Canlyniadau Chwilio - Paul Czodrowski
- Dangos 1 - 8 canlyniadau o 8
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Structural and chemical insights into the covalent-allosteric inhibition of the protein kinase Akt gan Niklas Uhlenbrock, Steven P. Smith, Jörn Weisner, Ina Landel, Marius Lindemann, Thien Anh Le, Julia Hardick, Rajesh Gontla, Rebekka Scheinpflug, Paul Czodrowski, Petra Janning, Laura Depta, Lena Quambusch, Matthias Müller, Bernd Engels, Daniel Rauh
Cyhoeddwyd 2019Artigo -
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Structure-Based Optimization of Potent, Selective, and Orally Bioavailable CDK8 Inhibitors Discovered by High-Throughput Screening gan Paul Czodrowski, Aurélie Mallinger, Dirk Wienke, Christina Esdar, Oliver Pöschke, Michael Busch, Felix Rohdich, Suzanne A. Eccles, Maria-Jesus Ortiz-Ruiz, Richard Schneider, Florence I. Raynaud, Paul A. Clarke, Djordje Müsil, Dániel Schwarz, Trevor Dale, Klaus Urbahns, Julian Blagg, Kai Schiemann
Cyhoeddwyd 2016Artigo -
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Resistance to Avapritinib in PDGFRA-Driven GIST Is Caused by Secondary Mutations in the PDGFRA Kinase Domain gan Susanne Grünewald, Lillian R. Klug, Thomas Mühlenberg, Jonas Lategahn, Johanna Falkenhorst, Ajia Town, Christiane Ehrt, Eva Wardelmann, Wolfgang Hartmann, Hans‐Ulrich Schildhaus, Juergen Treckmann, Jonathan A. Fletcher, Sascha Jung, Paul Czodrowski, Steven P. Miller, Oleg Schmidt-Kittler, Daniel Rauh, Michael C. Heinrich, Sebastian Bauer
Cyhoeddwyd 2020Carta -
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2,8-Disubstituted-1,6-Naphthyridines and 4,6-Disubstituted-Isoquinolines with Potent, Selective Affinity for CDK8/19 gan Aurélie Mallinger, Kai Schiemann, Christian Rink, Jimmy J. P. Sejberg, Mark A. Honey, Paul Czodrowski, Mark Stubbs, Oliver Poeschke, Michael Busch, Richard Schneider, Dániel Schwarz, Djordje Müsil, Rosemary Burke, Klaus Urbahns, Paul Workman, Dirk Wienke, Paul A. Clarke, Florence I. Raynaud, Suzanne A. Eccles, Christina Esdar, Felix Rohdich, Julian Blagg
Cyhoeddwyd 2016Artigo -
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Discovery of Potent, Selective, and Orally Bioavailable Small-Molecule Modulators of the Mediator Complex-Associated Kinases CDK8 and CDK19 gan Aurélie Mallinger, Kai Schiemann, Christian Rink, Frank Stieber, Michel Calderini, Simon Crumpler, Mark Stubbs, Olajumoke Adeniji-Popoola, Oliver Poeschke, Michael Busch, Paul Czodrowski, Djordje Müsil, Dániel Schwarz, Maria-Jesus Ortiz-Ruiz, Richard Schneider, Ching Thai, Melanie Valenti, Alexis de Haven Brandon, Rosemary Burke, Paul Workman, Trevor Dale, Dirk Wienke, Paul A. Clarke, Christina Esdar, Florence I. Raynaud, Suzanne A. Eccles, Felix Rohdich, Julian Blagg
Cyhoeddwyd 2016Artigo -
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A selective chemical probe for exploring the role of CDK8 and CDK19 in human disease gan Trevor Dale, Paul A. Clarke, Christina Esdar, Dennis Waalboer, Olajumoke Adeniji-Popoola, Maria-Jesus Ortiz-Ruiz, Aurélie Mallinger, Rahul S. Samant, Paul Czodrowski, Djordje Müsil, Dániel Schwarz, Klaus Schneider, Mark Stubbs, Kenneth Ewan, Elizabeth Fraser, Robert te Poele, Will Court, Gary Box, Melanie Valenti, Alexis de Haven Brandon, Sharon Gowan, Felix Rohdich, Florence I. Raynaud, Richard Schneider, Oliver Poeschke, Andree Blaukat, Paul Workman, Kai Schiemann, Suzanne A. Eccles, Dirk Wienke, Julian Blagg
Cyhoeddwyd 2015Artigo
Offerynnau Chwilio:
Pynciau Perthynol
Biology
Chemistry
Biochemistry
Biotechnology
In vivo
Kinase
Pharmacology
Signal transduction
Cancer research
Cell cycle
Computer science
Cyclin-dependent kinase
Gene
In vitro
Wnt signaling pathway
Acquired resistance
Allosteric regulation
Artificial intelligence
Binding site
Bioavailability
Bioinformatics
Biological system
Biomedical engineering
Biomolecule
Bubble
Cell
Cell biology
Combinatorial chemistry
Computational chemistry
Computational science