检索结果 - Robaa, Dina

Exploring aromatic cage flexibility of the histone methyllysine reader protein Spindlin1 and its impact on binding mode prediction: an in silico study 由 Luise, Chiara, Robaa, Dina, Sippl, Wolfgang

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Muscle Carnitine Palmitoyltransferase II Deficiency: A Review of Enzymatic Controversy and Clinical Features 由 Lehmann, Diana, Motlagh, Leila, Robaa, Dina, Zierz, Stephan

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Pharmacogenetic Aspects of the Interaction of AT1 Receptor Antagonists With ATP-Binding Cassette Transporter ABCG2 由 Ripperger, Anne, Krischer, Anna, Robaa, Dina, Sippl, Wolfgang, Benndorf, Ralf A.

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Histone Deacetylase (HDAC) Inhibitors for the Treatment of Schistosomiasis 由 Ghazy, Ehab, Abdelsalam, Mohamed, Robaa, Dina, Pierce, Raymond J., Sippl, Wolfgang

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Activity of bromodomain protein inhibitors/binders against asexual-stage Plasmodium falciparum parasites 由 Chua, Ming Jang, Robaa, Dina, Skinner-Adams, Tina S., Sippl, Wolfgang, Andrews, Katherine T.

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Binding Free Energy (BFE) Calculations and Quantitative Structure–Activity Relationship (QSAR) Analysis of Schistosoma mansoni Histone Deacetylase 8 (smHDAC8) Inhibitors 由 Simoben, Conrad V., Ghazy, Ehab, Zeyen, Patrik, Darwish, Salma, Schmidt, Matthias, Romier, Christophe, Robaa, Dina, Sippl, Wolfgang

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Docking, Binding Free Energy Calculations and In Vitro Characterization of Pyrazine Linked 2-Aminobenzamides as Novel Class I Histone Deacetylase (HDAC) Inhibitors 由 Bülbül, Emre F., Melesina, Jelena, Ibrahim, Hany S., Abdelsalam, Mohamed, Vecchio, Anita, Robaa, Dina, Zessin, Matthes, Schutkowski, Mike, Sippl, Wolfgang

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HaloTag‐Targeted Sirtuin‐Rearranging Ligand (SirReal) for the Development of Proteolysis‐Targeting Chimeras (PROTACs) against the Lysine Deacetylase Sirtuin 2 (Sirt2) 由 Schiedel, Matthias, Lehotzky, Attila, Szunyogh, Sandor, Oláh, Judit, Hammelmann, Sören, Wössner, Nathalie, Robaa, Dina, Einsle, Oliver, Sippl, Wolfgang, Ovádi, Judit, Jung, Manfred

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Structure–Activity Relationship of Anti-Mycobacterium abscessus Piperidine-4-carboxamides, a New Class of NBTI DNA Gyrase Inhibitors 由 Beuchel, Andreas, Robaa, Dina, Negatu, Dereje A., Madani, Abdeldjalil, Alvarez, Nadine, Zimmerman, Matthew D., Richter, Adrian, Mann, Lea, Hoenke, Sophie, Csuk, René, Dick, Thomas, Imming, Peter

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A Novel Class of Schistosoma mansoni Histone Deacetylase 8 (HDAC8) Inhibitors Identified by Structure-Based Virtual Screening and In Vitro Testing 由 Simoben, Conrad V., Robaa, Dina, Chakrabarti, Alokta, Schmidtkunz, Karin, Marek, Martin, Lancelot, Julien, Kannan, Srinivasaraghavan, Melesina, Jelena, Shaik, Tajith B., Pierce, Raymond J., Romier, Christophe, Jung, Manfred, Sippl, Wolfgang

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Design, Synthesis and Biological Characterization of Histone Deacetylase 8 (HDAC8) Proteolysis Targeting Chimeras (PROTACs) with Anti-Neuroblastoma Activity 由 Darwish, Salma, Ghazy, Ehab, Heimburg, Tino, Herp, Daniel, Zeyen, Patrik, Salem-Altintas, Rabia, Ridinger, Johannes, Robaa, Dina, Schmidtkunz, Karin, Erdmann, Frank, Schmidt, Matthias, Romier, Christophe, Jung, Manfred, Oehme, Ina, Sippl, Wolfgang

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Preclinical Evaluation of Benzazepine-Based PET Radioligands (R)- and (S)-(11)C-Me-NB1 Reveals Distinct Enantiomeric Binding Patterns and a Tightrope Walk Between GluN2B- and σ(1)-... 由 Haider, Ahmed, Herde, Adrienne Müller, Krämer, Stefanie D., Varisco, Jasmine, Keller, Claudia, Frauenknecht, Katrin, Auberson, Yves P., Temme, Louisa, Robaa, Dina, Sippl, Wolfgang, Schibli, Roger, Wünsch, Bernhard, Mu, Linjing, Ametamey, Simon M.

