Torthaí cuardaigh - James J.‐W. Duan
- 1 - 2 toradh as 2 á dtaispeáint
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1
Structure-based Discovery of Phenyl (3-Phenylpyrrolidin-3-yl)sulfones as Selective, Orally Active RORγt Inverse Agonists de réir James J.‐W. Duan, Zhonghui Lu, Bin Jiang, Sylwia Stachura, Carolyn A. Weigelt, John S. Sack, Javed Khan, Max Ruzanov, Michael A. Galella, Dauh‐Rurng Wu, Melissa Yarde, Ding–Ren Shen, David J. Shuster, Virna Borowski, Jenny Xie, Lisa Zhang, Sridhar Vanteru, Arun Kumar Gupta, Arvind Mathur, Qihong Zhao, William R. Foster, Luisa Salter–Cid, Percy H. Carter, T. G. Murali Dhar
Foilsithe / Cruthaithe 2019Artigo -
2
Discovery of BMS-986251: A Clinically Viable, Potent, and Selective RORγt Inverse Agonist de réir Robert J. Cherney, Lyndon A. M. Cornelius, Anurag Srivastava, Carolyn A. Weigelt, David Marcoux, James J.‐W. Duan, Qing Shi, Douglas G. Batt, Qingjie Liu, Shiuhang Yip, Dauh‐Rurng Wu, Max Ruzanov, John S. Sack, Javed Khan, Jinhong Wang, Melissa Yarde, Mary Ellen Cvijic, Arvind Mathur, Sha Li, David J. Shuster, Purnima Khandelwal, Virna Borowski, Jenny Xie, Mary T. Obermeier, Aberra Fura, Kevin Stefanski, Georgia Cornelius, Joseph A. Tino, John E. Macor, Luisa Salter–Cid, Rex Denton, Qihong Zhao, Percy H. Carter, T. G. Murali Dhar
Foilsithe / Cruthaithe 2020Artigo
Uirlisí cuardaigh:
Ábhair a bhaineann le hábhar
Agonist
Chemistry
Internal medicine
Inverse agonist
Medicine
Pharmacology
RAR-related orphan receptor gamma
Receptor
Bioavailability
Biochemistry
Biology
Combinatorial chemistry
Computational biology
Computer science
FOXP3
Gene
Geometry
Imiquimod
Immune system
Immunology
Information retrieval
Inverse
Mathematics
Oral administration
Orally active
Pharmacodynamics
Pharmacokinetics
Transcription factor