खोज परिणाम - Robaa, Dina
- प्रदर्शित 1 - 19 परिणाम 19
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Binding Free Energy (BFE) Calculations and Quantitative Structure–Activity Relationship (QSAR) Analysis of Schistosoma mansoni Histone Deacetylase 8 (smHDAC8) Inhibitors द्वारा Simoben, Conrad V., Ghazy, Ehab, Zeyen, Patrik, Darwish, Salma, Schmidt, Matthias, Romier, Christophe, Robaa, Dina, Sippl, Wolfgang
प्रकाशित 2021मूलपाठ -
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Docking, Binding Free Energy Calculations and In Vitro Characterization of Pyrazine Linked 2-Aminobenzamides as Novel Class I Histone Deacetylase (HDAC) Inhibitors द्वारा Bülbül, Emre F., Melesina, Jelena, Ibrahim, Hany S., Abdelsalam, Mohamed, Vecchio, Anita, Robaa, Dina, Zessin, Matthes, Schutkowski, Mike, Sippl, Wolfgang
प्रकाशित 2022मूलपाठ -
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HaloTag‐Targeted Sirtuin‐Rearranging Ligand (SirReal) for the Development of Proteolysis‐Targeting Chimeras (PROTACs) against the Lysine Deacetylase Sirtuin 2 (Sirt2) द्वारा Schiedel, Matthias, Lehotzky, Attila, Szunyogh, Sandor, Oláh, Judit, Hammelmann, Sören, Wössner, Nathalie, Robaa, Dina, Einsle, Oliver, Sippl, Wolfgang, Ovádi, Judit, Jung, Manfred
प्रकाशित 2020मूलपाठ -
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Structure–Activity Relationship of Anti-Mycobacterium abscessus Piperidine-4-carboxamides, a New Class of NBTI DNA Gyrase Inhibitors द्वारा Beuchel, Andreas, Robaa, Dina, Negatu, Dereje A., Madani, Abdeldjalil, Alvarez, Nadine, Zimmerman, Matthew D., Richter, Adrian, Mann, Lea, Hoenke, Sophie, Csuk, René, Dick, Thomas, Imming, Peter
प्रकाशित 2022मूलपाठ -
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A Novel Class of Schistosoma mansoni Histone Deacetylase 8 (HDAC8) Inhibitors Identified by Structure-Based Virtual Screening and In Vitro Testing द्वारा Simoben, Conrad V., Robaa, Dina, Chakrabarti, Alokta, Schmidtkunz, Karin, Marek, Martin, Lancelot, Julien, Kannan, Srinivasaraghavan, Melesina, Jelena, Shaik, Tajith B., Pierce, Raymond J., Romier, Christophe, Jung, Manfred, Sippl, Wolfgang
प्रकाशित 2018मूलपाठ -
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Design, Synthesis and Biological Characterization of Histone Deacetylase 8 (HDAC8) Proteolysis Targeting Chimeras (PROTACs) with Anti-Neuroblastoma Activity द्वारा Darwish, Salma, Ghazy, Ehab, Heimburg, Tino, Herp, Daniel, Zeyen, Patrik, Salem-Altintas, Rabia, Ridinger, Johannes, Robaa, Dina, Schmidtkunz, Karin, Erdmann, Frank, Schmidt, Matthias, Romier, Christophe, Jung, Manfred, Oehme, Ina, Sippl, Wolfgang
प्रकाशित 2022मूलपाठ -
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Preclinical Evaluation of Benzazepine-Based PET Radioligands (R)- and (S)-(11)C-Me-NB1 Reveals Distinct Enantiomeric Binding Patterns and a Tightrope Walk Between GluN2B- and σ(1)-... द्वारा Haider, Ahmed, Herde, Adrienne Müller, Krämer, Stefanie D., Varisco, Jasmine, Keller, Claudia, Frauenknecht, Katrin, Auberson, Yves P., Temme, Louisa, Robaa, Dina, Sippl, Wolfgang, Schibli, Roger, Wünsch, Bernhard, Mu, Linjing, Ametamey, Simon M.
