Hakutulokset - Matthew L. Dennis
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8‐Mercaptoguanine Derivatives as Inhibitors of Dihydropteroate Synthase Tekijä Matthew L. Dennis, Michael D. Lee, Jitendra R. Harjani, Mohamed Ahmed, Aaron DeBono, Noel P. Pitcher, Zhong‐Chang Wang, Sandeep Chhabra, Νicholas Barlow, Raphaël Rahmani, Ben Cleary, Olan Dolezal, Meghan Hattarki, Luigi Aurelio, Jeremy Shonberg, Bim Graham, Thomas S. Peat, Jonathan B. Baell, James Swarbrick
Julkaistu 2017Artigo -
2
Inhibitors of histone acetyltransferases KAT6A/B induce senescence and arrest tumour growth Tekijä Jonathan B. Baell, David J. Leaver, S.J. Hermans, Gemma L. Kelly, Margs S. Brennan, Natalie L. Downer, Nghi Nguyen, Johannes Wichmann, Helen M. McRae, Yuqing Yang, Ben Cleary, H. Rachel Lagiakos, Stephen Mieruszynski, Guido Pacini, Hannah Vanyai, Maria Bergamasco, Rose E. May, Bethany K. Davey, Kimberly J Morgan, A.J. Sealey, Beinan Wang, Natasha Zamudio, Stephen Wilcox, Alexandra L. Garnham, Bilal N. Sheikh, Brandon J. Aubrey, Karen Doggett, Matthew Chung, Melanie de Silva, John D. Bentley, Pat Pilling, Meghan Hattarki, Olan Dolezal, Matthew L. Dennis, Hendrik Falk, Bin Ren, Susan A. Charman, Karen L. White, Jai Rautela, Andrea Newbold, Edwin D. Hawkins, Ricky W. Johnstone, Nicholas D. Huntington, Thomas S. Peat, Joan K. Heath, Andreas Strasser, Michael W. Parker, Gordon K. Smyth, Ian P. Street, Brendon Monahan, Anne K. Voss, Tim Thomas
Julkaistu 2018Artigo -
3
Discovery of a highly potent, selective, orally bioavailable inhibitor of KAT6A/B histone acetyltransferases with efficacy against KAT6A-high ER+ breast cancer Tekijä Shikhar Sharma, Chi‐Yeh Chung, Sean Uryu, Jelena Petrovic, Joan Cao, Amanda J. Rickard, Nataliya Nady, S.E. Greasley, Eric F. Johnson, Oleg Brodsky, Showkhin Khan, Hui Wang, Zhenxiong Wang, Yong Zhang, Konstantinos Tsaparikos, Lei Chen, Anthony Mazurek, John D. Lapek, Pei‐Pei Kung, Scott C. Sutton, Paul Richardson, Eric C. Greenwald, Shinji Yamazaki, Rhys Jones, Karen A. Maegley, Patrick Bingham, Hieu Lam, Alexandra E. Stupple, Aileen Kamal, Anderly C. Chüeh, Anthony N. Cuzzupe, Benjamin J. Morrow, Bin Ren, Catalina Carrasco‐Pozo, Chin Wee Tan, Dharmesh D. Bhuva, Elizabeth Allan, Elliot Surgenor, François Vaillant, Havva Pehlivanoglu, Hendrik Falk, James R. Whittle, Janet Newman, Joseph Cursons, Judy P. Doherty, Karen L. White, Laura MacPherson, Mark Devlin, Matthew L. Dennis, Meghan Hattarki, Melanie de Silva, Michelle A. Camerino, Miriam Butler, Olan Dolezal, Patricia A. Pilling, Richard C. Foitzik, Paul A. Stupple, H. Rachel Lagiakos, Scott R. Walker, Soroor Hediyeh-zadeh, Stewart D. Nuttall, Sukhdeep K. Spall, Susan A. Charman, Theresa Connor, Thomas S. Peat, Vicky M. Avery, Ylva E. Bozikis, Yuqing Yang, Ming Zhang, Brendon Monahan, Anne K. Voss, Tim Thomas, Ian P. Street, Sarah‐Jane Dawson, Mark A. Dawson, Geoffrey J. Lindeman, Melissa J. Davis, Jane E. Visvader, Thomas A. Paul
Julkaistu 2023Artigo
Työkalut:
Liittyvät aiheet
Biology
Chemistry
Cancer research
Gene
Genetics
Histone
Histone Acetyltransferases
Acetylation
Active site
Biochemistry
Breast cancer
Bromodomain
Cancer
Cell biology
Chromatin
Cofactor
DHPS
Dihydropteroate synthase
Enzyme
Epigenetics
Immunology
Malaria
Plasmodium falciparum
Pterin
Pyrimethamine
Senescence
Stereochemistry
Sulfonamide