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Synthesis and Biological Investigation of Phenothiazine-Based Benzhydroxamic Acids as Selective Histone Deacetylase 6 (HDAC6) Inhibitors 由 Vögerl, Katharina, Ong, Nghia, Senger, Johanna, Herp, Daniel, Schmidtkunz, Karin, Marek, Martin, Müller, Martin, Bartel, Karin, Shaik, Tajith B., Porter, Nicholas J., Robaa, Dina, Christianson, David W., Romier, Christophe, Sippl, Wolfgang, Jung, Manfred, Bracher, Franz

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Structure-Based Design, Docking and Binding Free Energy Calculations of A366 Derivatives as Spindlin1 Inhibitors 由 Luise, Chiara, Robaa, Dina, Regenass, Pierre, Maurer, David, Ostrovskyi, Dmytro, Seifert, Ludwig, Bacher, Johannes, Burgahn, Teresa, Wagner, Tobias, Seitz, Johannes, Greschik, Holger, Park, Kwang-Su, Xiong, Yan, Jin, Jian, Schüle, Roland, Breit, Bernhard, Jung, Manfred, Sippl, Wolfgang

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Identification of Histone Deacetylase 10 (HDAC10) Inhibitors that Modulate Autophagy in Transformed Cells 由 Zeyen, Patrik, Zeyn, Yanira, Herp, Daniel, Mahmoudi, Fereshteh, Yesiloglu, Talha Z., Erdmann, Frank, Schmidt, Matthias, Robaa, Dina, Romier, Christophe, Ridinger, Johannes, Herbst-Gervasoni, Corey J., Christianson, David W., Oehme, Ina, Jung, Manfred, Krämer, Oliver H., Sippl, Wolfgang

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Synthesis, Molecular Docking and Biological Characterization of Pyrazine Linked 2-Aminobenzamides as New Class I Selective Histone Deacetylase (HDAC) Inhibitors with Anti-Leukemic... 由 Ibrahim, Hany S., Abdelsalam, Mohamed, Zeyn, Yanira, Zessin, Matthes, Mustafa, Al-Hassan M., Fischer, Marten A., Zeyen, Patrik, Sun, Ping, Bülbül, Emre F., Vecchio, Anita, Erdmann, Frank, Schmidt, Matthias, Robaa, Dina, Barinka, Cyril, Romier, Christophe, Schutkowski, Mike, Krämer, Oliver H., Sippl, Wolfgang

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First Fluorescent Acetylspermidine Deacetylation Assay for HDAC10 Identifies Selective Inhibitors with Cellular Target Engagement 由 Herp, Daniel, Ridinger, Johannes, Robaa, Dina, Shinsky, Stephen A., Schmidtkunz, Karin, Yesiloglu, Talha Z., Bayer, Theresa, Steimbach, Raphael R., Herbst‐Gervasoni, Corey J., Merz, Annika, Romier, Christophe, Sehr, Peter, Gunkel, Nikolas, Miller, Aubry K., Christianson, David W., Oehme, Ina, Sippl, Wolfgang, Jung, Manfred

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Selective agonist of TRPML2 reveals direct role in chemokine release from innate immune cells 由 Plesch, Eva, Chen, Cheng-Chang, Butz, Elisabeth, Scotto Rosato, Anna, Krogsaeter, Einar K, Yinan, Hua, Bartel, Karin, Keller, Marco, Robaa, Dina, Teupser, Daniel, Holdt, Lesca M, Vollmar, Angelika M, Sippl, Wolfgang, Puertollano, Rosa, Medina, Diego, Biel, Martin, Wahl-Schott, Christian, Bracher, Franz, Grimm, Christian

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Pharmacological inhibition of lysine-specific demethylase 1 (LSD1) induces global transcriptional deregulation and ultrastructural alterations that impair viability in Schistosoma... 由 Coutinho Carneiro, Vitor, de Abreu da Silva, Isabel Caetano, Amaral, Murilo Sena, Pereira, Adriana S. A., Silveira, Gilbert Oliveira, Pires, David da Silva, Verjovski-Almeida, Sergio, Dekker, Frank J., Rotili, Dante, Mai, Antonello, Lopes-Torres, Eduardo José, Robaa, Dina, Sippl, Wolfgang, Pierce, Raymond J., Borrello, M. Teresa, Ganesan, A., Lancelot, Julien, Thiengo, Silvana, Fernandez, Monica Ammon, Vicentino, Amanda Roberta Revoredo, Mourão, Marina Moraes, Coelho, Fernanda Sales, Fantappié, Marcelo Rosado

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