Rezultati - Jean‐Yves Winum
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Carbonic Anhydrase Activators: Gold Nanoparticles Coated with Derivatized Histamine, Histidine, and Carnosine Show Enhanced Activatory Effects on Several Mammalian Isoforms od Mohamed-Chiheb Saada, Jean‐Louis Montero, Daniela Vullo, Andrea Scozzafava, Jean‐Yves Winum, Claudiu T. Supuran
Izdano 2011Artigo -
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Carbonic Anhydrase Inhibitor Coated Gold Nanoparticles Selectively Inhibit the Tumor-Associated Isoform IX over the Cytosolic Isozymes I and II od Maamar Stiti, Alessandro Cecchi, Marouan Rami, Mohamed Abdaoui, Véronique Barragan-Montero, Andrea Scozzafava, Yannick Guari≠, Jean‐Yves Winum, Claudiu T. Supuran
Izdano 2008Artigo -
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Benzoxaboroles: New Potent Inhibitors of the Carbonic Anhydrases of the Pathogenic Bacterium <i>Vibrio cholerae</i> od Alessandro Bonardi, Alessio Nocentini, Roberta Cadoni, Sonia Del Prete, Pascal Dumy, Clemente Capasso, Paola Gratteri, Claudiu T. Supuran, Jean‐Yves Winum
Izdano 2020Artigo -
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Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase od Alessio Nocentini, Andrea Angeli, Fabrizio Carta, Jean‐Yves Winum, Raivis Žalubovskis, Simone Carradori, Clemente Capasso, William A. Donald, Claudiu T. Supuran
Izdano 2021Revisão -
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Targeting the Human 80S Ribosome in Cancer: From Structure to Function and Drug Design for Innovative Adjuvant Therapeutic Strategies od Arnaud Gilles, Léo Fréchin, Kundhavai Natchiar, Giulia Biondani, Ottilie von Loeffelholz, Samuel Holvec, Julie-Lisa Malaval, Jean‐Yves Winum, Bruno P. Klaholz, Jean‐François Peyron
Izdano 2020Revisão -
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Addition to “Stereochemistry Game: Creating and Playing a Fun Board Game To Engage Students in Reviewing Stereochemistry Concepts—The Online Version” od José Nunes da Silva, Daniel Esdras de Andrade Uchoa, Mary Anne Sousa Lima, André Jalles Monteiro, Antonio José Melo Leite, Jean‐Yves Winum, Andrea Basso
Izdano 2021Artigo -
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Hypoxia-Targeting Carbonic Anhydrase IX Inhibitors by a New Series of Nitroimidazole-Sulfonamides/Sulfamides/Sulfamates od Marouan Rami, Ludwig J. Dubois, Nanda-Kumar Parvathaneni, Vincenzo Alterio, Sander M. J. van Kuijk, Simona Maria Monti, Philippe Lambin, Giuseppina De Simone, Claudiu T. Supuran, Jean‐Yves Winum
Izdano 2013Artigo -
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Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment od Andrea Angeli, Fabrizio Carta, Alessio Nocentini, Jean‐Yves Winum, Raivis Žalubovskis, Atilla Akdemir, Valentina Onnis, Wagdy M. Eldehna, Clemente Capasso, Giuseppina De Simone, Simona Maria Monti, Simone Carradori, William A. Donald, Shoukat Dedhar, Claudiu T. Supuran
Izdano 2020Revisão -
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Targeting carbonic anhydrase IX by nitroimidazole based sulfamides enhances the therapeutic effect of tumor irradiation: A new concept of dual targeting drugs od Ludwig J. Dubois, Sarah G.J.A. Peeters, Sander M. J. van Kuijk, Ala Yaromina, Natasja G. Lieuwes, Ruchi Saraya, Rianne Biemans, Marouan Rami, Nanda Kumar Parvathaneni, Daniela Vullo, Marc Vooijs, Claudiu T. Supuran, Jean‐Yves Winum, Philippe Lambin
Izdano 2013Artigo
Iskalna orodja:
Sorodne teme
Chemistry
Biochemistry
Biology
Enzyme
Carbonic anhydrase
Medicine
Cancer
Cancer research
Internal medicine
Organic chemistry
Pharmacology
Gene
Stereochemistry
Genetics
Active site
Combinatorial chemistry
Biotechnology
Breast cancer
Cancer cell
Computer science
Gene isoform
In vitro
In vivo
Isozyme
Materials science
Metastasis
Nanotechnology
Pathology
Sulfamide
Sulfonamide