Výsledky vyhledávání - van der Stelt, Mario
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Protein Dynamics Influence the Enzymatic Activity of Phospholipase A/Acyltransferases 3 and 4 Autor Chatterjee, Soumya Deep, Zhou, Juan, Dasgupta, Rubin, Cramer-Blok, Anneloes, Timmer, Monika, van der Stelt, Mario, Ubbink, Marcellus
Vydáno 2021Text -
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Forebrain-Specific Inactivation of G(q)/G(11) Family G Proteins Results in Age-Dependent Epilepsy and Impaired Endocannabinoid Formation Autor Wettschureck, Nina, van der Stelt, Mario, Tsubokawa, Hiroshi, Krestel, Heinz, Moers, Alexandra, Petrosino, Stefania, Schütz, Günther, Di Marzo, Vincenzo, Offermanns, Stefan
Vydáno 2006Text -
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Development of a Multiplexed Activity-Based Protein Profiling Assay to Evaluate Activity of Endocannabinoid Hydrolase Inhibitors Autor Janssen, Antonius P. A., van der Vliet, Daan, Bakker, Alexander T., Jiang, Ming, Grimm, Sebastian H., Campiani, Giuseppe, Butini, Stefania, van der Stelt, Mario
Vydáno 2018Text -
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Anandamide acts as an intracellular messenger amplifying Ca(2+) influx via TRPV1 channels Autor van der Stelt, Mario, Trevisani, Marcello, Vellani, Vittorio, De Petrocellis, Luciano, Schiano Moriello, Aniello, Campi, Barbara, McNaughton, Peter, Geppetti, Piero, Di Marzo, Vincenzo
Vydáno 2005Text -
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Anti-neuroinflammatory effects of GPR55 antagonists in LPS-activated primary microglial cells Autor Saliba, Soraya Wilke, Jauch, Hannah, Gargouri, Brahim, Keil, Albrecht, Hurrle, Thomas, Volz, Nicole, Mohr, Florian, van der Stelt, Mario, Bräse, Stefan, Fiebich, Bernd L.
Vydáno 2018Text -
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Structure Kinetics Relationships and Molecular Dynamics Show Crucial Role for Heterocycle Leaving Group in Irreversible Diacylglycerol Lipase Inhibitors Autor Janssen, Antonius P.A., van Hengst, Jacob M.A., Béquignon, Olivier J.M., Deng, Hui, van Westen, Gerard J.P., van der Stelt, Mario
Vydáno 2019Text -
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Evaluation of different drug classes on transient sciatic nerve injury-depressed marble burying in mice Autor Wilkerson, Jenny L, Curry, Zachary A, Kinlow, Pamela D, Mason, Brittany L, Hsu, Ku-Lung, van der Stelt, Mario, Cravatt, Benjamin F, Lichtman, Aron H
Vydáno 2018Text -
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Structure–Activity Relationship Studies of Pyrimidine-4-Carboxamides as Inhibitors of N-Acylphosphatidylethanolamine Phospholipase D Autor Mock, Elliot D., Kotsogianni, Ioli, Driever, Wouter P. F., Fonseca, Carmen S., Vooijs, Jelle M., den Dulk, Hans, van Boeckel, Constant A. A., van der Stelt, Mario
Vydáno 2020Text -
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Development of a Cannabinoid-Based Photoaffinity Probe to Determine the Δ(8/9)-Tetrahydrocannabinol Protein Interaction Landscape in Neuroblastoma Cells Autor Soethoudt, Marjolein, Alachouzos, Georgios, van Rooden, Eva J., Moya-Garzón, María Dolores, van den Berg, Richard J.B.H.N., Heitman, Laura H., van der Stelt, Mario
Vydáno 2018Text -
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An Affinity-Based Probe for the Human Adenosine A(2A) Receptor Autor Yang, Xue, Michiels, Thomas J. M., de Jong, Coen, Soethoudt, Marjolein, Dekker, Niek, Gordon, Euan, van der Stelt, Mario, Heitman, Laura H., van der Es, Daan, IJzerman, Adriaan P.
Vydáno 2018Text -
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Stress-induced modulation of endocannabinoid signaling leads to delayed strengthening of synaptic connectivity in the amygdala Autor Yasmin, Farhana, Colangeli, Roberto, Morena, Maria, Filipski, Sarah, van der Stelt, Mario, Pittman, Quentin J., Hillard, Cecilia J., Teskey, G. Campbell, McEwen, Bruce S., Hill, Matthew N., Chattarji, Sumantra
Vydáno 2020Text -
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Olaparib‐Based Photoaffinity Probes for PARP‐1 Detection in Living Cells Autor Voorneveld, Jim, Florea, Bogdan I., Bakkum, Thomas, Mendowicz, Rafal J., van der Veer, Miriam S., Gagestein, Berend, van Kasteren, Sander I., van der Stelt, Mario, Overkleeft, Herman S., Filippov, Dmitri V.
Vydáno 2020Text -
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Cannabinoid type 1 receptor inverse agonism attenuates dyslipidemia and atherosclerosis in APOE∗3-Leiden.CETP mice Autor van Eenige, Robin, Ying, Zhixiong, Tambyrajah, Lauren, Pronk, Amanda C.M., Blomberg, Niek, Giera, Martin, Wang, Yanan, Coskun, Tamer, van der Stelt, Mario, Rensen, Patrick C.N., Kooijman, Sander
Vydáno 2021Text -
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Chemical Proteomics Reveals Off-Targets of the Anandamide Reuptake Inhibitor WOBE437 Autor Gagestein, Berend, Stevens, Anna F., Fazio, Domenico, Florea, Bogdan I., van der Wel, Tom, Bakker, Alexander T., Fezza, Filomena, Dulk, Hans den, Overkleeft, Herman S., Maccarrone, Mauro, van der Stelt, Mario
Vydáno 2022Text