Resultats de la cerca - Joan Subrath
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1
Synthesis and Characterization of a Dual Kappa-Delta Opioid Receptor Agonist Analgesic Blocking Cocaine Reward Behavior per András Váradi, Gina F. Marrone, Shainnel O. Eans, Michelle L. Ganno, Joan Subrath, Valerie Le Rouzic, Amanda Hunkele, Gavril W. Pasternak, Jay P. McLaughlin, Susruta Majumdar
Publicat 2015Artigo -
2
Synthesis and Evaluation of Aryl-Naloxamide Opiate Analgesics Targeting Truncated Exon 11-Associated μ Opioid Receptor (MOR-1) Splice Variants per Susruta Majumdar, Joan Subrath, Valerie Le Rouzic, Lisa Polikar, Maxim Burgman, Kuni Nagakura, Julie Ocampo, Nathan Haselton, Anna R. Pasternak, Steven G. Grinnell, Ying‐Xian Pan, Gavril W. Pasternak
Publicat 2012Artigo -
3
Mitragynine/Corynantheidine Pseudoindoxyls As Opioid Analgesics with Mu Agonism and Delta Antagonism, Which Do Not Recruit β-Arrestin-2 per András Váradi, Gina F. Marrone, Travis C. Palmer, Ankita Narayan, Márton Richárd Szabó, Valerie Le Rouzic, Steven G. Grinnell, Joan Subrath, Evelyn Warner, Sanjay Kalra, Amanda Hunkele, Jeremy Pagirsky, Shainnel O. Eans, Jéssica Medina, Jin Xu, Ying‐Xian Pan, Attila Borics, Gavril W. Pasternak, Jay P. McLaughlin, Susruta Majumdar
Publicat 2016Artigo -
4
Controlling opioid receptor functional selectivity by targeting distinct subpockets of the orthosteric site per Rajendra Uprety, Tao Che, Saheem A. Zaidi, Steven G. Grinnell, Balázs R. Varga, Abdelfattah Faouzi, Samuel T. Slocum, Abdullah Allaoa, András Váradi, Melissa Nelson, Sarah M. Bernhard, Elizaveta Kulko, Valerie Le Rouzic, Shainnel O. Eans, Chloe A. Simons, Amanda Hunkele, Joan Subrath, Ying‐Xian Pan, Jonathan A. Javitch, Jay P. McLaughlin, Bryan L. Roth, Gavril W. Pasternak, Vsevolod Katritch, Susruta Majumdar
Publicat 2021Artigo
Eines de cerca:
Matèries relacionades
Biochemistry
Chemistry
Opioid
Pharmacology
Receptor
Medicine
Analgesic
G protein-coupled receptor
(+)-Naloxone
Agonism
Agonist
Alkyl
Antagonism
Arrestin
Aryl
Biology
Conditioned place preference
ED50
Exon
Functional selectivity
Gene
In vitro
Law
Morphine
Narcotic antagonists
Opiate
Opioid receptor
Organic chemistry
Political science
Politics