Хайлтын үр дүнгүүд - Paul D. Kirchhoff
- 10-н 1 - 10 үр дүнгүүдийг харуулж байна
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Property-based design of a glucosylceramide synthase inhibitor that reduces glucosylceramide in the brain -н Scott D. Larsen, Michael W. Wilson, Akira Abe, Liming Shu, Christopher H. George, Paul D. Kirchhoff, Hollis D. Showalter, Jianming Xiang, Richard F. Keep, James A. Shayman
Хэвлэсэн 2011Artigo -
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Discovery of ARD-2585 as an Exceptionally Potent and Orally Active PROTAC Degrader of Androgen Receptor for the Treatment of Advanced Prostate Cancer -н Weiguo Xiang, Lijie Zhao, Xin Han, Chong Qin, Bukeyan Miao, Donna McEachern, Yu Wang, Hoda Metwally, Paul D. Kirchhoff, Lu Wang, Aleksas Matvekas, Miao He, Bo Wen, Duxin Sun, Shaomeng Wang
Хэвлэсэн 2021Artigo -
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Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors -н Helen V. Waldschmidt, Kristoff T. Homan, Osvaldo Cruz-Rodríguez, M.C. Cato, Jessica Waninger‐Saroni, Kelly M. Larimore, Alessandro Cannavò, Jianliang Song, Joseph Y. Cheung, Paul D. Kirchhoff, Walter J. Koch, J.J.G. Tesmer, Scott D. Larsen
Хэвлэсэн 2016Artigo -
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Development of PVTX-405 as a potent and highly selective molecular glue degrader of IKZF2 for cancer immunotherapy -н Zhixiang Chen, Harshil Dhruv, Xuqing Zhang, Rohan Kalyan Rej, Longchuan Bai, Donna McEachern, Paul D. Kirchhoff, Rakesh Nagilla, Larry J. Jolivette, Cory Rice, Peter Orth, Corey O. Strickland, E. Scott Priestley, Helai P. Mohammad, Meilin Wang, Bo Wen, Duxin Sun, Zhihua Sui, Shaomeng Wang
Хэвлэсэн 2025Artigo -
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Discovery of ARD-1676 as a Highly Potent and Orally Efficacious AR PROTAC Degrader with a Broad Activity against AR Mutants for the Treatment of AR + Human Prostate Cancer -н Weiguo Xiang, Lijie Zhao, Xin Han, Tianfeng Xu, Steven Kregel, Mi Wang, Bukeyan Miao, Chong Qin, Mingliang Wang, Donna McEachern, Jianfeng Lü, Longchuan Bai, Chao‐Yie Yang, Paul D. Kirchhoff, John Takyi‐Williams, Lu Wang, Bo Wen, Duxin Sun, Mark A. Ator, Robert McKean, Arul M. Chinnaiyan, Shaomeng Wang
Хэвлэсэн 2023Artigo -
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Itaconate transporter SLC13A3 impairs tumor immunity via endowing ferroptosis resistance -н Heng Lin, Kole Tison, Yuheng Du, Paul D. Kirchhoff, Chan Kim, Weichao Wang, Hannah Yang, Michael Pitter, Jiali Yu, Peng Liao, Jiajia Zhou, Linda Vatan, Sara Grove, Shuang Wei, Thomas M. Vigil, Yatrik M. Shah, Richard M. Mortensen, Ilona Kryczek, Lana X. Garmire, Jwala Priyadarsini Sivaccumar, Ashwin Ramesh, Ningyan Zhang, Zhiqiang An, Shaomeng Wang, Weiping Zou
Хэвлэсэн 2024Artigo
Хайх хэрэгслүүд:
Холбогдох сэдвүүд
Biology
Chemistry
Biochemistry
Pharmacology
Cancer
Cancer research
Gene
Internal medicine
Medicine
Stereochemistry
In vitro
Androgen receptor
Antibiotics
Bioavailability
Cell biology
Enzyme
Escherichia coli
Genetics
IC50
LNCaP
Prostate
Prostate cancer
Receptor
ATP-binding cassette transporter
Acetylcholine receptor
Acetylcholinesterase
Active center
Active site
Amide
Anemia