Որոնման արդյունքները - Swee Y. Sharp
- Ցուցադրվում են 1 - 19 արդյունքները 19
-
1
-
2
-
3
-
4
-
5
Mechanistic Evaluation of the Novel HSP90 Inhibitor NVP-AUY922 in Adult and Pediatric Glioblastoma Nathalie Gaspar, Swee Y. Sharp, Suzanne A. Eccles, Sharon Gowan, Sergey Popov, Chris Jones, Andrew D.J. Pearson, Gilles Vassal, Paul Workman
Հրապարակվել է 2010Artigo -
6
Acquired Resistance to 17-Allylamino-17-Demethoxygeldanamycin (17-AAG, Tanespimycin) in Glioblastoma Cells Nathalie Gaspar, Swee Y. Sharp, Simon Pacey, Chris Jones, Michael I. Walton, Gilles Vassal, Suzanne A. Eccles, Andrew D.J. Pearson, Paul Workman
Հրապարակվել է 2009Artigo -
7
MGMT-Independent Temozolomide Resistance in Pediatric Glioblastoma Cells Associated with a PI3-Kinase–Mediated <i>HOX</i>/Stem Cell Gene Signature Nathalie Gaspar, Lynley V. Marshall, Lara Perryman, Dorine A. Bax, Suzanne E. Little, Marta Viana‐Pereira, Swee Y. Sharp, Gilles Vassal, Andrew D.J. Pearson, Rui Manuel Reis, Darren Hargrave, Paul Workman, Chris Jones
Հրապարակվել է 2010Artigo -
8
Demonstrating In-Cell Target Engagement Using a Pirin Protein Degradation Probe (CCT367766) N. Chessum, Swee Y. Sharp, John Caldwell, Elisa Pasqua, Birgit Wilding, Giampiero Colombano, Ian Collins, Buǧra Özer, Meirion Richards, Martin Rowlands, Mark Stubbs, Rosemary Burke, Craig McAndrew, Paul A. Clarke, Paul Workman, Matthew D. Cheeseman, Keith Jones
Հրապարակվել է 2017Artigo -
9
Structure-Activity Relationships in Purine-Based Inhibitor Binding to HSP90 Isoforms Lisa Wright, Xavier Barril, Brian Dymock, Louisa Sheridan, A.E. Surgenor, Mandy Beswick, Martin J. Drysdale, Adam J. Collier, Andy Massey, Nicholas G. Davies, Alex Fink, Christophe Fromont, Wynne Aherne, Kathy Boxall, Swee Y. Sharp, Paul Workman, Roderick E. Hubbard
Հրապարակվել է 2004Artigo -
10
The Association of CCND1 Overexpression and Cisplatin Resistance in Testicular Germ Cell Tumors and Other Cancers Elodie Noël, Marc Yeste‐Velasco, Xueying Mao, Jackie Perry, Sakunthala C. Kudahetti, Ningfeng Fiona Li, Swee Y. Sharp, Tracy Chaplin, Liyan Xue, Alan McIntyre, Ling Shan, Thomas Powles, R.T.D. Oliver, Bryan D. Young, Janet Shipley, Daniel M. Berney, Simon P. Joel, Yong‐Jie Lu
Հրապարակվել է 2010Artigo -
11
Second-Generation HSP90 Inhibitor Onalespib Blocks mRNA Splicing of Androgen Receptor Variant 7 in Prostate Cancer Cells Roberta Ferraldeschi, Jonathan Welti, Marissa Powers, Wei Yuan, Tomoko Smyth, George Seed, Ruth Riisnaes, Somaieh Hedayat, Hannah Wang, Mateus Crespo, Daniel Nava Rodrigues, Ines Figueiredo, Susana Miranda, Suzanne Carreira, John F. Lyons, Swee Y. Sharp, Stephen R. Plymate, Gerhardt Attard, Nicola G. Wallis, Paul Workman, Johann S. de Bono
Հրապարակվել է 2016Artigo -
12
Gene and Protein Expression Profiling of Human Ovarian Cancer Cells Treated with the Heat Shock Protein 90 Inhibitor 17-Allylamino-17-Demethoxygeldanamycin Alison Maloney, Paul A. Clarke, Søren Naaby‐Hansen, Robert C. Stein, Jens-Oliver Koopman, Akunna Akpan, Alice Yang, Marketa Zvelebil, Rainer Cramer, Lindsay Stimson, Wynne Aherne, Udai Banerji, Ian Judson, Swee Y. Sharp, Marissa Powers, Emmanuel de Billy, Joanne Salmons, Michael I. Walton, A. L. Burlingame, Michael Waterfield, Paul Workman
Հրապարակվել է 2007Artigo -
13
EGFRvIII Deletion Mutations in Pediatric High-Grade Glioma and Response to Targeted Therapy in Pediatric Glioma Cell Lines Dorine A. Bax, Nathalie Gaspar, Suzanne E. Little, Lynley V. Marshall, Lara Perryman, Marie Regairaz, Marta Viana‐Pereira, Raisa Vuononvirta, Swee Y. Sharp, Jorge S. Reis‐Filho, João N. Stávale, Safa Al‐Sarraj, Rui Manuel Reis, Gilles Vassal, Andrew D.J. Pearson, Darren Hargrave, David W. Ellison, Paul Workman, Chris Jones
Հրապարակվել է 2009Artigo -
14
