Výsledky vyhledávání - Nicholas A. Malmquist
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Triazolopyrimidine-Based Dihydroorotate Dehydrogenase Inhibitors with Potent and Selective Activity against the Malaria Parasite <i>Plasmodium falciparum</i> Autor Margaret A. Phillips, Ramesh Gujjar, Nicholas A. Malmquist, John White, Farah El Mazouni, Jeffrey Baldwin, Pradipsinh K. Rathod
Vydáno 2008Artigo -
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High-throughput Screening for Potent and Selective Inhibitors of Plasmodium falciparum Dihydroorotate Dehydrogenase Autor Jeffrey Baldwin, Carolyn H. Michnoff, Nicholas A. Malmquist, John White, Michael G. Roth, Pradipsinh K. Rathod, Margaret A. Phillips
Vydáno 2005Artigo -
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Host Cell Entry by Apicomplexa Parasites Requires Actin Polymerization in the Host Cell Autor Virginie Gonzalez, Audrey Combe, Violaine David, Nicholas A. Malmquist, Violaine Delorme, Carole Leroy, Samantha Blazquez, Robert Ménard, Isabelle Tardieux
Vydáno 2009Artigo -
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Structural Plasticity of Malaria Dihydroorotate Dehydrogenase Allows Selective Binding of Diverse Chemical Scaffolds Autor Xiaoyi Deng, Ramesh Gujjar, Farah El Mazouni, Werner Kaminsky, Nicholas A. Malmquist, Elizabeth J. Goldsmith, Pradipsinh K. Rathod, Margaret A. Phillips
Vydáno 2009Artigo -
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Characterization of <i>Trypanosoma brucei</i> dihydroorotate dehydrogenase as a possible drug target; structural, kinetic and RNAi studies Autor T.L. Arakaki, Frederick S. Buckner, J. Robert Gillespie, Nicholas A. Malmquist, Margaret A. Phillips, Oleksandr Kalyuzhniy, Joseph R. Luft, George T. DeTitta, Christophe L. M. J. Verlinde, Wesley C. Van Voorhis, Wim G. J. Hol, E.A. Merritt
Vydáno 2008Artigo -
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Exonuclease-mediated degradation of nascent RNA silences genes linked to severe malaria Autor Qingfeng Zhang, T. Nicolai Siegel, Rafael M. Martins, Fei Wang, Jun Cao, Qi Gao, Xiu Cheng, Lubin Jiang, Chung-Chau Hon, Christine Scheidig‐Benatar, Hiroshi Sakamoto, Louise Turner, Anja T. R. Jensen, Aurélie Claës, Julien Guizetti, Nicholas A. Malmquist, Artur Scherf
Vydáno 2014Artigo -
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Histone Methyltransferase Inhibitors Are Orally Bioavailable, Fast-Acting Molecules with Activity against Different Species Causing Malaria in Humans Autor Nicholas A. Malmquist, Sandeep Sundriyal, Joachim Caron, Patty Chen, Benoît Witkowski, Didier Ménard, Rossarin Suwanarusk, Laurent Rénia, François Nosten, Marı́a Belén Jiménez-Dı́az, Íñigo Angulo‐Barturen, María Santos Martínez, Santiago Ferrer, Laura M. Sanz, Francisco‐Javier Gamo, Sergio Wittlin, Sandra Duffy, Vicky M. Avery, Andrea Ruecker, Michael J. Delves, Robert E. Sinden, Matthew J. Fuchter, Artur Scherf
Vydáno 2014Artigo
Vyhledávací nástroje:
Související témata
Biochemistry
Biology
Immunology
Malaria
Dihydroorotate dehydrogenase
Enzyme
Chemistry
Gene
Plasmodium falciparum
Cell biology
Computer science
Pharmacology
Purine
Pyrimidine metabolism
Cofactor
Dehydrogenase
Genetics
Methylation
Methyltransferase
Parasite hosting
Plasmodium berghei
RNA
Stereochemistry
World Wide Web
Actin
Active site
Allosteric regulation
Apicomplexa
Aspartate carbamoyltransferase
Binding site