Search Results - Satoki Doi
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Broad Antiretroviral Activity and Resistance Profile of the Novel Human Immunodeficiency Virus Integrase Inhibitor Elvitegravir (JTK-303/GS-9137) by Kazuya Shimura, Eiichi Kodama, Yasuko Sakagami, Yumi Matsuzaki, Wataru Watanabe, Kazunobu Yamataka, Yasuo Watanabe, Yoshitsugu Ohata, Satoki Doi, Motohide Sato, Mitsuki Kano, Satoru Ikeda, Masao Matsuoka
Published 2007Artigo -
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SAR Exploration Guided by LE and Fsp<sup>3</sup>: Discovery of a Selective and Orally Efficacious RORγ Inhibitor by Kazuyuki Hirata, Masayuki Kotoku, Noriyoshi Seki, Takaki Maeba, Katsuya Maeda, Shintaro Hirashima, Takayuki Sakai, Shingo Obika, Akimi Hori, Yasunori Hase, Takayuki Yamaguchi, Yoshiaki Katsuda, Takahiro Hata, Naoki Miyagawa, Kojo Arita, Yukihiro Nomura, Kota Asahina, Yusuke Aratsu, Masafumi Kamada, Tsuyoshi Adachi, Masato Noguchi, Satoki Doi, Paul D. Crowe, Erin K. Bradley, Ruo Steensma, Hai‐Yan Tao, Morgan Fenn, Robert E. Babine, Xiaolin Li, Scott M. Thacher, Hiromasa Hashimoto, Makoto Shiozaki
Published 2015Artigo
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Antiretroviral therapy
Biochemistry
Biology
Chemistry
Combinatorial chemistry
Drug discovery
Drug resistance
Elvitegravir
Gene
Genetics
Human immunodeficiency virus (HIV)
In vitro
Integrase
Integrase inhibitor
Internal medicine
Ligand (biochemistry)
Medicine
Metabolic stability
Mutation
Oral administration
Orally active
Pharmacology
Receptor
Viral load
Viral replication
Virology
Virus