Výsledky vyhledávání - Xavier Langlois
- Zobrazuji výsledky 1 - 16 z 16
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Pyrido[4,3-<i>e</i>][1,2,4]triazolo[4,3-<i>a</i>]pyrazines as Selective, Brain Penetrant Phosphodiesterase 2 (PDE2) Inhibitors Autor Frederik Rombouts, Gary Tresadern, Peter Buijnsters, Xavier Langlois, Fulgencio Tovar, Thomas Steinbrecher, Greet Vanhoof, Marijke Somers, José-Ignacio Andrés, Andrés A. Trabanco
Vydáno 2015Artigo -
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Peripheral Administration of Tumor Necrosis Factor-Alpha Induces Neuroinflammation and Sickness but Not Depressive-Like Behavior in Mice Autor Steven Biesmans, J Adriaan Bouwknecht, Luc Ver Donck, Xavier Langlois, Paul D. Acton, Patrick De Haes, Nima Davoodi, Theo Meert, Niels Hellings, Rony Nuydens
Vydáno 2015Artigo -
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Pharmacological and pharmacokinetic properties of JNJ‐40411813, a positive allosteric modulator of the mGlu2 receptor Autor Hilde Lavreysen, A. Ahnaou, Wilhelmus Drinkenburg, Xavier Langlois, Claire Mackie, Stefan Pype, Robert Lütjens, Emmanuel Le Poul, Andrés A. Trabanco, José María Cid Nuñez
Vydáno 2014Artigo -
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Structure-Based Design of a Potent, Selective, and Brain Penetrating PDE2 Inhibitor with Demonstrated Target Engagement Autor Peter Buijnsters, Meri De Angelis, Xavier Langlois, Frederik Rombouts, Wendy E. Sanderson, Gary Tresadern, Alison Ritchie, Andrés A. Trabanco, Greet Vanhoof, Yves Van Roosbroeck, José-Ignacio Andrés
Vydáno 2014Artigo -
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Characterization of an orphan G protein-coupled receptor localized in the dorsal root ganglia reveals adenine as a signaling molecule Autor Eckhard Bender, Arjan Buist, Mirek Jurzak, Xavier Langlois, Geert Baggerman, Peter Verhasselt, Martine Ercken, Hongqing Guo, Cindy Wintmolders, Ilse Van den Wyngaert, Irma Van Oers, Liliane Schoofs, Walter Luyten
Vydáno 2002Artigo -
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Systemic Immune Activation Leads to Neuroinflammation and Sickness Behavior in Mice Autor Steven Biesmans, Theo Meert, J Adriaan Bouwknecht, Paul D. Acton, Nima Davoodi, Patrick De Haes, Jacobine Kuijlaars, Xavier Langlois, Liam J. R. Matthews, Luc Ver Donck, Niels Hellings, Rony Nuydens
Vydáno 2013Artigo -
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Preclinical Evaluation of <sup>18</sup>F-JNJ41510417 as a Radioligand for PET Imaging of Phosphodiesterase-10A in the Brain Autor Sofie Celen, Michel Koole, Meri De Angelis, I. SANNEN, Satish K. Chitneni, Jesús Alcázar, Stefanie Dedeurwaerdere, Dieder Moechars, Mark E. Schmidt, Alfons Verbruggen, Xavier Langlois, Koen Van Laere, José Ignacio Andrés, Guy Bormans
Vydáno 2010Artigo -
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Preclinical Evaluation of<sup>18</sup>F-JNJ64349311, a Novel PET Tracer for Tau Imaging Autor Lieven Declercq, Frederik Rombouts, Michel Koole, Katleen Fierens, Jonas Mariën, Xavier Langlois, José Ignacio Andrés, Mark E. Schmidt, Gregor J. Macdonald, Diederik Moechars, Wim Vanduffel, Thomas Tousseyn, Rik Vandenberghe, Koen Van Laere, Alfons Verbruggen, Guy Bormans
