Ngā hua rapu - Stefania Colarusso
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Discovery of (7<i>R</i>)-14-Cyclohexyl-7-{[2-(dimethylamino)ethyl](methyl) amino}-7,8-dihydro-6<i>H</i>-indolo[1,2-<i>e</i>][1,5]benzoxazocine-11-carboxylic Acid (MK-3281), a Poten... mā Frank Narjes, Benedetta Crescenzi, Marco Ferrara, Jörg Habermann, Stefania Colarusso, Marı́a del Rosario Rico Ferreira, Ian Stansfield, Angela Mackay, Immacolata Conte, Caterina Ercolani, Simone Zaramella, Maria-Cecilia Palumbi, Philip Meuleman, Geert Leroux‐Roels, Claudio Giuliano, Fabrizio Fiore, Stefania Di Marco, Paola Baiocco, Uwe Koch, Giovanni Migliaccio, Sergio Altamura, Ralph Laufer, Raffaele De Francesco, Michael Rowley
I whakaputaina 2010Artigo
Ngā utauta rapu:
Ngā marau whai pānga
Biochemistry
Biology
Chemistry
Enzyme
Hepatitis C virus
Virology
Virus
Allosteric regulation
Drug discovery
Gene
Genetics
Genome
Human immunodeficiency virus (HIV)
In vitro
In vivo
Lead compound
NS2-3 protease
NS3
Potency
Protease
Stereochemistry
Structure–activity relationship
Subgenomic mRNA
Viremia