檢索結果 - Emma K. Lendy
- Showing 1 - 7 results of 7
-
1
-
2
Indole Chloropyridinyl Ester-Derived SARS-CoV-2 3CLpro Inhibitors: Enzyme Inhibition, Antiviral Efficacy, Structure–Activity Relationship, and X-ray Structural Studies 由 Arun K. Ghosh, Jakka Raghavaiah, Dana Shahabi, Monika Yadav, Brandon J. Anson, Emma K. Lendy, Shin-ichiro Hattori, Nobuyo Higashi‐Kuwata, Hiroaki Mitsuya, Andrew D. Mesecar
出版 2021Artigo -
3
A small molecule compound with an indole moiety inhibits the main protease of SARS-CoV-2 and blocks virus replication 由 Shin-ichiro Hattori, Nobuyo Higashi‐Kuwata, Hironori Hayashi, Srinivasa Rao Allu, Jakka Raghavaiah, Haydar Bulut, Debananda Das, Brandon J. Anson, Emma K. Lendy, Yuki Takamatsu, Nobutoki Takamune, Naoki Kishimoto, Kazutaka Murayama, Kazuya Hasegawa, Mi Li, David A. Davis, Eiichi Kodama, Robert Yarchoan, Alexander Wlodawer, Shogo Misumi, Andrew D. Mesecar, Arun K. Ghosh, Hiroaki Mitsuya
出版 2021Artigo -
4
Genetic variants of phospholipase C-γ2 alter the phenotype and function of microglia and confer differential risk for Alzheimer’s disease 由 Andy P. Tsai, Chuanpeng Dong, Peter Bor‐Chian Lin, Adrian L. Oblak, Gonzalo Viana Di Prisco, Nian Wang, Nicole Hajicek, Adam J. Carr, Emma K. Lendy, Oliver Hãhn, Micaiah Atkins, Aulden Foltz, Jheel Patel, Guixiang Xu, Miguel Moutinho, John Sondek, Qisheng Zhang, Andrew D. Mesecar, Yunlong Liu, Brady K. Atwood, Tony Wyss‐Coray, Kwangsik Nho, Stephanie J. Bissel, Bruce T. Lamb, Gary E. Landreth
出版 2023Artigo -
5
Discovery of SARS-CoV-2 antiviral drugs through large-scale compound repurposing 由 Laura Riva, Shuofeng Yuan, Xin Yin, Laura Martin‐Sancho, Naoko Matsunaga, Lars Pache, Sebastian Burgstaller-Muehlbacher, Paul D. De Jesus, Peter Teriete, Mitchell Hull, Max W. Chang, Jasper Fuk‐Woo Chan, Jianli Cao, Vincent Kwok‐Man Poon, Kristina M. Herbert, Kuoyuan Cheng, Tu-Trinh H. Nguyen, Andrey Rubanov, Yuan Pu, Courtney Nguyen, Angela Choi, Raveen Rathnasinghe, Michael Schotsaert, Lisa Miorin, Marion Déjosez, Thomas P. Zwaka, Ko-Yung Sit, Luis Martínez‐Sobrido, Wen‐Chun Liu, Kris M. White, Mackenzie E. Chapman, Emma K. Lendy, Richard Glynne, Randy A. Albrecht, Eytan Ruppin, Andrew D. Mesecar, Jeffrey R. Johnson, Christopher Benner, Ren Sun, Peter G. Schultz, Andrew I. Su, Adolfo García‐Sastre, Arnab K. Chatterjee, Kwok‐Yung Yuen, Sumit K. Chanda
出版 2020Artigo -
6
Discovery of a Novel Inhibitor of Coronavirus 3CL Protease for the Potential Treatment of COVID-19 由 Britton Boras, Rhys Jones, Brandon J. Anson, Dan Arenson, Lisa Aschenbrenner, Malina A. Bakowski, Nathan Beutler, Joseph Binder, Emily Chen, Heather Eng, Holly Hammond, Jennifer Hammond, Robert Haupt, Robert L. Hoffman, Eugene P. Kadar, Rob Kania, Emi Kimoto, Melanie G. Kirkpatrick, Lorraine F. Lanyon, Emma K. Lendy, Jonathan R. Lillis, James Logue, Suman Luthra, Chunlong Ma, Stephen W. Mason, Marisa E. McGrath, Stephen Noell, R. Scott Obach, Matthew N. O’Brien, Rebecca E. O’Connor, Kevin Ogilvie, Dafydd R. Owen, Martin Pettersson, Matthew R. Reese, Thomas F. Rogers, Michelle I. Rossulek, Jean G. Sathish, Norimitsu Shirai, Claire M. Steppan, Martyn D. Ticehurst, Lawrence W. Updyke, Stuart Weston, Yuao Zhu, Jun Wang, Arnab K. Chatterjee, Andrew D. Mesecar, Matthew B. Frieman, Annaliesa S. Anderson, Charlotte Allerton
出版 2020Pré-impressão -
7
Preclinical characterization of an intravenous coronavirus 3CL protease inhibitor for the potential treatment of COVID19 由 Britton Boras, Rhys Jones, Brandon J. Anson, Dan Arenson, Lisa Aschenbrenner, Malina A. Bakowski, Nathan Beutler, Joseph Binder, Emily Chen, Heather Eng, Holly Hammond, Jennifer Hammond, Robert Haupt, Robert L. Hoffman, Eugene P. Kadar, Rob Kania, Emi Kimoto, Melanie G. Kirkpatrick, Lorraine F. Lanyon, Emma K. Lendy, Jonathan R. Lillis, James Logue, Suman Luthra, Chunlong Ma, Stephen W. Mason, Marisa E. McGrath, Stephen Noell, R. Scott Obach, Matthew N. O’ Brien, Rebecca E. O’Connor, Kevin Ogilvie, Dafydd R. Owen, Martin Pettersson, Matthew R. Reese, Thomas F. Rogers, Romel Rosales, Michelle I. Rossulek, Jean G. Sathish, Norimitsu Shirai, Claire M. Steppan, Martyn D. Ticehurst, Lawrence W. Updyke, Stuart Weston, Yuao Zhu, Kris M. White, Adolfo García‐Sastre, Jun Wang, Arnab K. Chatterjee, Andrew D. Mesecar, Matthew B. Frieman, Annaliesa S. Anderson, Charlotte Allerton
出版 2021Artigo
相關主題
Biochemistry
Biology
Chemistry
Disease
Enzyme
Medicine
Coronavirus disease 2019 (COVID-19)
In vitro
Infectious disease (medical specialty)
Pathology
Virology
Virus
Coronavirus
Genetics
Pharmacology
Protease
Stereochemistry
ADME
Antiretroviral therapy
Antiviral drug
Drug
Gene
In vivo
Indole test
Prodrug
Protease inhibitor (pharmacology)
Viral load
Viral replication
Aerospace engineering
Alzheimer's disease