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William R. Pitt
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On the Origins of Enzyme Inhibitor Selectivity and Promiscuity: A Case Study of Protein Kinase Binding to Staurosporine
by
Duangrudee Tanramluk
,
Adrian Schreyer
,
William R. Pitt
,
Tom L. Blundell
Published 2009
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Related Subjects
Allosteric regulation
Binding site
Biochemistry
Chemistry
Cooperative binding
Enzyme
Hydrogen bond
Molecule
Organic chemistry
Plasma protein binding
Protein kinase A
Protein kinase inhibitor
Staurosporine
Stereochemistry
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