Suchergebnisse - Satyawan Jadhav
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1
Statins and osteoporosis: new role for old drugs von Satyawan Jadhav, Girish Kumar Jain
Veröffentlicht 2005Revisão -
2
Synthesis and Evaluation of a Series of Heterobiarylamides That Are Centrally Penetrant Metabotropic Glutamate Receptor 4 (mGluR4) Positive Allosteric Modulators (PAMs) von Darren W. Engers, Colleen M. Niswender, C. David Weaver, Satyawan Jadhav, Usha N. Menon, Rocio Zamorano, P. Jeffrey Conn, Craig W. Lindsley, Corey R. Hopkins
Veröffentlicht 2009Artigo -
3
Design, Synthesis, and Biological Evaluation of Halogenated <i>N</i>-(2-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)ethyl)benzamides: Discovery of an Isoform-Selective Small M... von Robert R. Lavieri, Sarah Scott, Paige E. Selvy, Kwang‐Ho Kim, Satyawan Jadhav, Ryan D. Morrison, J. Scott Daniels, H. Alex Brown, Craig W. Lindsley
Veröffentlicht 2010Artigo -
4
Discovery of the First Highly M5-Preferring Muscarinic Acetylcholine Receptor Ligand, an M5 Positive Allosteric Modulator Derived from a Series of 5-Trifluoromethoxy <i>N</i>-Benzy... von Thomas M. Bridges, Joy E. Marlo, Colleen M. Niswender, Carrie K. Jones, Satyawan Jadhav, Patrick R. Gentry, Hyekyung C. Plumley, C. David Weaver, P. Jeffrey Conn, Craig W. Lindsley
Veröffentlicht 2009Artigo -
5
Centrally Active Allosteric Potentiators of the M<sub>4</sub> Muscarinic Acetylcholine Receptor Reverse Amphetamine-Induced Hyperlocomotor Activity in Rats von Ashley E. Brady, Carrie K. Jones, Thomas M. Bridges, J. Phillip Kennedy, Analisa D. Thompson, J.U. Heiman, Micah L. Breininger, Patrick R. Gentry, Huiyong Yin, Satyawan Jadhav, Jana K. Shirey, P. Jeffrey Conn, Craig W. Lindsley
Veröffentlicht 2008Artigo -
6
Discovery and Characterization of Novel Subtype-Selective Allosteric Agonists for the Investigation of M<sub>1</sub> Receptor Function in the Central Nervous System von Evan P. Lebois, Thomas M. Bridges, L. Michelle Lewis, Eric S. Dawson, Alexander S. Kane, Zixiu Xiang, Satyawan Jadhav, Huiyong Yin, J. Phillip Kennedy, Jens Meiler, Colleen M. Niswender, Carrie K. Jones, P. Jeffrey Conn, C. David Weaver, Craig W. Lindsley
Veröffentlicht 2009Artigo -
7
A Novel Selective Muscarinic Acetylcholine Receptor Subtype 1 Antagonist Reduces Seizures without Impairing Hippocampus-Dependent Learning von Douglas J. Sheffler, Richard D. Williams, Thomas M. Bridges, Zixiu Xiang, Alexander S. Kane, Nellie Byun, Satyawan Jadhav, Mathew M. Mock, Fang Zheng, L. Michelle Lewis, Carrie K. Jones, Colleen M. Niswender, Charles D. Weaver, Craig W. Lindsley, P. Jeffrey Conn
Veröffentlicht 2009Artigo -
8
The Metabotropic Glutamate Receptor 4-Positive Allosteric Modulator VU0364770 Produces Efficacy Alone and in Combination with l-DOPA or an Adenosine 2A Antagonist in Preclinical Ro... von Carrie K. Jones, Michael Bubser, Analisa D. Thompson, Jonathan W. Dickerson, N. Turle-Lorenzo, Marianne Amalric, Anna L. Blobaum, Thomas M. Bridges, Ryan D. Morrison, Satyawan Jadhav, Darren W. Engers, Kimberly Italiano, Jacob Bode, J. Scott Daniels, Craig W. Lindsley, Corey R. Hopkins, P. Jeffrey Conn, Colleen M. Niswender
