نتائج البحث - Francisco‐Javier Gamo
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In Vitro Resistance Selections for Plasmodium falciparum Dihydroorotate Dehydrogenase Inhibitors Give Mutants with Multiple Point Mutations in the Drug-binding Site and Altered Gro... حسب Leila S. Ross, Francisco‐Javier Gamo, María José Lafuente-Monasterio, Onkar Singh, Paul Rowland, Roger C. Wiegand, Dyann F. Wirth
منشور في 2014Artigo -
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P. falciparum In Vitro Killing Rates Allow to Discriminate between Different Antimalarial Mode-of-Action حسب Laura M. Sanz, Benigno Crespo, Cristina De-Cózar, Xavier C. Ding, Jose Luis Llergo, Jeremy N. Burrows, José Garcia-Bustos, Francisco‐Javier Gamo
منشور في 2012Artigo -
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Identifying rapidly parasiticidal anti-malarial drugs using a simple and reliable in vitro parasite viability fast assay حسب María Linares, Sara Viera, Benigno Crespo, Virginia Franco, Marı́a G. Gómez-Lorenzo, Marı́a Belén Jiménez-Dı́az, Íñigo Angulo‐Barturen, Laura M. Sanz, Francisco‐Javier Gamo
منشور في 2015Artigo -
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Harnessing evolutionary fitness in <i>Plasmodium falciparum</i> for drug discovery and suppressing resistance حسب Amanda K. Lukens, Leila S. Ross, Richard W. Heidebrecht, Francisco‐Javier Gamo, María José Lafuente-Monasterio, Michael L. Booker, Daniel L. Hartl, Roger C. Wiegand, Dyann F. Wirth
منشور في 2013Artigo -
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Unravelling the mode of action of the Tres Cantos Antimalarial Set (TCAMS): investigating the mechanism of potent antimalarial compounds potentially targeting the human serotonin r... حسب Benedito Matheus dos Santos, Lenna Rosanie Cordero Mallaupoma, Mateus Fila Pecenin, Abhinab Mohanty, Angela Lu, Paula J. Bartlett, Andrew P. Thomas, Francisco‐Javier Gamo, Célia R. S. Garcia
منشور في 2025Artigo -
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Identification of Plasmodium falciparum Mitochondrial Malate: Quinone Oxidoreductase Inhibitors from the Pathogen Box حسب Xinying Wang, Yukiko Miyazaki, D.K. Inaoka, Endah Dwi Hartuti, Yoh‐ichi Watanabe, T. Shiba, Shigeharu Harada, Hiroyuki Saimoto, Jeremy N. Burrows, Francisco Javier Gamo Benito, Tomoyoshi Nozaki, Kiyoshi Kita
منشور في 2019Artigo -
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Drug Screen Targeted at Plasmodium Liver Stages Identifies a Potent Multistage Antimalarial Drug حسب Filipa P. da Cruz, Cécilie Martin, Kathrin Buchholz, María José Lafuente-Monasterio, Tiago Rodrigues, Birte Sönnichsen, Rui Moreira, Francisco‐Javier Gamo, Matthias Marti, Maria M. Mota, Michael Hannus, Miguel Prudêncio
منشور في 2012Artigo -
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Identification of Plasmodium falciparum Mitochondrial Malate: Quinone Oxidoreductase Inhibitors from the Pathogen Box حسب Wang, Xinying, Miyazaki, Yukiko, Inaoka, Daniel Ken, Hartuti, Endah Dwi, Watanabe, Yoh-Ichi, Shiba, Tomoo, Harada, Shigeharu, Saimoto, Hiroyuki, Burrows, Jeremy Nicholas, Benito, Francisco Javier Gamo, Nozaki, Tomoyoshi, Kita, Kiyoshi
منشور في 2019نص -
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Overexpression of plasmepsin II and plasmepsin III does not directly cause reduction in Plasmodium falciparum sensitivity to artesunate, chloroquine and piperaquine حسب Duangkamon Loesbanluechai, Namfon Kotanan, Cristina de Cózar, Theerarat Kochakarn, Megan R. Ansbro, Kesinee Chotivanich, Nicholas J. White, Prapon Wilairat, Lee M, Francisco‐Javier Gamo, Laura M. Sanz, Thanat Chookajorn, Krittikorn Kümpornsin
منشور في 2018Artigo -
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The Parasite Reduction Ratio (PRR) Assay Version 2: Standardized Assessment of Plasmodium falciparum Viability after Antimalarial Treatment In Vitro حسب Annabelle Walz, Maëlle Duffey, Ghaith Aljayyoussi, Sibylle Sax, Didier Leroy, Dominique Besson, Jeremy N. Burrows, Mohammed H. Cherkaoui‐Rbati, Nathalie Gobeau, Marie-Anne Westwood, Christoph Siethoff, Francisco‐Javier Gamo, Pascal Mäser, Sergio Wittlin
منشور في 2023Artigo -
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An Invitation to Open Innovation in Malaria Drug Discovery: 47 Quality Starting Points from the TCAMS حسب Félix Calderón, David Barros, José M. Bueno, José M. Coterón, Esther Fernández, Francisco‐Javier Gamo, José Luís Lavandera, María Luisa León, Simon J. F. Macdonald, Araceli Mallo, Pilar Manzano, Esther Porras, José M. Fiandor, Julia Castro
