نتائج البحث - Stefania Colarusso
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Discovery of (7<i>R</i>)-14-Cyclohexyl-7-{[2-(dimethylamino)ethyl](methyl) amino}-7,8-dihydro-6<i>H</i>-indolo[1,2-<i>e</i>][1,5]benzoxazocine-11-carboxylic Acid (MK-3281), a Poten... حسب Frank Narjes, Benedetta Crescenzi, Marco Ferrara, Jörg Habermann, Stefania Colarusso, Marı́a del Rosario Rico Ferreira, Ian Stansfield, Angela Mackay, Immacolata Conte, Caterina Ercolani, Simone Zaramella, Maria-Cecilia Palumbi, Philip Meuleman, Geert Leroux‐Roels, Claudio Giuliano, Fabrizio Fiore, Stefania Di Marco, Paola Baiocco, Uwe Koch, Giovanni Migliaccio, Sergio Altamura, Ralph Laufer, Raffaele De Francesco, Michael Rowley
منشور في 2010Artigo
أدوات البحث:
موضوعات ذات صلة
Biochemistry
Biology
Chemistry
Enzyme
Hepatitis C virus
Virology
Virus
Allosteric regulation
Drug discovery
Gene
Genetics
Genome
Human immunodeficiency virus (HIV)
In vitro
In vivo
Lead compound
NS2-3 protease
NS3
Potency
Protease
Stereochemistry
Structure–activity relationship
Subgenomic mRNA
Viremia