Resultats de la cerca - Simone Brogi
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A Repurposing Approach for Uncovering the Anti-Tubercular Activity of FDA-Approved Drugs with Potential Multi-Targeting Profiles per Basem Battah, Giulia Chemi, Stefania Butini, Giuseppe Campiani, Simone Brogi, Giovanni Delogu, Sandra Gemma
Publicat 2019Artigo -
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Covalent Reversible Inhibitors of Cysteine Proteases Containing the Nitrile Warhead: Recent Advancement in the Field of Viral and Parasitic Diseases per Simone Brogi, Roberta Ibba, Sara Rossi, Stefania Butini, Vincenzo Calderone, Sandra Gemma, Giuseppe Campiani
Publicat 2022Revisão -
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Anti‐inflammatory and antiviral roles of hydrogen sulfide: Rationale for considering H<sub>2</sub>S donors in COVID‐19 therapy per Valentina Citi, Alma Martelli, Vincenzo Brancaleone, Simone Brogi, Gabriel Gojon, Rosangela Montanaro, Guillermo Morales, Lara Testai, Vincenzo Calderone
Publicat 2020Revisão -
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Discovery and Cardioprotective Effects of the First Non-Peptide Agonists of the G Protein-Coupled Prokineticin Receptor-1 per Adeline Gasser, Simone Brogi, Kyoji Urayama, Toshishide Nishi, Hitoshi Kurose, Andrea Tafi, Nigel Ribeiro, Laurent Désaubry, Canan G. Nebigil
Publicat 2015Artigo -
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New cinnamid and rosmarinic acid derived compounds biosynthesized in <i>Escherichia coli</i> as <i>Leishmania amazonensis</i> arginase inhibitors per Júlio Abel Alfredo dos Santos Simone Come, Yibin Zhuang, Tianzhen Li, Simone Brogi, Sandra Gemma, Tao Liu, Edson Roberto da Silva
Publicat 2020Pré-impressão -
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In Vitro and In Silico Analyses of New Cinnamid and Rosmarinic Acid-Derived Compounds Biosynthesized in Escherichia coli as Leishmania amazonensis Arginase Inhibitors per Júlio Abel Alfredo dos Santos Simone Come, Yibin Zhuang, Tianzhen Li, Simone Brogi, Sandra Gemma, Tao Liu, Edson Roberto da Silva
Publicat 2022Artigo -
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Identification of Novel 3-Hydroxy-pyran-4-One Derivatives as Potent HIV-1 Integrase Inhibitors Using in silico Structure-Based Combinatorial Library Design Approach per Hajar Sirous, Giulia Chemi, Sandra Gemma, Stefania Butini, Zeger Debyser, Frauke Christ, Lotfollah Saghaie, Simone Brogi, Afshin Fassihi, Giuseppe Campiani, Margherita Brindisi
Publicat 2019Artigo -
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Structure-based discovery of the first non-covalent inhibitors of Leishmania major tryparedoxin peroxidase by high throughput docking per Margherita Brindisi, Simone Brogi, Nicola Relitti, Alessandra Vallone, Stefania Butini, Sandra Gemma, Ettore Novellino, Gianni Colotti, Gabriella Angiulli, Francesco Di Chiaro, Annarita Fiorillo, Andrea Ilari, Giuseppe Campiani
Publicat 2015Artigo -
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Multitarget compounds bearing tacrine- and donepezil-like structural and functional motifs for the potential treatment of Alzheimer's disease per Lhassane Ismaïli, Bernard Refouvelet, Mohamed Benchekroun, Simone Brogi, Margherita Brindisi, Sandra Gemma, Giuseppe Campiani, Slavica Filipić, Danica Agbaba, Gerard Esteban, Mercedes Unzeta, Katarina Nikolić, Stefania Butini, José Marco‐Contelles
Publicat 2016Revisão -
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Structure-activity relationships study of isothiocyanates for H2S releasing properties: 3-Pyridyl-isothiocyanate as a new promising cardioprotective agent per Valentina Citi, Angela Corvino, Ferdinando Fiorino, Francesco Frecentese, Elisa Magli, Elisa Perissutti, Vincenzo Santagada, Simone Brogi, Lorenzo Flori, Era Gorica, Lara Testai, Alma Martelli, Vincenzo Calderone, Giuseppe Caliendo, Beatrice Severino
Publicat 2020Revisão -
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Disease‐Modifying Anti‐Alzheimer's Drugs: Inhibitors of Human Cholinesterases Interfering with <i>β</i>‐Amyloid Aggregation per Simone Brogi, Stefania Butini, Samuele Maramai, Raffaella Colombo, Laura Verga, Cristina Lanni, Ersilia De Lorenzi, Stefania Lamponi, Maria Grazia Andreassi, Manuela Bartolini, Vincenza Andrisano, Ettore Novellino, Giuseppe Campiani, Margherita Brindisi, Sandra Gemma
Publicat 2014Artigo -
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Cinnamides Target Leishmania amazonensis Arginase Selectively per Edson Roberto da Silva, Júlio Abel Alfredo dos Santos Simone Come, Simone Brogi, Vincenzo Calderone, Giulia Chemi, Giuseppe Campiani, Trícia Maria Ferrreira de Sousa Oliveira, Thanh‐Nhat Pham, Marc Pudlo, C. Girard, Claudia do Carmo Maquiaveli
Publicat 2020Artigo
Eines de cerca:
Matèries relacionades
Biochemistry
Chemistry
Biology
Medicine
Pharmacology
Gene
In vitro
Enzyme
Computational biology
Internal medicine
Organic chemistry
Stereochemistry
Antioxidant
Computer science
Genetics
Receptor
Combinatorial chemistry
Disease
Docking (animal)
Hydrogen sulfide
In silico
Leishmania
Neuroscience
Nursing
Parasite hosting
Pathology
Sulfur
World Wide Web
Amino acid
Apoptosis