نتائج البحث - Michael Rowley
- يعرض 1 - 6 نتائج من 6
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Interdomain Communication in Hepatitis C Virus Polymerase Abolished by Small Molecule Inhibitors Bound to a Novel Allosteric Site حسب Stefania Di Marco, Cinzia Volpari, Licia Tomei, Sergio Altamura, Steven Harper, Frank Narjes, Uwe Koch, Michael Rowley, Raffaele De Francesco, Giovanni Migliaccio, Andrea Carfı́
منشور في 2005Artigo -
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Mechanismof Action and Antiviral Activity of Benzimidazole-Based AllostericInhibitors of the Hepatitis C Virus RNA-Dependent RNAPolymerase حسب Licia Tomei, Sergio Altamura, Linda Bartholomew, Antonino Biroccio, Alessandra Ceccacci, Laura Pacini, Frank Narjes, Nadia Gennari, Monica Bisbocci, Ilario Incitti, Laura Orsatti, Steven Harper, Ian Stansfield, Michael Rowley, Raffaele De Francesco, Giovanni Migliaccio
منشور في 2003Artigo -
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Discovery of (7<i>R</i>)-14-Cyclohexyl-7-{[2-(dimethylamino)ethyl](methyl) amino}-7,8-dihydro-6<i>H</i>-indolo[1,2-<i>e</i>][1,5]benzoxazocine-11-carboxylic Acid (MK-3281), a Poten... حسب Frank Narjes, Benedetta Crescenzi, Marco Ferrara, Jörg Habermann, Stefania Colarusso, Marı́a del Rosario Rico Ferreira, Ian Stansfield, Angela Mackay, Immacolata Conte, Caterina Ercolani, Simone Zaramella, Maria-Cecilia Palumbi, Philip Meuleman, Geert Leroux‐Roels, Claudio Giuliano, Fabrizio Fiore, Stefania Di Marco, Paola Baiocco, Uwe Koch, Giovanni Migliaccio, Sergio Altamura, Ralph Laufer, Raffaele De Francesco, Michael Rowley
منشور في 2010Artigo -
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MK-5172, a Selective Inhibitor of Hepatitis C Virus NS3/4a Protease with Broad Activity across Genotypes and Resistant Variants حسب Vincenzo Summa, Steven W. Ludmerer, John A. McCauley, Christine Fandozzi, Christine Burlein, Claudio Giuliano, Paul J. Coleman, Jillian DiMuzio, Marco Ferrara, Marcello Di Filippo, Adam Gates, Donald J. Graham, Steven J. Harper, Daria J. Hazuda, Carolyn McHale, Edith Monteagudo, Vincenzo Pucci, Michael Rowley, Michael T. Rudd, Aileen Soriano, Mark W. Stahlhut, Joseph P. Vacca, David B. Olsen, Nigel J. Liverton, Steven S. Carroll
منشور في 2012Artigo -
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Discovery of MK-5172, a Macrocyclic Hepatitis C Virus NS3/4a Protease Inhibitor حسب Steven J. Harper, John A. McCauley, Michael T. Rudd, Marco Ferrara, Marcello DiFilippo, Benedetta Crescenzi, Uwe Koch, Alessia Petrocchi, M. Katharine Holloway, John W. Butcher, Joseph J. Romano, Kimberly J. Bush, Kevin F. Gilbert, Charles McIntyre, Kevin T. Nguyen, Emanuela Nizi, Steven S. Carroll, Steven W. Ludmerer, Christine Burlein, Jillian DiMuzio, Donald J. Graham, Carolyn McHale, Mark W. Stahlhut, David B. Olsen, Edith Monteagudo, Simona Cianetti, Claudio Giuliano, Vincenzo Pucci, Nicole Trainor, Christine Fandozzi, Michael Rowley, Paul J. Coleman, Joseph P. Vacca, Vincenzo Summa, Nigel J. Liverton
منشور في 2012Artigo
أدوات البحث:
موضوعات ذات صلة
Biochemistry
Biology
Enzyme
Hepatitis C virus
Virology
Virus
Chemistry
Gene
Allosteric regulation
Antiretroviral therapy
Binding site
Genetics
Genotype
In vitro
NS3
Polymerase
Potency
Protease
Protease inhibitor (pharmacology)
Viral load
Anatomy
Benzimidazole
Computer science
Drug discovery
Foot (prosody)
Genome
Hepacivirus
Human immunodeficiency virus (HIV)
In vivo
Lead compound