Hakutulokset - Roberto Parise‐Filho
- Näytetään 1 - 16 yhteensä 16 tuloksesta
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Multi-Spectroscopic and Theoretical Analysis on the Interaction between Human Serum Albumin and a Capsaicin Derivative—RPF101 Tekijä Otávio Augusto Chaves, Maurício T. Tavares, Micael Rodrigues Cunha, Roberto Parise‐Filho, Carlos Maurício R. Sant’Anna, José Carlos Netto‐Ferreira
Julkaistu 2018Artigo -
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Natural product inspired optimization of a selective TRPV6 calcium channel inhibitor Tekijä Micael Rodrigues Cunha, Rajesh Bhardwaj, Aline Lucie Carrel, Sonja Lindinger, Christoph Romanin, Roberto Parise‐Filho, Matthias A. Hediger, Jean‐Louis Reymond
Julkaistu 2020Artigo -
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Enhancing venetoclax efficacy in leukemia through association with HDAC inhibitors Tekijä Jorge Antonio Elias Godoy Carlos, Maurício T. Tavares, Keli Lima, Larissa Costa de Almeida, Karoline B. Waitman, Letícia V. Costa‐Lotufo, Roberto Parise‐Filho, João Agostinho Machado‐Neto
Julkaistu 2025Artigo -
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Hybrid histone deacetylase-kinase inhibitor potentiates venetoclax-induced cell death in chronic lymphocytic leukemia Tekijä Anali M. B. Garnique, Jorge Antonio Elias Godoy Carlos, Natália Sudan Parducci, Maurício T. Tavares, Karoline B. Waitman, Keli Lima, Letícia V. Costa‐Lotufo, Roberto Parise‐Filho, João Agostinho Machado‐Neto
Julkaistu 2025Carta -
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Synthesis and crystal structure of a new anticancer candidate: RPF151 Tekijä Maurício T. Tavares, Mariana C. F. C. B. Damião, Adilson Ferreira, Cecília M. P. Rodrigues, José Alexandre Marzagão Barbuto, Ricardo Azevedo, Paulo Luiz de-Sá-Júnior, Roberto Parise‐Filho, Fábio Furlan Ferreira
Julkaistu 2014Artigo -
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Another Reason for Using Caffeine in Dermocosmetics: Sunscreen Adjuvant Tekijä Catarina Rosado, Viviane Kaori Tokunaga, Rafael Sauce, Camila Areias de Oliveira, Fernanda Daud Sarruf, Roberto Parise‐Filho, Elisabete Muchagato Maurício, Tânia Santos de Almeida, Maria Valéria Robles Velasco, André Rolim Baby
Julkaistu 2019Artigo -
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Using a fragment-based approach to identify novel chemical scaffolds targeting the dihydrofolate reductase (DHFR) from <i>Mycobacterium tuberculosis</i> Tekijä João Augusto Ribeiro, Alexander Hammer, Gerardo Andrés Libreros Zúñiga, S.M. Chavez-Pacheco, Petros A. Tyrakis, Gabriel S. de Oliveira, Timothy Kirkman, Jamal El Bakali, Silvana A. Rocco, Maurício L. Sforça, Roberto Parise‐Filho, Anthony G. Coyne, Tom L. Blundell, Chris Abell, M.V.B. Dias
Julkaistu 2020Pré-impressão -
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Using a Fragment-Based Approach to Identify Alternative Chemical Scaffolds Targeting Dihydrofolate Reductase from <i>Mycobacterium tuberculosis</i> Tekijä João Augusto Ribeiro, Alexander Hammer, Gerardo Andrés Libreros-Zúñiga, S.M. Chavez-Pacheco, Petros A. Tyrakis, Gabriel S. de Oliveira, Timothy Kirkman, Jamal El Bakali, Silvana A. Rocco, Maurício L. Sforça, Roberto Parise‐Filho, Anthony G. Coyne, Tom L. Blundell, Chris Abell, M.V.B. Dias
Julkaistu 2020Artigo -
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Dona Flor and her two husbands: Discovery of novel HDAC6/AKT2 inhibitors for myeloid cancer treatment Tekijä Karoline B. Waitman, Holli‐Joi Martin, Jorge Antonio Elias Godoy Carlos, Rodolpho C. Braga, V. Souza, Cleber C. Melo‐Filho, Sebastian Hilscher, Mônica F. Z. J. Toledo, Maurício T. Tavares, Letícia V. Costa‐Lotufo, João Agostinho Machado‐Neto, Mike Schutkowski, Wolfgang Sippl, Thales Kronenberger, Vinícius M. Alves, Roberto Parise‐Filho, Eugene Muratov
Julkaistu 2024Pré-impressão -
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Cytotoxic effects of dillapiole on MDA-MB-231 cells involve the induction of apoptosis through the mitochondrial pathway by inducing an oxidative stress while altering the cytoskel... Tekijä Adilson Kleber Ferreira, Paulo Luiz de-Sá-Júnior, Kerly Fernanda Mesquita Pasqualoto, Ricardo Azevedo, Diana Aparecida Dias Câmara, André Santos Costa, Carlos R. Figueiredo, Alisson L. Matsuo, Mariana H. Massaoka, Aline Vivian Vatti Auada, Ivo Lebrun, Mariana Celestina Frojuello Costa Bernstorff Damião, Maurício T. Tavares, Fátima Maria Motter Magri, Irina Kerkis, Roberto Parise‐Filho
Julkaistu 2013Artigo -
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1,3-Diphenylureido hydroxamate as a promising scaffold for generation of potent antimalarial histone deacetylase inhibitors Tekijä Maurício T. Tavares, Arne Krüger, Sun Yan, Karoline B. Waitman, Vinícius M. Gomes, Daffiny Sumam de Oliveira, Franciarli Paz, Sebastian Hilscher, Mike Schutkowski, Wolfgang Sippl, Claudia Ruiz, Mônica F. Z. J. Toledo, Neuza Mariko Aymoto Hassimotto, João Agostinho Machado‐Neto, Antti Poso, Michael D. Cameron, Thomas D. Bannister, Giuseppe Palmisano, Carsten Wrenger, Thales Kronenberger, Roberto Parise‐Filho
Julkaistu 2023Artigo
Työkalut:
Liittyvät aiheet
Medicine
Biology
Biochemistry
Chemistry
Pharmacology
Cancer
Pathology
Apoptosis
Computational biology
Dihydrofolate reductase
Enzyme
Gene
Genetics
Histone
Histone deacetylase
Immunology
In vitro
Internal medicine
Mycobacterium tuberculosis
Organic chemistry
Tuberculosis
Cancer cell
Cancer research
Chronic lymphocytic leukemia
Crystallography
Cytotoxic T cell
Drug discovery
Histone deacetylase inhibitor
Leukemia
Molecule