Veröffentlicht 2011Artigo -
9
Discovery, Synthesis, and Structure–Activity Relationship Development of a Series of <i>N</i>-4-(2,5-Dioxopyrrolidin-1-yl)phenylpicolinamides (VU0400195, ML182): Characterization o... von Carrie K. Jones, Darren W. Engers, Analisa D. Thompson, Julie R. Field, Anna L. Blobaum, Stacey R. Lindsley, Ya Zhou, Rocco D. Gogliotti, Satyawan Jadhav, Rocio Zamorano, James W. Bogenpohl, Yoland Smith, Ryan D. Morrison, J. Scott Daniels, C. David Weaver, P. Jeffrey Conn, Craig W. Lindsley, Colleen M. Niswender, Corey R. Hopkins
Veröffentlicht 2011Artigo -
10
A Selective Allosteric Potentiator of the M<sub>1</sub>Muscarinic Acetylcholine Receptor Increases Activity of Medial Prefrontal Cortical Neurons and Restores Impairments in Revers... von Jana K. Shirey, Ashley E. Brady, Paulianda J. Jones, Albert A. Davis, Thomas M. Bridges, J. Phillip Kennedy, Satyawan Jadhav, Usha N. Menon, Zixiu Xiang, Mona L. Watson, Edward P. Christian, James Doherty, Michael C. Quirk, Dean H. Snyder, James J. Lah, Allan I. Levey, Michelle M. Nicolle, Craig W. Lindsley, P. Jeffrey Conn
Veröffentlicht 2009Artigo -
11
Discovery of Novel Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5 Reveals Chemical and Functional Diversity and In Vivo Activity in Rat Behavioral Models of Anx... von Alice L. Rodriguez, Mark D. Grier, Carrie K. Jones, Elizabeth J. Herman, Alexander S. Kane, Randy L. Smith, Richard D. Williams, Ya Zhou, Joy E. Marlo, Emily Days, Tasha N. Blatt, Satyawan Jadhav, Usha N. Menon, Paige N. Vinson, Jerri M. Rook, Shaun R. Stauffer, Colleen M. Niswender, Craig W. Lindsley, C. David Weaver, P. Jeffrey Conn
Veröffentlicht 2010Artigo -
12
<i>N</i>-Aryl Piperazine Metabotropic Glutamate Receptor 5 Positive Allosteric Modulators Possess Efficacy in Preclinical Models of NMDA Hypofunction and Cognitive Enhancement von Karen J. Gregory, Elizabeth J. Herman, Amy J. Ramsey, Alexis S. Hammond, Nellie Byun, Shaun R. Stauffer, Jason Manka, Satyawan Jadhav, Thomas M. Bridges, C. David Weaver, Colleen M. Niswender, Thomas Steckler, Wilhelmus Drinkenburg, A. Ahnaou, Hilde Lavreysen, Gregor J. Macdonald, José M. Bartolomé, Claire Mackie, Brian Hrupka, Marc G. Caron, Tanya L. Daigle, Craig W. Lindsley, P. Jeffrey Conn, Carrie K. Jones
Veröffentlicht 2013Artigo
Suchwerkzeuge:
Ähnliche Schlagworte
Chemistry
Biochemistry
Biology
Receptor
Allosteric modulator
Allosteric regulation
Pharmacology
Neuroscience
Medicine
Stereochemistry
Acetylcholine
Glutamate receptor
In vitro
Metabotropic glutamate receptor
Muscarinic acetylcholine receptor
Agonist
Metabotropic glutamate receptor 5
Muscarinic acetylcholine receptor M1
Antagonist
Dopamine
Endocrinology
Enzyme
Genetics
Internal medicine
Metabotropic glutamate receptor 2
Metabotropic glutamate receptor 4
Metabotropic receptor
Muscarinic acetylcholine receptor M2
Muscarinic acetylcholine receptor M3
Potentiator