نتائج البحث - Nicholas A. Malmquist
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Triazolopyrimidine-Based Dihydroorotate Dehydrogenase Inhibitors with Potent and Selective Activity against the Malaria Parasite <i>Plasmodium falciparum</i> حسب Margaret A. Phillips, Ramesh Gujjar, Nicholas A. Malmquist, John White, Farah El Mazouni, Jeffrey Baldwin, Pradipsinh K. Rathod
منشور في 2008Artigo -
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High-throughput Screening for Potent and Selective Inhibitors of Plasmodium falciparum Dihydroorotate Dehydrogenase حسب Jeffrey Baldwin, Carolyn H. Michnoff, Nicholas A. Malmquist, John White, Michael G. Roth, Pradipsinh K. Rathod, Margaret A. Phillips
منشور في 2005Artigo -
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Host Cell Entry by Apicomplexa Parasites Requires Actin Polymerization in the Host Cell حسب Virginie Gonzalez, Audrey Combe, Violaine David, Nicholas A. Malmquist, Violaine Delorme, Carole Leroy, Samantha Blazquez, Robert Ménard, Isabelle Tardieux
منشور في 2009Artigo -
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Structural Plasticity of Malaria Dihydroorotate Dehydrogenase Allows Selective Binding of Diverse Chemical Scaffolds حسب Xiaoyi Deng, Ramesh Gujjar, Farah El Mazouni, Werner Kaminsky, Nicholas A. Malmquist, Elizabeth J. Goldsmith, Pradipsinh K. Rathod, Margaret A. Phillips
منشور في 2009Artigo -
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Characterization of <i>Trypanosoma brucei</i> dihydroorotate dehydrogenase as a possible drug target; structural, kinetic and RNAi studies حسب T.L. Arakaki, Frederick S. Buckner, J. Robert Gillespie, Nicholas A. Malmquist, Margaret A. Phillips, Oleksandr Kalyuzhniy, Joseph R. Luft, George T. DeTitta, Christophe L. M. J. Verlinde, Wesley C. Van Voorhis, Wim G. J. Hol, E.A. Merritt
منشور في 2008Artigo -
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Exonuclease-mediated degradation of nascent RNA silences genes linked to severe malaria حسب Qingfeng Zhang, T. Nicolai Siegel, Rafael M. Martins, Fei Wang, Jun Cao, Qi Gao, Xiu Cheng, Lubin Jiang, Chung-Chau Hon, Christine Scheidig‐Benatar, Hiroshi Sakamoto, Louise Turner, Anja T. R. Jensen, Aurélie Claës, Julien Guizetti, Nicholas A. Malmquist, Artur Scherf
منشور في 2014Artigo -
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Histone Methyltransferase Inhibitors Are Orally Bioavailable, Fast-Acting Molecules with Activity against Different Species Causing Malaria in Humans حسب Nicholas A. Malmquist, Sandeep Sundriyal, Joachim Caron, Patty Chen, Benoît Witkowski, Didier Ménard, Rossarin Suwanarusk, Laurent Rénia, François Nosten, Marı́a Belén Jiménez-Dı́az, Íñigo Angulo‐Barturen, María Santos Martínez, Santiago Ferrer, Laura M. Sanz, Francisco‐Javier Gamo, Sergio Wittlin, Sandra Duffy, Vicky M. Avery, Andrea Ruecker, Michael J. Delves, Robert E. Sinden, Matthew J. Fuchter, Artur Scherf
منشور في 2014Artigo
أدوات البحث:
موضوعات ذات صلة
Biochemistry
Biology
Immunology
Malaria
Dihydroorotate dehydrogenase
Enzyme
Chemistry
Gene
Plasmodium falciparum
Cell biology
Computer science
Pharmacology
Purine
Pyrimidine metabolism
Cofactor
Dehydrogenase
Genetics
Methylation
Methyltransferase
Parasite hosting
Plasmodium berghei
RNA
Stereochemistry
World Wide Web
Actin
Active site
Allosteric regulation
Apicomplexa
Aspartate carbamoyltransferase
Binding site