Resultats de la cerca - van der Stelt, Mario
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Further evidence for the existence of a specific process for the membrane transport of anandamide. per Ligresti, Alessia, Morera, Enrico, Van Der Stelt, Mario, Monory, Krisztina, Lutz, Beat, Ortar, Giorgio, Di Marzo, Vincenzo
Publicat 2004Text -
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Protein Dynamics Influence the Enzymatic Activity of Phospholipase A/Acyltransferases 3 and 4 per Chatterjee, Soumya Deep, Zhou, Juan, Dasgupta, Rubin, Cramer-Blok, Anneloes, Timmer, Monika, van der Stelt, Mario, Ubbink, Marcellus
Publicat 2021Text -
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Forebrain-Specific Inactivation of G(q)/G(11) Family G Proteins Results in Age-Dependent Epilepsy and Impaired Endocannabinoid Formation per Wettschureck, Nina, van der Stelt, Mario, Tsubokawa, Hiroshi, Krestel, Heinz, Moers, Alexandra, Petrosino, Stefania, Schütz, Günther, Di Marzo, Vincenzo, Offermanns, Stefan
Publicat 2006Text -
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A natural substrate-based fluorescence assay for inhibitor screening on diacylglycerol lipase α per van der Wel, Tom, Janssen, Freek J., Baggelaar, Marc P., Deng, Hui, den Dulk, Hans, Overkleeft, Herman S., van der Stelt, Mario
Publicat 2015Text -
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Development of a Multiplexed Activity-Based Protein Profiling Assay to Evaluate Activity of Endocannabinoid Hydrolase Inhibitors per Janssen, Antonius P. A., van der Vliet, Daan, Bakker, Alexander T., Jiang, Ming, Grimm, Sebastian H., Campiani, Giuseppe, Butini, Stefania, van der Stelt, Mario
Publicat 2018Text -
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Anandamide acts as an intracellular messenger amplifying Ca(2+) influx via TRPV1 channels per van der Stelt, Mario, Trevisani, Marcello, Vellani, Vittorio, De Petrocellis, Luciano, Schiano Moriello, Aniello, Campi, Barbara, McNaughton, Peter, Geppetti, Piero, Di Marzo, Vincenzo
Publicat 2005Text -
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Anti-neuroinflammatory effects of GPR55 antagonists in LPS-activated primary microglial cells per Saliba, Soraya Wilke, Jauch, Hannah, Gargouri, Brahim, Keil, Albrecht, Hurrle, Thomas, Volz, Nicole, Mohr, Florian, van der Stelt, Mario, Bräse, Stefan, Fiebich, Bernd L.
Publicat 2018Text -
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Structure Kinetics Relationships and Molecular Dynamics Show Crucial Role for Heterocycle Leaving Group in Irreversible Diacylglycerol Lipase Inhibitors per Janssen, Antonius P.A., van Hengst, Jacob M.A., Béquignon, Olivier J.M., Deng, Hui, van Westen, Gerard J.P., van der Stelt, Mario
Publicat 2019Text -
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Evaluation of different drug classes on transient sciatic nerve injury-depressed marble burying in mice per Wilkerson, Jenny L, Curry, Zachary A, Kinlow, Pamela D, Mason, Brittany L, Hsu, Ku-Lung, van der Stelt, Mario, Cravatt, Benjamin F, Lichtman, Aron H
Publicat 2018Text -
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Structure–Activity Relationship Studies of Pyrimidine-4-Carboxamides as Inhibitors of N-Acylphosphatidylethanolamine Phospholipase D per Mock, Elliot D., Kotsogianni, Ioli, Driever, Wouter P. F., Fonseca, Carmen S., Vooijs, Jelle M., den Dulk, Hans, van Boeckel, Constant A. A., van der Stelt, Mario
Publicat 2020Text -
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Development of a Cannabinoid-Based Photoaffinity Probe to Determine the Δ(8/9)-Tetrahydrocannabinol Protein Interaction Landscape in Neuroblastoma Cells per Soethoudt, Marjolein, Alachouzos, Georgios, van Rooden, Eva J., Moya-Garzón, María Dolores, van den Berg, Richard J.B.H.N., Heitman, Laura H., van der Stelt, Mario
Publicat 2018Text -
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An Affinity-Based Probe for the Human Adenosine A(2A) Receptor per Yang, Xue, Michiels, Thomas J. M., de Jong, Coen, Soethoudt, Marjolein, Dekker, Niek, Gordon, Euan, van der Stelt, Mario, Heitman, Laura H., van der Es, Daan, IJzerman, Adriaan P.
Publicat 2018Text -
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Stress-induced modulation of endocannabinoid signaling leads to delayed strengthening of synaptic connectivity in the amygdala per Yasmin, Farhana, Colangeli, Roberto, Morena, Maria, Filipski, Sarah, van der Stelt, Mario, Pittman, Quentin J., Hillard, Cecilia J., Teskey, G. Campbell, McEwen, Bruce S., Hill, Matthew N., Chattarji, Sumantra
Publicat 2020Text -
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Olaparib‐Based Photoaffinity Probes for PARP‐1 Detection in Living Cells per Voorneveld, Jim, Florea, Bogdan I., Bakkum, Thomas, Mendowicz, Rafal J., van der Veer, Miriam S., Gagestein, Berend, van Kasteren, Sander I., van der Stelt, Mario, Overkleeft, Herman S., Filippov, Dmitri V.
Publicat 2020Text -
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Cannabinoid type 1 receptor inverse agonism attenuates dyslipidemia and atherosclerosis in APOE∗3-Leiden.CETP mice per van Eenige, Robin, Ying, Zhixiong, Tambyrajah, Lauren, Pronk, Amanda C.M., Blomberg, Niek, Giera, Martin, Wang, Yanan, Coskun, Tamer, van der Stelt, Mario, Rensen, Patrick C.N., Kooijman, Sander
Publicat 2021Text -
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Chemical Proteomics Reveals Off-Targets of the Anandamide Reuptake Inhibitor WOBE437 per Gagestein, Berend, Stevens, Anna F., Fazio, Domenico, Florea, Bogdan I., van der Wel, Tom, Bakker, Alexander T., Fezza, Filomena, Dulk, Hans den, Overkleeft, Herman S., Maccarrone, Mauro, van der Stelt, Mario
Publicat 2022Text