תוצאות חיפוש - John S. Sack

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  1. 1
    Crystal structure of microtubule affinity-regulating kinase 4 catalytic domain in complex with a pyrazolopyrimidine inhibitor

    Crystal structure of microtubule affinity-regulating kinase 4 catalytic domain in complex with a pyrazolopyrimidine inhibitor מאת John S. Sack, Mian Gao, Susan E. Kiefer, Joseph E. Myers, John A. Newitt, Sophie Wu, Chunhong Yan

    יצא לאור 2016
    קבל טקסט מלא
    Artigo
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    שמור ב:
  2. 2
    Crystallographic structures of the ligand-binding domains of the androgen receptor and its T877A mutant complexed with the natural agonist dihydrotestosterone

    Crystallographic structures of the ligand-binding domains of the androgen receptor and its T877A mutant complexed with the natural agonist dihydrotestosterone מאת John S. Sack, Kevin Kish, Chihuei Wang, Ricardo M. Attar, Susan E. Kiefer, Yongmi An, Ginger Wu, Julie E. Scheffler, Mark Salvati, Stanley R. Krystek, Roberto Weinmann, Howard Einspahr

    יצא לאור 2001
    קבל טקסט מלא
    Artigo
    הוספה למועדפים
    שמור ב:
  3. 3
    Structural basis for CARM1 inhibition by indole and pyrazole inhibitors

    Structural basis for CARM1 inhibition by indole and pyrazole inhibitors מאת John S. Sack, Sandrine Thieffine, Tiziano Bandiera, Marina Fasolini, Gerald J. Duke, Lata Jayaraman, Kevin Kish, Herbert E. Klei, Ashok V. Purandare, Pamela Rosettani, Sonia Troiani, Dianlin Xie, J. A. Bertrand

    יצא לאור 2011
    קבל טקסט מלא
    Artigo
    הוספה למועדפים
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  4. 4
    Pharmacological and X-Ray Structural Characterization of a Novel Selective Androgen Receptor Modulator: Potent Hyperanabolic Stimulation of Skeletal Muscle with Hypostimulation of Prostate in Rats

    Pharmacological and X-Ray Structural Characterization of a Novel Selective Androgen Receptor Modulator: Potent Hyperanabolic Stimulation of Skeletal Muscle with Hypostimulation of... מאת Jacek Ostrowski, Joyce E. Kuhns, John A. Lupisella, Mark C. Manfredi, Blake C. Beehler, Stanley R. Krystek, Yingzhi Bi, Chong‐Qing Sun, Ramakrishna Seethala, Rajasree Golla, Paul G. Sleph, Aberra Fura, Yongmi An, Kevin Kish, John S. Sack, Kasim A. Mookhtiar, Gary J. Grover, Lawrence G. Hamann

    יצא לאור 2006
    קבל טקסט מלא
    Artigo
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  5. 5
    Structure-based Discovery of Phenyl (3-Phenylpyrrolidin-3-yl)sulfones as Selective, Orally Active RORγt Inverse Agonists

    Structure-based Discovery of Phenyl (3-Phenylpyrrolidin-3-yl)sulfones as Selective, Orally Active RORγt Inverse Agonists מאת James J.‐W. Duan, Zhonghui Lu, Bin Jiang, Sylwia Stachura, Carolyn A. Weigelt, John S. Sack, Javed Khan, Max Ruzanov, Michael A. Galella, Dauh‐Rurng Wu, Melissa Yarde, Ding–Ren Shen, David J. Shuster, Virna Borowski, Jenny Xie, Lisa Zhang, Sridhar Vanteru, Arun Kumar Gupta, Arvind Mathur, Qihong Zhao, William R. Foster, Luisa Salter–Cid, Percy H. Carter, T. G. Murali Dhar

    יצא לאור 2019
    קבל טקסט מלא
    Artigo
    הוספה למועדפים
    שמור ב:
  6. 6
    Identification of imidazo[1,2-<i>b</i>]pyridazine TYK2 pseudokinase ligands as potent and selective allosteric inhibitors of TYK2 signalling

    Identification of imidazo[1,2-<i>b</i>]pyridazine TYK2 pseudokinase ligands as potent and selective allosteric inhibitors of TYK2 signalling מאת Ryan Moslin, Daniel S. Gardner, Joseph B. Santella, Y. Zhang, John V. Duncia, C. Liu, Jian‐Xian Lin, John S. Tokarski, Joann Strnad, Donna L. Pedicord, J. Chen, Yuval Blat, Adriana Zupa-Fernandez, Lihong Cheng, Hongzhi Sun, Charu Chaudhry, Christine Huang, Celia D’Arienzo, John S. Sack, J.K. Muckelbauer, ChiehYing Y. Chang, Jeffrey Tredup, Dan Xie, Nelly Aranı́bar, James R. Burke, P. H. Carter, David S. Weinstein

    יצא לאור 2016
    קבל טקסט מלא
    Artigo
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  7. 7
    Discovery of BMS-986251: A Clinically Viable, Potent, and Selective RORγt Inverse Agonist

    Discovery of BMS-986251: A Clinically Viable, Potent, and Selective RORγt Inverse Agonist מאת Robert J. Cherney, Lyndon A. M. Cornelius, Anurag Srivastava, Carolyn A. Weigelt, David Marcoux, James J.‐W. Duan, Qing Shi, Douglas G. Batt, Qingjie Liu, Shiuhang Yip, Dauh‐Rurng Wu, Max Ruzanov, John S. Sack, Javed Khan, Jinhong Wang, Melissa Yarde, Mary Ellen Cvijic, Arvind Mathur, Sha Li, David J. Shuster, Purnima Khandelwal, Virna Borowski, Jenny Xie, Mary T. Obermeier, Aberra Fura, Kevin Stefanski, Georgia Cornelius, Joseph A. Tino, John E. Macor, Luisa Salter–Cid, Rex Denton, Qihong Zhao, Percy H. Carter, T. G. Murali Dhar

    יצא לאור 2020
    קבל טקסט מלא
    Artigo
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