Resultats de la cerca - Ester Fernández‐Salas
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Potato Carboxypeptidase Inhibitor, a T-knot Protein, Is an Epidermal Growth Factor Antagonist That Inhibits Tumor Cell Growth per Carmen Blanco‐Aparicio, Miguel Ángel Molina‐Vila, Ester Fernández‐Salas, Marsha L. Frazier, José Manuel Mas, Enrique Querol, Francesc Avilés, Rafael de Llorens
Publicat 1998Artigo -
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CLIC4 is a tumor suppressor for cutaneous squamous cell cancer per Kwang S. Suh, Mariam Malik, Anjali Shukla, Andrew Ryscavage, Lisa Nolan Wright, Kasey Jividen, John Crutchley, Rebecca A. Dumont, Ester Fernández‐Salas, Joshua D. Webster, Richard J. Simpson, Stuart H. Yuspa
Publicat 2012Artigo -
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Androgen receptor degraders overcome common resistance mechanisms developed during prostate cancer treatment per Steven Kregel, Chao Wang, Xin Han, Lanbo Xiao, Ester Fernández‐Salas, Pushpinder Bawa, Brooke L. McCollum, Kari Wilder-Romans, Ingrid J. Apel, Xuhong Cao, Corey Speers, Shaomeng Wang, Arul M. Chinnaiyan
Publicat 2020Artigo -
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Discovery of a Small-Molecule Degrader of Bromodomain and Extra-Terminal (BET) Proteins with Picomolar Cellular Potencies and Capable of Achieving Tumor Regression per Bing Zhou, Jiantao Hu, Fuming Xu, Zhuo Chen, Longchuan Bai, Ester Fernández‐Salas, Mei Lin, Liu Liu, Chao‐Yie Yang, Yujun Zhao, Donna McEachern, Sally Przybranowski, Bo Wen, Duxin Sun, Shaomeng Wang
Publicat 2017Artigo -
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A potent small-molecule inhibitor of the DCN1-UBC12 interaction that selectively blocks cullin 3 neddylation per Haibin Zhou, Jianfeng Lü, Liu Liu, Denzil Bernard, Chao-Yie Yang, Ester Fernández‐Salas, Krishnapriya Chinnaswamy, Stephanie Danielle Layton, Jeanne A. Stuckey, Qing Yu, Weihua Zhou, Zhen‐Qiang Pan, Yi Sun, Shaomeng Wang
Publicat 2017Artigo -
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Identification of Fibroblast Growth Factor Receptor 3 (FGFR3) as a Protein Receptor for Botulinum Neurotoxin Serotype A (BoNT/A) per Birgitte P. S. Jacky, Patton E. Garay, Jérôme Dupuy, Jeremy B. Nelson, Brian B. Cai, Yanira Molina, Joanne Wang, Lance E. Steward, Ron S. Broide, Joseph Francis, K. Roger Aoki, Raymond C. Stevens, Ester Fernández‐Salas
Publicat 2013Artigo -
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mtCLIC/CLIC4, an Organellular Chloride Channel Protein, Is Increased by DNA Damage and Participates in the Apoptotic Response to p53 per Ester Fernández‐Salas, Kwang S. Suh, Vladislav V. Speransky, Wendy L. Bowers, Joshua M. Levy, Tracey Adams, Kamal Pathak, Lindsay E. Edwards, Daniel Hayes, Christina Cheng, Alasdair C. Steven, Wendy C. Weinberg, Stuart H. Yuspa
Publicat 2002Artigo -
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Design of the First‐in‐Class, Highly Potent Irreversible Inhibitor Targeting the Menin‐MLL Protein–Protein Interaction per Shilin Xu, Angelo Aguilar, Tianfeng Xu, Ke Zheng, Liyue Huang, Jeanne A. Stuckey, Krishnapriya Chinnaswamy, Denzil Bernard, Ester Fernández‐Salas, Liu Liu, Mi Wang, Donna McEachern, Sally Przybranowski, C.L. Foster, Shaomeng Wang
Publicat 2017Artigo -
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Targeted Degradation of BET Proteins in Triple-Negative Breast Cancer per Longchuan Bai, Bing Zhou, Chao‐Yie Yang, Jiao Ji, Donna McEachern, Sally Przybranowski, Hui Jiang, Jiantao Hu, Fuming Xu, Yujun Zhao, Liu Liu, Ester Fernández‐Salas, Jing Xu, Yali Dou, Bo Wen, Duxin Sun, Jennifer L. Meagher, Jeanne A. Stuckey, Daniel F. Hayes, Shunqiang Li, Matthew J. Ellis, Shaomeng Wang
Publicat 2017Artigo -
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Discovery of QCA570 as an Exceptionally Potent and Efficacious Proteolysis Targeting Chimera (PROTAC) Degrader of the Bromodomain and Extra-Terminal (BET) Proteins Capable of Induc... per Chong Qin, Yang Hu, Bing Zhou, Ester Fernández‐Salas, Chao‐Yie Yang, Liu Liu, Donna McEachern, Sally Przybranowski, Mi Wang, Jeanne A. Stuckey, Jennifer L. Meagher, Longchuan Bai, Zhuo Chen, Mei Lin, Jiuling Yang, Danya N. Ziazadeh, Fuming Xu, Jiantao Hu, Weiguo Xiang, Liyue Huang, Siwei Li, Bo Wen, Duxin Sun, Shaomeng Wang
Publicat 2018Artigo -
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Autophagy inhibition by targeting PIKfyve potentiates response to immune checkpoint blockade in prostate cancer per Yuanyuan Qiao, Jae Eun Choi, Jean C. Tien, Stephanie A. Simko, Thekkelnaycke M. Rajendiran, Josh N. Vo, Andrew Delekta, Lisha Wang, Lanbo Xiao, Nathan Hodge, Parth Desai, Sergio Mendoza, Kristin Juckette, Alice Xu, Tanu Soni, Fengyun Su, Rui Wang, Xuhong Cao, Jiali Yu, Ilona Kryczek, Xiao Ming Wang, Xiaoju Wang, Javed Siddiqui, Zhen Wang, Amélie Bernard, Ester Fernández‐Salas, Nora M. Navone, Stephanie J. Ellison, Ke Ding, Eeva‐Liisa Eskelinen, Elisabeth I. Heath, Daniel J. Klionsky, Weiping Zou, Arul M. Chinnaiyan
Publicat 2021Artigo
Eines de cerca:
Matèries relacionades
Biology
Biochemistry
Chemistry
Cancer research
Cell biology
Gene
Cancer
Medicine
Genetics
Internal medicine
Apoptosis
Immunology
Molecular biology
Receptor
BET inhibitor
BRD4
Botulinum neurotoxin
Bromodomain
Cell growth
Chloride channel
Computational biology
Enzyme
Epidermal growth factor receptor
Epigenetics
Exocytosis
Fusion protein
Prostate cancer
Protein–protein interaction
Proteolysis
Recombinant DNA