منشور في 2011Artigo -
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Repositioning: the fast track to new anti-malarial medicines? حسب Julie Lotharius, Francisco Javier Gamo‐Benito, Íñigo Angulo‐Barturen, Julie Clark, Michele Connelly, Santiago Ferrer, Tanya Parkinson, Pavithra Viswanath, Balachandra Bandodkar, Nikhil Rautela, Sowmya Bharath, Sandra Duffy, Vicky M. Avery, Jörg J. Möhrle, R. Kiplin Guy, Timothy N. C. Wells
منشور في 2014Artigo -
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Identification and Validation of Tetracyclic Benzothiazepines as Plasmodium falciparum Cytochrome bc1 Inhibitors حسب Carolyn K. Dong, Sameer Urgaonkar, Joseph F. Cortese, Francisco‐Javier Gamo, José Garcia-Bustos, María José Lafuente, Vishal Patel, Leila S. Ross, Bradley I. Coleman, Emily R. Derbyshire, Clary B. Clish, Adelfa E. Serrano, Mandy Cromwell, Robert H. Barker, Jeffrey D. Dvorin, Manoj T. Duraisingh, Dyann F. Wirth, Jon Clardy, Ralph Mazitschek
منشور في 2011Artigo -
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A high throughput screen for next-generation leads targeting malaria parasite transmission حسب Michael J. Delves, Celia Miguel-Blanco, Holly Matthews, Irene T. Molina‐Martínez, Andrea Ruecker, Sabrina Yahiya, Ursula Straschil, Matthew Abraham, María Luisa León, Oliver Fischer, Ainoa Rueda‐Zubiaurre, Jochen R. Brandt, Álvaro Cortés-Cabrera, Anna Barnard, Matthew J. Fuchter, Félix Calderón, Elizabeth A. Winzeler, Robert E. Sinden, Esperanza Herreros, Francisco‐Javier Gamo, Jake Baum
منشور في 2018Artigo -
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A potent antimalarial benzoxaborole targets a Plasmodium falciparum cleavage and polyadenylation specificity factor homologue حسب Ebere Sonoiki, Caroline L. Ng, Lee M, Denghui Guo, Yong-Kang Zhang, Yasheen Zhou, M.R. Alley, Vida Ahyong, Laura M. Sanz, María José Lafuente-Monasterio, Chen Dong, Patrick G. Schupp, Jiří Gut, Jenny Legac, Roland A. Cooper, Francisco‐Javier Gamo, Joseph L. DeRisi, Yvonne R. Freund, David A. Fidock, Philip J. Rosenthal
منشور في 2017Artigo -
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Histone Methyltransferase Inhibitors Are Orally Bioavailable, Fast-Acting Molecules with Activity against Different Species Causing Malaria in Humans حسب Nicholas A. Malmquist, Sandeep Sundriyal, Joachim Caron, Patty Chen, Benoît Witkowski, Didier Ménard, Rossarin Suwanarusk, Laurent Rénia, François Nosten, Marı́a Belén Jiménez-Dı́az, Íñigo Angulo‐Barturen, María Santos Martínez, Santiago Ferrer, Laura M. Sanz, Francisco‐Javier Gamo, Sergio Wittlin, Sandra Duffy, Vicky M. Avery, Andrea Ruecker, Michael J. Delves, Robert E. Sinden, Matthew J. Fuchter, Artur Scherf
منشور في 2014Artigo -
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MalDA, Accelerating Malaria Drug Discovery حسب Tuo Yang, Sabine Ottilie, Eva S. Istvan, Karla P. Godinez‐Macias, Amanda K. Lukens, Beatriz Baragaña, Brice Campo, Chris Walpole, Jacquin C. Niles, Kelly Chibale, Koen J. Dechering, Manuel Llinás, Lee M, Nobutaka Kato, Susan Wyllie, Case W. McNamara, Francisco‐Javier Gamo, Jeremy N. Burrows, David A. Fidock, Daniel E. Goldberg, Ian H. Gilbert, Dyann F. Wirth, Elizabeth A. Winzeler
منشور في 2021Revisão -
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Generation of a mutator parasite to drive resistome discovery in Plasmodium falciparum حسب Krittikorn Kümpornsin, Theerarat Kochakarn, Tomas Yeo, John Okombo, Madeline R. Luth, Johanna Hoshizaki, Mukul Rawat, Richard D. Pearson, Kyra A. Schindler, Sachel Mok, Heekuk Park, Anne‐Catrin Uhlemann, Gouranga P. Jana, Bikash C. Maity, Benoı̂t Laleu, Elodie Chenu, James Duffy, Sonia Moliner Cubel, Virginia Franco, Marı́a G. Gómez-Lorenzo, Francisco‐Javier Gamo, Elizabeth A. Winzeler, David A. Fidock, Thanat Chookajorn, Lee M
منشور في 2023Artigo
أدوات البحث:
موضوعات ذات صلة
Biology
Immunology
Malaria
Plasmodium falciparum
Pharmacology
Biochemistry
Computer science
Genetics
Gene
Drug
Drug discovery
Medicine
Computational biology
Parasite hosting
Virology
World Wide Web
In vitro
Drug resistance
Bioinformatics
Enzyme
In vivo
Chemistry
Microbiology
Artemisinin
Cell biology
Drug development
Pharmacokinetics
Plasmodium (life cycle)
Potency
Biotechnology