria Honnell, Monica Ocarz, Kaley Blankenship, Jason Dapper, Elaine R. Mardis, Richard K. Wilson, James R. Downing, Jinghui Zhang, John Easton, Alberto S. Pappo, Michael A. Dyer
Published 2017Artigo -
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Targeting the DNA Repair Pathway in Ewing Sarcoma by Elizabeth Stewart, Ross Goshorn, Cori Bradley, Lyra Griffiths, Claudia A. Benavente, Nathaniel Twarog, Gregory M. Miller, William Caufield, Burgess B. Freeman, Armita Bahrami, Alberto S. Pappo, Jianrong Wu, Amos Hong Pheng Loh, Åsa Karlström, Chris Calabrese, Brittney Gordon, Lyudmila Tsurkan, M. Jason Hatfield, Philip M. Potter, Scott E. Snyder, Suresh Thiagarajan, Abbas Shirinifard, András Sablauer, Anang A. Shelat, Michael A. Dyer
Published 2014Artigo -
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Modeling and targeting of erythroleukemia by hematopoietic genome editing by Ilaria Iacobucci, Chunxu Qu, Elena Varotto, Laura J. Janke, Yang Xu, Aman Seth, Anang A. Shelat, Jake D. Friske, Reiji Fukano, Jiyang Yu, Burgess B. Freeman, James A. Kennedy, Adam S. Sperling, Rena Zheng, Yingzhe Wang, Harini Jogiraju, Kirsten Dickerson, Debbie Payne-Turner, Sarah M. Morris, Emily Hollis, Nina J Ghosn, Georgia E. Haggard, R. Coleman Lindsley, Benjamin L. Ebert, Charles G. Mullighan
Published 2021Artigo -
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Phenyl‐Glutarimides: Alternative Cereblon Binders for the Design of PROTACs by Jaeki Min, Anand Mayasundari, Fatemeh Keramatnia, Barbara Jonchère, Seung Wook Yang, Jamie Jarusiewicz, Marisa Actis, Sourav Das, Brandon Young, Jake Slavish, Lei Yang, Yong Li, Xiang Fu, Shalandus H. Garrett, Mi‐Kyung Yun, Zhenmei Li, Stanley Nithianantham, Sergio C. Chai, Taosheng Chen, Anang A. Shelat, Richard Lee, Gisele Nishiguchi, Stephen W. White, Martine F. Roussel, Patrick Ryan Potts, Marcus Fischer, Zoran Ranković
Published 2021Artigo -
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An Integrated In Vitro and In Vivo High-Throughput Screen Identifies Treatment Leads for Ependymoma by Jennifer M. Atkinson, Anang A. Shelat, Ángel M. Carcaboso, Tanya A. Kranenburg, Leggy A. Arnold, Nidal Boulos, Karen Wright, Robert A. Johnson, Helen Poppleton, Kumarasamypet M. Mohankumar, Clémentine Féau, Timothy N. Phoenix, Paul Gibson, Liqin Zhu, Yiai Tong, C.G. van Eden, David W. Ellison, Waldemar Priebe, Dimpy Koul, W.K. Alfred Yung, Amar Gajjar, Clinton F. Stewart, R. Kiplin Guy, Richard J. Gilbertson
Published 2011Artigo
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