Vydáno 2017Artigo -
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Acute wake‐promoting actions of JNJ‐5207852, a novel, diamine‐based H<sub>3</sub> antagonist Autor Ann Barbier, Craig W. Berridge, Christine Dugovic, Aaron D. Laposky, Sandy J. Wilson, Jamin D. Boggs, Leah Aluisio, Brian Lord, Curt Mazur, Cindy M. Pudiak, Xavier Langlois, Wei Xiao, Richard L. Apodaca, Nicholas I. Carruthers, Timothy W. Lovenberg
Vydáno 2004Artigo -
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Common mouse models of tauopathy reflect early but not late human disease Autor Kathrin Wenger, Arthur Viodé, Christoph N. Schlaffner, Patrick van Zalm, Long Cheng, Tammy Dellovade, Xavier Langlois, Anthony W. Bannon, Rui B. Chang, Theresa R. Connors, Derek H. Oakley, Bernhard Y. Renard, Juri Rappsilber, Bradley T. Hyman, Hanno Steen, Judith A. Steen
Vydáno 2023Artigo -
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Preclinical Evaluation of a P2X7 Receptor–Selective Radiotracer: PET Studies in a Rat Model with Local Overexpression of the Human P2X7 Receptor and in Nonhuman Primates Autor Dieter Ory, Sofie Celen, Rik Gijsbers, Chris Van den Haute, Andrey Postnov, Michel Koole, Caroline Vandeputte, José-Ignacio Andrés, Jesús Alcázar, Meri De Angelis, Xavier Langlois, Anindya Bhattacharya, Mark E. Schmidt, Michael A. Letavic, Wim Vanduffel, Koen Van Laere, Alfons Verbruggen, Zeger Debyser, Guy Bormans
Vydáno 2016Artigo -
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Discovery of VU0409551/JNJ-46778212: An mGlu<sub>5</sub> Positive Allosteric Modulator Clinical Candidate Targeting Schizophrenia Autor Susana Conde-Ceide, Carlos M. Martínez‐Viturro, Jesús Alcázar, Pedro M. García-Barrantes, Hilde Lavreysen, Claire Mackie, Paige N. Vinson, Jerri M. Rook, Thomas M. Bridges, J. Scott Daniels, Anton A. H. P. Megens, Xavier Langlois, Wilhelmus Drinkenburg, A. Ahnaou, Colleen M. Niswender, Carrie K. Jones, Gregor J. Macdonald, Thomas Steckler, P. Jeffrey Conn, Shaun R. Stauffer, José M. Bartolomé-Nebreda, Craig W. Lindsley
Vydáno 2015Artigo -
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Landscape of brain myeloid cell transcriptome along the spatiotemporal progression of Alzheimer’s disease reveals distinct sequential responses to Aβ and tau Autor Astrid Wachter, Maya E. Woodbury, Sylvia Lombardo, Aicha Abdourahman, Carolin Wuest, Emily J. McGlame, Timothy Pastika, Joseph A. Tamm, Nandini Romanul, Kiran Yanamandra, Rachel E. Bennett, Gen Lin, Taekyung Kwon, Fan Liao, Corinna Klein, Yelena Y. Grinberg, Methasit Jaisa-aad, Li Huan, Matthew P. Frosch, Markus P. Kummer, Sudeshna Das, Tammy Dellovade, Eric Karran, Xavier Langlois, Janina S. Ried, Alberto Serrano‐Pozo, Robert V. Talanian, Knut Biber, Bradley T. Hyman
Vydáno 2024Artigo
Vyhledávací nástroje:
Související témata
Medicine
Chemistry
Internal medicine
Biology
Biochemistry
Receptor
Neuroscience
Pharmacology
In vivo
Antagonist
Biotechnology
Enzyme
Gene
Psychology
Allosteric modulator
Allosteric regulation
Central nervous system
Disease
Endocrinology
Genetics
Immunology
Inflammation
Microglia
Nuclear medicine
Pathology
Phosphodiesterase
Agonist
Alzheimer's disease
Astrocyte
Cognition