Data from EGFRvIII Deletion Mutations in Pediatric High-Grade Glioma and Response to Targeted Therapy in Pediatric Glioma Cell Lines Dorine A. Bax, Nathalie Gaspar, Suzanne E. Little, Lynley V. Marshall, Lara Perryman, Marie Regairaz, Marta Viana‐Pereira, Raisa Vuononvirta, Swee Y. Sharp, Jorge S. Reis‐Filho, João Norberto Stávale, Safa Al‐Sarraj, Rui Manuel Reis, Gilles Vassal, Andrew D.J. Pearson, Darren Hargrave, David W. Ellison, Paul Workman, Chris Jones
Հրապարակվել է 2023Pré-impressão -
15
<i>In vitro</i> Biological Characterization of a Novel, Synthetic Diaryl Pyrazole Resorcinol Class of Heat Shock Protein 90 Inhibitors Swee Y. Sharp, Kathy Boxall, Martin Rowlands, Chrisostomos Prodromou, S. Mark Roe, Alison Maloney, Marissa Powers, Paul A. Clarke, Gary Box, Sharon Sanderson, Lisa Patterson, Thomas P. Matthews, Kwai-Ming J. Cheung, Karen Ball, Angela Hayes, Florence I. Raynaud, Richard Marais, Laurence H. Pearl, Sue Eccles, Wynne Aherne, Edward McDonald, Paul Workman
Հրապարակվել է 2007Artigo -
16
HSF1 Pathway Inhibitor Clinical Candidate (CCT361814/NXP800) Developed from a Phenotypic Screen as a Potential Treatment for Refractory Ovarian Cancer and Other Malignancies Elisa Pasqua, Swee Y. Sharp, N. Chessum, Angela Hayes, Loredana Pellegrino, Michael Tucker, Asadh Miah, Birgit Wilding, Lindsay E. Evans, Carl S. Rye, N. Yi Mok, Manjuan Liu, Alan T. Henley, Sharon Gowan, Emmanuel de Billy, Robert te Poele, Marissa Powers, Suzanne A. Eccles, Paul A. Clarke, Florence I. Raynaud, Paul Workman, Keith Jones, Matthew D. Cheeseman
Հրապարակվել է 2023Artigo -
17
Discovery of a Chemical Probe Bisamide (CCT251236): An Orally Bioavailable Efficacious Pirin Ligand from a Heat Shock Transcription Factor 1 (HSF1) Phenotypic Screen Matthew D. Cheeseman, N. Chessum, Carl S. Rye, Elisa Pasqua, Michael Tucker, Birgit Wilding, Lindsay E. Evans, Susan Lepri, Meirion Richards, Swee Y. Sharp, Salyha Ali, Martin Rowlands, Lisa O’Fee, Asadh Miah, Angela Hayes, Alan T. Henley, Marissa Powers, Robert te Poele, Emmanuel de Billy, Loredana Pellegrino, Florence I. Raynaud, Rosemary Burke, Rob L. M. van Montfort, Suzanne A. Eccles, Paul Workman, Keith Jones
Հրապարակվել է 2016Artigo -
18
Inhibition of the heat shock protein 90 molecular chaperone <i>in vitro</i> and <i>in vivo</i> by novel, synthetic, potent resorcinylic pyrazole/isoxazole amide analogues Swee Y. Sharp, Chrisostomos Prodromou, Kathy Boxall, Marissa Powers, Joanna L. Holmes, Gary Box, Thomas P. Matthews, Kwai-Ming J. Cheung, Andrew Kalusa, Karen James, Angela Hayes, Anthea Hardcastle, Brian Dymock, Paul A. Brough, Xavier Barril, Julie E. Cansfield, Lisa Wright, A.E. Surgenor, Nicolas Foloppe, Roderick E. Hubbard, Wynne Aherne, Laurence H. Pearl, Keith Jones, Edward McDonald, Florence I. Raynaud, Sue Eccles, Martin J. Drysdale, Paul Workman
Հրապարակվել է 2007Artigo -
19
NVP-AUY922: A Novel Heat Shock Protein 90 Inhibitor Active against Xenograft Tumor Growth, Angiogenesis, and Metastasis Suzanne A. Eccles, Andy Massey, Florence I. Raynaud, Swee Y. Sharp, Gary Box, Melanie Valenti, Lisa Patterson, Alexis de Haven Brandon, Sharon Gowan, Frances Boxall, Wynne Aherne, Martin Rowlands, Angela Hayes, Vanessa Martins, Frederique Urban, Kathy Boxall, Chrisostomos Prodromou, Laurence H. Pearl, Karen James, Thomas P. Matthews, Kwai-Ming J. Cheung, Andrew Kalusa, Keith Jones, Edward McDonald, Xavier Barril, Paul A. Brough, Julie E. Cansfield, Brian Dymock, Martin J. Drysdale, Harry Finch, Rob Howes, Roderick E. Hubbard, Alan Surgenor, Paul Webb, Mike Wood, Lisa Wright, Paul Workman
Հրապարակվել է 2008Artigo
Որոնման գործիքներ:
Առնչվող խորագիր
Biology
Gene
Biochemistry
Cancer research
Chemistry
Heat shock protein
Genetics
Hsp90
Molecular biology
Cancer
Hsp90 inhibitor
Medicine
Cell culture
Pharmacology
Apoptosis
Internal medicine
Chemotherapy
Cisplatin
Gene expression
Glioma
Hsp70
Ovarian cancer
PI3K/AKT/mTOR pathway
Signal transduction
Cell biology
Cell growth
Clonogenic assay
Computational biology
Enzyme
Epidermal growth factor receptor