תוצאות חיפוש - Tianfeng Xu
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Discovery of Highly Potent and Efficient PROTAC Degraders of Androgen Receptor (AR) by Employing Weak Binding Affinity VHL E3 Ligase Ligands מאת Xin Han, Lijie Zhao, Weiguo Xiang, Chong Qin, Bukeyan Miao, Tianfeng Xu, Mi Wang, Chao‐Yie Yang, Krishnapriya Chinnaswamy, Jeanne A. Stuckey, Shaomeng Wang
יצא לאור 2019Artigo -
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Design, Synthesis, and Bioevaluation of Pyrido[2,3-<i>d</i>]pyrimidin-7-ones as Potent SOS1 Inhibitors מאת Meiying Liu, Guizhen Zhou, Wenhong Su, Yuejiao Gu, Mingshan Gao, Kun Wang, Ruifeng Huo, Yupeng Li, Zehui Zhou, Kaixian Chen, Mingyue Zheng, Sulin Zhang, Tianfeng Xu
יצא לאור 2023Artigo -
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Engineered bioorthogonal POLY-PROTAC nanoparticles for tumour-specific protein degradation and precise cancer therapy מאת Jing Gao, Bo Hou, Qiwen Zhu, Lei Yang, Xingyu Jiang, Zhifeng Zou, Xutong Li, Tianfeng Xu, Mingyue Zheng, Yi‐Hung Chen, Zhiai Xu, Huixiong Xu, Haijun Yu
יצא לאור 2022Artigo -
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Design of the First‐in‐Class, Highly Potent Irreversible Inhibitor Targeting the Menin‐MLL Protein–Protein Interaction מאת Shilin Xu, Angelo Aguilar, Tianfeng Xu, Ke Zheng, Liyue Huang, Jeanne A. Stuckey, Krishnapriya Chinnaswamy, Denzil Bernard, Ester Fernández‐Salas, Liu Liu, Mi Wang, Donna McEachern, Sally Przybranowski, C.L. Foster, Shaomeng Wang
יצא לאור 2017Artigo -
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Discovery of <b>ERD-3111</b> as a Potent and Orally Efficacious Estrogen Receptor PROTAC Degrader with Strong Antitumor Activity מאת Zhixiang Chen, Biao Hu, Rohan Kalyan Rej, Dimin Wu, Ranjan Kumar Acharyya, Mingliang Wang, Tianfeng Xu, Jianfeng Lü, Hoda Metwally, Yu Wang, Donna McEachern, Longchuan Bai, Christina L. Gersch, Meilin Wang, Wenjing Zhang, Qiuxia Li, Bo Wen, Duxin Sun, James M. Rae, Shaomeng Wang
יצא לאור 2023Artigo -
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Discovery of ARD-1676 as a Highly Potent and Orally Efficacious AR PROTAC Degrader with a Broad Activity against AR Mutants for the Treatment of AR + Human Prostate Cancer מאת Weiguo Xiang, Lijie Zhao, Xin Han, Tianfeng Xu, Steven Kregel, Mi Wang, Bukeyan Miao, Chong Qin, Mingliang Wang, Donna McEachern, Jianfeng Lü, Longchuan Bai, Chao‐Yie Yang, Paul D. Kirchhoff, John Takyi‐Williams, Lu Wang, Bo Wen, Duxin Sun, Mark A. Ator, Robert McKean, Arul M. Chinnaiyan, Shaomeng Wang
יצא לאור 2023Artigo
כלי חיפוש:
נושאים קשורים
Chemistry
Biochemistry
Cancer
Cancer research
Gene
Medicine
Pharmacology
Biology
Internal medicine
Androgen receptor
Bioavailability
Enzyme
Genetics
Mutant
Mutation
Prostate cancer
Amphiphile
Benzamide
Bioorthogonal chemistry
Breast cancer
Cell growth
Click chemistry
Combinatorial chemistry
Copolymer
DNA ligase
EGFR inhibitors
Epidermal growth factor receptor
Erlotinib
Estrogen
Estrogen receptor