Search Results - van der Stelt, Mario
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Forebrain-Specific Inactivation of G(q)/G(11) Family G Proteins Results in Age-Dependent Epilepsy and Impaired Endocannabinoid Formation by Wettschureck, Nina, van der Stelt, Mario, Tsubokawa, Hiroshi, Krestel, Heinz, Moers, Alexandra, Petrosino, Stefania, Schütz, Günther, Di Marzo, Vincenzo, Offermanns, Stefan
Published 2006Text -
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Development of a Multiplexed Activity-Based Protein Profiling Assay to Evaluate Activity of Endocannabinoid Hydrolase Inhibitors by Janssen, Antonius P. A., van der Vliet, Daan, Bakker, Alexander T., Jiang, Ming, Grimm, Sebastian H., Campiani, Giuseppe, Butini, Stefania, van der Stelt, Mario
Published 2018Text -
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Anandamide acts as an intracellular messenger amplifying Ca(2+) influx via TRPV1 channels by van der Stelt, Mario, Trevisani, Marcello, Vellani, Vittorio, De Petrocellis, Luciano, Schiano Moriello, Aniello, Campi, Barbara, McNaughton, Peter, Geppetti, Piero, Di Marzo, Vincenzo
Published 2005Text -
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Anti-neuroinflammatory effects of GPR55 antagonists in LPS-activated primary microglial cells by Saliba, Soraya Wilke, Jauch, Hannah, Gargouri, Brahim, Keil, Albrecht, Hurrle, Thomas, Volz, Nicole, Mohr, Florian, van der Stelt, Mario, Bräse, Stefan, Fiebich, Bernd L.
Published 2018Text -
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Structure Kinetics Relationships and Molecular Dynamics Show Crucial Role for Heterocycle Leaving Group in Irreversible Diacylglycerol Lipase Inhibitors by Janssen, Antonius P.A., van Hengst, Jacob M.A., Béquignon, Olivier J.M., Deng, Hui, van Westen, Gerard J.P., van der Stelt, Mario
Published 2019Text -
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Evaluation of different drug classes on transient sciatic nerve injury-depressed marble burying in mice by Wilkerson, Jenny L, Curry, Zachary A, Kinlow, Pamela D, Mason, Brittany L, Hsu, Ku-Lung, van der Stelt, Mario, Cravatt, Benjamin F, Lichtman, Aron H
Published 2018Text -
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Structure–Activity Relationship Studies of Pyrimidine-4-Carboxamides as Inhibitors of N-Acylphosphatidylethanolamine Phospholipase D by Mock, Elliot D., Kotsogianni, Ioli, Driever, Wouter P. F., Fonseca, Carmen S., Vooijs, Jelle M., den Dulk, Hans, van Boeckel, Constant A. A., van der Stelt, Mario
Published 2020Text -
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Development of a Cannabinoid-Based Photoaffinity Probe to Determine the Δ(8/9)-Tetrahydrocannabinol Protein Interaction Landscape in Neuroblastoma Cells by Soethoudt, Marjolein, Alachouzos, Georgios, van Rooden, Eva J., Moya-Garzón, María Dolores, van den Berg, Richard J.B.H.N., Heitman, Laura H., van der Stelt, Mario
Published 2018Text -
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An Affinity-Based Probe for the Human Adenosine A(2A) Receptor by Yang, Xue, Michiels, Thomas J. M., de Jong, Coen, Soethoudt, Marjolein, Dekker, Niek, Gordon, Euan, van der Stelt, Mario, Heitman, Laura H., van der Es, Daan, IJzerman, Adriaan P.
Published 2018Text -
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Stress-induced modulation of endocannabinoid signaling leads to delayed strengthening of synaptic connectivity in the amygdala by Yasmin, Farhana, Colangeli, Roberto, Morena, Maria, Filipski, Sarah, van der Stelt, Mario, Pittman, Quentin J., Hillard, Cecilia J., Teskey, G. Campbell, McEwen, Bruce S., Hill, Matthew N., Chattarji, Sumantra
Published 2020Text -
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Olaparib‐Based Photoaffinity Probes for PARP‐1 Detection in Living Cells by Voorneveld, Jim, Florea, Bogdan I., Bakkum, Thomas, Mendowicz, Rafal J., van der Veer, Miriam S., Gagestein, Berend, van Kasteren, Sander I., van der Stelt, Mario, Overkleeft, Herman S., Filippov, Dmitri V.
Published 2020Text -
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Cannabinoid type 1 receptor inverse agonism attenuates dyslipidemia and atherosclerosis in APOE∗3-Leiden.CETP mice by van Eenige, Robin, Ying, Zhixiong, Tambyrajah, Lauren, Pronk, Amanda C.M., Blomberg, Niek, Giera, Martin, Wang, Yanan, Coskun, Tamer, van der Stelt, Mario, Rensen, Patrick C.N., Kooijman, Sander
Published 2021Text -
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Chemical Proteomics Reveals Off-Targets of the Anandamide Reuptake Inhibitor WOBE437 by Gagestein, Berend, Stevens, Anna F., Fazio, Domenico, Florea, Bogdan I., van der Wel, Tom, Bakker, Alexander T., Fezza, Filomena, Dulk, Hans den, Overkleeft, Herman S., Maccarrone, Mauro, van der Stelt, Mario
Published 2022Text