Sökresultat - Jason R. Clapper
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A Second Generation of Carbamate‐Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo av Jason R. Clapper, Federica Vacondio, Alvin R. King, Andrea Duranti, Andrea Tontini, Cláudia Silva, Silvano Sanchini, Giorgio Tarzia, Marco Mor, Daniele Piomelli
Publicerad 2009Artigo -
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Synthesis and Quantitative Structure−Activity Relationship of Fatty Acid Amide Hydrolase Inhibitors: Modulation at the N-Portion of Biphenyl-3-yl Alkylcarbamates av Marco Mor, Alessio Lodola, Silvia Rivara, Federica Vacondio, Andrea Duranti, Andrea Tontini, Silvano Sanchini, Giovanni Piersanti, Jason R. Clapper, Alvin R. King, Giorgio Tarzia, Daniele Piomelli
Publicerad 2008Artigo -
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URB602 Inhibits Monoacylglycerol Lipase and Selectively Blocks 2-Arachidonoylglycerol Degradation in Intact Brain Slices av Alvin R. King, Andrea Duranti, Andrea Tontini, Silvia Rivara, Anja Rosengarth, Jason R. Clapper, Giuseppe Astarita, Jennifer A. Geaga, Hartmut Luecke, Marco Mor, Giorgio Tarzia, Daniele Piomelli
Publicerad 2007Artigo -
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Fatty Acid Amide Hydrolase Inhibition Heightens Anandamide Signaling Without Producing Reinforcing Effects in Primates av Zuzana Justinová, Regina A. Mangieri, Marco Bortolato, Svetlana I. Chefer, Alexey G. Mukhin, Jason R. Clapper, Alvin R. King, Godfrey H. Redhi, Sevil Yaşar, Daniele Piomelli, Steven R. Goldberg
Publicerad 2008Artigo -
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2-Arachidonoylglycerol Signaling in Forebrain Regulates Systemic Energy Metabolism av Kwang‐Mook Jung, Jason R. Clapper, Jin Fu, Giuseppe D’Agostino, Ana Guijarro, Dean Thongkham, Agnesa Avanesian, Giuseppe Astarita, Nicholas V. DiPatrizio, Andrea Frontini, Saverio Cinti, Sabrina Diano, Daniele Piomelli
Publicerad 2012Artigo -
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Identification of ABX-1431, a Selective Inhibitor of Monoacylglycerol Lipase and Clinical Candidate for Treatment of Neurological Disorders av Justin S. Cisar, Olivia D. Weber, Jason R. Clapper, Jacqueline L. Blankman, Cassandra L. Henry, Gabriel M. Simon, Jessica P. Alexander, Todd K. Jones, R. Alan B. Ezekowitz, Gary P. O’Neill, Cheryl A. Grice
Publicerad 2018Artigo -
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Anandamide suppresses pain initiation through a peripheral endocannabinoid mechanism av Jason R. Clapper, Guillermo Moreno‐Sanz, Roberto Russo, Ana Guijarro, Federica Vacondio, Andrea Duranti, Andrea Tontini, Silvano Sanchini, Natale R. Sciolino, Jessica Marie Spradley, Andrea G. Hohmann, Antonio Calignano, Marco Mor, Giorgio Tarzia, Daniele Piomelli
Publicerad 2010Artigo
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Relaterade ämnen
Cannabinoid receptor
Receptor
Endocannabinoid system
Fatty acid amide hydrolase
Anandamide
Biochemistry
Cannabinoid
Chemistry
Biology
Pharmacology
Agonist
Antagonist
Medicine
2-Arachidonoylglycerol
Diacylglycerol lipase
Enzyme
Internal medicine
Monoacylglycerol lipase
Neuroscience
Serine
Serine hydrolase
Fatty acid
In vitro
Psychology
Stereochemistry
Adipose tissue
Amide
Arachidonic acid
Benzimidazole
Biotechnology