Resultats de la cerca - Elliot D. Mock
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Design of a Highly Selective Quenched Activity-Based Probe and Its Application in Dual Color Imaging Studies of Cathepsin S Activity Localization per Kristina Oresic Bender, Leslie O. Ofori, Wouter A. van der Linden, Elliot D. Mock, Gopal K. Datta, Somenath Chowdhury, Hao Li, Ehud Segal, Mateo I. Sánchez, Jonathan A. Ellman, Carl G. Figdor, Matthew Bogyo, Martijn Verdoes
Publicat 2015Artigo -
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Incorporation of Non-natural Amino Acids Improves Cell Permeability and Potency of Specific Inhibitors of Proteasome Trypsin-like Sites per Paul P. Geurink, Wouter A. van der Linden, Anne Mirabella, Nerea Gallastegui, Gerjan de Bruin, Annet E. M. Blom, Mathias J. Voges, Elliot D. Mock, Bogdan I. Florea, Gijs A. van der Marel, Christoph Driessen, Mario van der Stelt, M. Groll, Herman S. Overkleeft, Alexei F. Kisselev
Publicat 2013Artigo -
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Mitochondrial dysfunction and mitophagy defects in <i>LRRK2-R1441C</i> Parkinson’s disease models per Matthew G Williamson, Marta Madureira, William McGuinness, Rachel Héon-Roberts, Elliot D. Mock, Kalina Naidoo, Kaitlyn M. L. Cramb, Maria Claudia Caiazza, Ana Belén Malpartida, Martha Lavelle, Katrina Savory, Stewart W. Humble, Ryan Patterson, John B. Davis, Natalie Connor‐Robson, Brent J. Ryan, Richard Wade‐Martins
Publicat 2023Artigo -
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USP30 inhibition improves mitochondrial health through both PINK1-dependent and independent mechanisms per Matthew G Williamson, Rachel Héon-Roberts, Sarah N. J. Franks, Elliot D. Mock, Hannah B. L. Jones, Elena Britti, Ana Belén Malpartida, Mahmoud A. Bassal, Martha Lavelle, J. W. Connor, Aina Mogas Barcons, Katherine L. Hammond, Katrina Savory, Pavandeep Rai, Anna Lavayssiere, William McGuinness, Natalie Sepke, Jane Vowles, Iolanda Vendrell, Franziska Guenther, Benedikt M. Kessler, Sally A. Cowley, Katherine S. England, Emma J. Murphy, John B. Davis, Richard Wade‐Martins, Brent J. Ryan
Publicat 2025Pré-impressão -
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Cannabinoid CB2 receptor ligand profiling reveals biased signalling and off-target activity per Marjolein Soethoudt, Uwe Grether, Jürgen Fingerle, Travis W. Grim, Filomena Fezza, Luciano De Petrocellis, Christoph Ullmer, Benno Rothenhäusler, Camille Perret, Noortje van Gils, David B. Finlay, Christa MacDonald, Andrea Chicca, Marianela Dalghi Gens, Jordyn Stuart, Henk de Vries, Nicolina Mastrangelo, Lizi Xia, Georgios Alachouzos, Marc P. Baggelaar, Andrea Martella, Elliot D. Mock, Hui Deng, Laura H. Heitman, Mark Connor, Vincenzo Di Marzo, Jürg Gertsch, Aron H. Lichtman, Mauro Maccarrone, Pál Pacher, Michelle Glass, Mario van der Stelt
Publicat 2017Artigo -
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Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474 per Annelot C. M. van Esbroeck, Antonius P. A. Janssen, Armand B. Cognetta, Daisuke Ogasawara, Guy Shpak, Mark van der Kroeg, Vasudev Kantae, Marc P. Baggelaar, Femke M.S. de Vrij, Hui Deng, Marco Allarà, Filomena Fezza, Zhanmin Lin, Tom van der Wel, Marjolein Soethoudt, Elliot D. Mock, Hans den Dulk, Ilse L. Baak, Bogdan I. Florea, Giel Hendriks, Luciano De Petrocellis, Herman S. Overkleeft, Thomas Hankemeier, Chris I. De Zeeuw, Vincenzo Di Marzo, Mauro Maccarrone, Benjamin F. Cravatt, Steven A. Kushner, Mario van der Stelt
Publicat 2017Artigo -
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Discovery of a NAPE-PLD inhibitor that modulates emotional behavior in mice per Elliot D. Mock, Mohammed Ahmed Mustafa, Ozge Gunduz‐Cinar, Reşat Çınar, Gavin N. Petrie, Vasudev Kantae, Xinyu Di, Daisuke Ogasawara, Zoltán V. Varga, János Pálóczi, Cristina Miliano, Giulia Donvito, Annelot C. M. van Esbroeck, Anouk M. F. van der Gracht, Ioli Kotsogianni, Joshua K. Park, Andrea Martella, Tom van der Wel, Marjolein Soethoudt, Ming Jiang, Tiemen J. Wendel, Antonius P. A. Janssen, Alexander T. Bakker, Colleen Donovan, Laura I. Castillo, Bogdan I. Florea, Jesse W.Y. Wat, Helma van den Hurk, Matthias Wittwer, Uwe Grether, Andrew Holmes, C. A. A. VAN BOECKEL, Thomas Hankemeier, Benjamin F. Cravatt, Matthew W. Buczynski, Matthew N. Hill, Pál Pacher, Aron H. Lichtman, Mario van der Stelt
Publicat 2020Artigo
Eines de cerca:
Matèries relacionades
Biology
Biochemistry
Chemistry
Cell biology
Cannabinoid receptor
Receptor
Cannabinoid
Endocannabinoid system
Pharmacology
Agonist
Anandamide
Antagonist
Apoptosis
Autophagy
Cannabinoid receptor type 2
Drug
Enzyme
Fatty acid amide hydrolase
Immunology
In vitro
Lipid signaling
Mitochondrion
Mitophagy
PINK1
Bortezomib
Cannabinoid Receptor Agonists
Carfilzomib
Cathepsin
Cathepsin B
Cathepsin D