Resultados de procura - van der Stelt, Mario
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Further evidence for the existence of a specific process for the membrane transport of anandamide. por Ligresti, Alessia, Morera, Enrico, Van Der Stelt, Mario, Monory, Krisztina, Lutz, Beat, Ortar, Giorgio, Di Marzo, Vincenzo
Publicado 2004Text -
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Protein Dynamics Influence the Enzymatic Activity of Phospholipase A/Acyltransferases 3 and 4 por Chatterjee, Soumya Deep, Zhou, Juan, Dasgupta, Rubin, Cramer-Blok, Anneloes, Timmer, Monika, van der Stelt, Mario, Ubbink, Marcellus
Publicado 2021Text -
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Forebrain-Specific Inactivation of G(q)/G(11) Family G Proteins Results in Age-Dependent Epilepsy and Impaired Endocannabinoid Formation por Wettschureck, Nina, van der Stelt, Mario, Tsubokawa, Hiroshi, Krestel, Heinz, Moers, Alexandra, Petrosino, Stefania, Schütz, Günther, Di Marzo, Vincenzo, Offermanns, Stefan
Publicado 2006Text -
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A natural substrate-based fluorescence assay for inhibitor screening on diacylglycerol lipase α por van der Wel, Tom, Janssen, Freek J., Baggelaar, Marc P., Deng, Hui, den Dulk, Hans, Overkleeft, Herman S., van der Stelt, Mario
Publicado 2015Text -
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Development of a Multiplexed Activity-Based Protein Profiling Assay to Evaluate Activity of Endocannabinoid Hydrolase Inhibitors por Janssen, Antonius P. A., van der Vliet, Daan, Bakker, Alexander T., Jiang, Ming, Grimm, Sebastian H., Campiani, Giuseppe, Butini, Stefania, van der Stelt, Mario
Publicado 2018Text -
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Anandamide acts as an intracellular messenger amplifying Ca(2+) influx via TRPV1 channels por van der Stelt, Mario, Trevisani, Marcello, Vellani, Vittorio, De Petrocellis, Luciano, Schiano Moriello, Aniello, Campi, Barbara, McNaughton, Peter, Geppetti, Piero, Di Marzo, Vincenzo
Publicado 2005Text -
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Anti-neuroinflammatory effects of GPR55 antagonists in LPS-activated primary microglial cells por Saliba, Soraya Wilke, Jauch, Hannah, Gargouri, Brahim, Keil, Albrecht, Hurrle, Thomas, Volz, Nicole, Mohr, Florian, van der Stelt, Mario, Bräse, Stefan, Fiebich, Bernd L.
Publicado 2018Text -
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Structure Kinetics Relationships and Molecular Dynamics Show Crucial Role for Heterocycle Leaving Group in Irreversible Diacylglycerol Lipase Inhibitors por Janssen, Antonius P.A., van Hengst, Jacob M.A., Béquignon, Olivier J.M., Deng, Hui, van Westen, Gerard J.P., van der Stelt, Mario
Publicado 2019Text -
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Evaluation of different drug classes on transient sciatic nerve injury-depressed marble burying in mice por Wilkerson, Jenny L, Curry, Zachary A, Kinlow, Pamela D, Mason, Brittany L, Hsu, Ku-Lung, van der Stelt, Mario, Cravatt, Benjamin F, Lichtman, Aron H
Publicado 2018Text -
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Structure–Activity Relationship Studies of Pyrimidine-4-Carboxamides as Inhibitors of N-Acylphosphatidylethanolamine Phospholipase D por Mock, Elliot D., Kotsogianni, Ioli, Driever, Wouter P. F., Fonseca, Carmen S., Vooijs, Jelle M., den Dulk, Hans, van Boeckel, Constant A. A., van der Stelt, Mario
Publicado 2020Text -
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Development of a Cannabinoid-Based Photoaffinity Probe to Determine the Δ(8/9)-Tetrahydrocannabinol Protein Interaction Landscape in Neuroblastoma Cells por Soethoudt, Marjolein, Alachouzos, Georgios, van Rooden, Eva J., Moya-Garzón, María Dolores, van den Berg, Richard J.B.H.N., Heitman, Laura H., van der Stelt, Mario
Publicado 2018Text -
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An Affinity-Based Probe for the Human Adenosine A(2A) Receptor por Yang, Xue, Michiels, Thomas J. M., de Jong, Coen, Soethoudt, Marjolein, Dekker, Niek, Gordon, Euan, van der Stelt, Mario, Heitman, Laura H., van der Es, Daan, IJzerman, Adriaan P.
Publicado 2018Text -
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Stress-induced modulation of endocannabinoid signaling leads to delayed strengthening of synaptic connectivity in the amygdala por Yasmin, Farhana, Colangeli, Roberto, Morena, Maria, Filipski, Sarah, van der Stelt, Mario, Pittman, Quentin J., Hillard, Cecilia J., Teskey, G. Campbell, McEwen, Bruce S., Hill, Matthew N., Chattarji, Sumantra
Publicado 2020Text -
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Olaparib‐Based Photoaffinity Probes for PARP‐1 Detection in Living Cells por Voorneveld, Jim, Florea, Bogdan I., Bakkum, Thomas, Mendowicz, Rafal J., van der Veer, Miriam S., Gagestein, Berend, van Kasteren, Sander I., van der Stelt, Mario, Overkleeft, Herman S., Filippov, Dmitri V.
Publicado 2020Text -
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Cannabinoid type 1 receptor inverse agonism attenuates dyslipidemia and atherosclerosis in APOE∗3-Leiden.CETP mice por van Eenige, Robin, Ying, Zhixiong, Tambyrajah, Lauren, Pronk, Amanda C.M., Blomberg, Niek, Giera, Martin, Wang, Yanan, Coskun, Tamer, van der Stelt, Mario, Rensen, Patrick C.N., Kooijman, Sander
Publicado 2021Text -
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Chemical Proteomics Reveals Off-Targets of the Anandamide Reuptake Inhibitor WOBE437 por Gagestein, Berend, Stevens, Anna F., Fazio, Domenico, Florea, Bogdan I., van der Wel, Tom, Bakker, Alexander T., Fezza, Filomena, Dulk, Hans den, Overkleeft, Herman S., Maccarrone, Mauro, van der Stelt, Mario
Publicado 2022Text