प्रकाशित 2019मूलपाठ -
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Synthesis and Biological Investigation of Phenothiazine-Based Benzhydroxamic Acids as Selective Histone Deacetylase 6 (HDAC6) Inhibitors द्वारा Vögerl, Katharina, Ong, Nghia, Senger, Johanna, Herp, Daniel, Schmidtkunz, Karin, Marek, Martin, Müller, Martin, Bartel, Karin, Shaik, Tajith B., Porter, Nicholas J., Robaa, Dina, Christianson, David W., Romier, Christophe, Sippl, Wolfgang, Jung, Manfred, Bracher, Franz
प्रकाशित 2019मूलपाठ -
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Structure-Based Design, Docking and Binding Free Energy Calculations of A366 Derivatives as Spindlin1 Inhibitors द्वारा Luise, Chiara, Robaa, Dina, Regenass, Pierre, Maurer, David, Ostrovskyi, Dmytro, Seifert, Ludwig, Bacher, Johannes, Burgahn, Teresa, Wagner, Tobias, Seitz, Johannes, Greschik, Holger, Park, Kwang-Su, Xiong, Yan, Jin, Jian, Schüle, Roland, Breit, Bernhard, Jung, Manfred, Sippl, Wolfgang
प्रकाशित 2021मूलपाठ -
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Identification of Histone Deacetylase 10 (HDAC10) Inhibitors that Modulate Autophagy in Transformed Cells द्वारा Zeyen, Patrik, Zeyn, Yanira, Herp, Daniel, Mahmoudi, Fereshteh, Yesiloglu, Talha Z., Erdmann, Frank, Schmidt, Matthias, Robaa, Dina, Romier, Christophe, Ridinger, Johannes, Herbst-Gervasoni, Corey J., Christianson, David W., Oehme, Ina, Jung, Manfred, Krämer, Oliver H., Sippl, Wolfgang
प्रकाशित 2022मूलपाठ -
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Synthesis, Molecular Docking and Biological Characterization of Pyrazine Linked 2-Aminobenzamides as New Class I Selective Histone Deacetylase (HDAC) Inhibitors with Anti-Leukemic... द्वारा Ibrahim, Hany S., Abdelsalam, Mohamed, Zeyn, Yanira, Zessin, Matthes, Mustafa, Al-Hassan M., Fischer, Marten A., Zeyen, Patrik, Sun, Ping, Bülbül, Emre F., Vecchio, Anita, Erdmann, Frank, Schmidt, Matthias, Robaa, Dina, Barinka, Cyril, Romier, Christophe, Schutkowski, Mike, Krämer, Oliver H., Sippl, Wolfgang
प्रकाशित 2021मूलपाठ -
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First Fluorescent Acetylspermidine Deacetylation Assay for HDAC10 Identifies Selective Inhibitors with Cellular Target Engagement द्वारा Herp, Daniel, Ridinger, Johannes, Robaa, Dina, Shinsky, Stephen A., Schmidtkunz, Karin, Yesiloglu, Talha Z., Bayer, Theresa, Steimbach, Raphael R., Herbst‐Gervasoni, Corey J., Merz, Annika, Romier, Christophe, Sehr, Peter, Gunkel, Nikolas, Miller, Aubry K., Christianson, David W., Oehme, Ina, Sippl, Wolfgang, Jung, Manfred
प्रकाशित 2022मूलपाठ -
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Selective agonist of TRPML2 reveals direct role in chemokine release from innate immune cells द्वारा Plesch, Eva, Chen, Cheng-Chang, Butz, Elisabeth, Scotto Rosato, Anna, Krogsaeter, Einar K, Yinan, Hua, Bartel, Karin, Keller, Marco, Robaa, Dina, Teupser, Daniel, Holdt, Lesca M, Vollmar, Angelika M, Sippl, Wolfgang, Puertollano, Rosa, Medina, Diego, Biel, Martin, Wahl-Schott, Christian, Bracher, Franz, Grimm, Christian
प्रकाशित 2018मूलपाठ -
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Pharmacological inhibition of lysine-specific demethylase 1 (LSD1) induces global transcriptional deregulation and ultrastructural alterations that impair viability in Schistosoma... द्वारा Coutinho Carneiro, Vitor, de Abreu da Silva, Isabel Caetano, Amaral, Murilo Sena, Pereira, Adriana S. A., Silveira, Gilbert Oliveira, Pires, David da Silva, Verjovski-Almeida, Sergio, Dekker, Frank J., Rotili, Dante, Mai, Antonello, Lopes-Torres, Eduardo José, Robaa, Dina, Sippl, Wolfgang, Pierce, Raymond J., Borrello, M. Teresa, Ganesan, A., Lancelot, Julien, Thiengo, Silvana, Fernandez, Monica Ammon, Vicentino, Amanda Roberta Revoredo, Mourão, Marina Moraes, Coelho, Fernanda Sales, Fantappié, Marcelo Rosado
प्रकाशित 2020मूलपाठ