検索結果 - Régis Denay
- 検索結果 1 - 2 結果 / 2
-
1
Optimization of a Dibenzodiazepine Hit to a Potent and Selective Allosteric PAK1 Inhibitor 著者: Alexei S. Karpov, Payman Amiri, Cornelia Bellamacina, Marie-Hélène Bellance, Werner Breitenstein, Dylan Daniel, Régis Denay, Doriano Fabbro, César Fernández Fernández, Inga Galuba, Stephanie Guerro-Lagasse, Sascha Gutmann, Linda Hinh, Wolfgang Jahnke, Julia Klopp, Albert Lai, Mika Lindvall, Sylvia Ma, Henrik Möbitz, Sabina Pecchi, Gabriele Rummel, Kevin Shoemaker, Joerg Trappe, Charles F. Voliva, Sandra W. Cowan‐Jacob, Andreas L. Marzinzik
出版事項 2015Artigo -
2
Identification and characterization of ternary complexes consisting of FKBP12, MAPRE1 and macrocyclic molecular glues 著者: Michael Salcius, Antonin Tutter, Marianne Fouché, Halіl Koç, Dan King, Anxhela Dhembi, Andrei A. Golosov, Wolfgang Jahnke, Chrystèle Henry, Dayana Argoti, Weiping Jia, Liliana Pedro, Lauren E. Connor, Philippe Piéchon, F.P.A. Fabbiani, Régis Denay, Emine Sager, Juergen Kuehnoel, Marie-Anne Lozac’h, Fabio Lima, Angela Vitrey, Shuyu Chen, Gregory A. Michaud, Marianne Fouche
出版事項 2025Artigo
関連主題
Biochemistry
Biology
Chemistry
Enzyme
Allosteric regulation
Biophysics
Computational biology
Computer science
Cooperativity
Crystallography
Drug discovery
FKBP
Fluorescence
Förster resonance energy transfer
Kinase
Kinome
Nuclear magnetic resonance spectroscopy
PAK1
Physics
Programming language
Quantum mechanics
Stereochemistry
Ternary complex
Ternary operation