Výsledky vyhledávání - Elisa Uliassi
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Enriching Proteolysis Targeting Chimeras with a Second Modality: When Two Are Better Than One Autor Alessandra Salerno, Francesca Seghetti, Jessica Caciolla, Elisa Uliassi, Eleonora Testi, Melissa Guardigni, Marinella Roberti, Andrea Milelli, María Laura Bolognesi
Vydáno 2022Revisão -
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The Use of Zidovudine Pharmacophore in Multi-Target-Directed Ligands for AIDS Therapy Autor Maria da Conceição Avelino Dias Bianco, Débora Inácio Leite, Frederico Silva Castelo Branco, Núbia Boechat, Elisa Uliassi, María Laura Bolognesi, Mônica M. Bastos
Vydáno 2022Revisão -
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Structure-Based Design of 3-(4-Aryl-1<i>H</i>-1,2,3-triazol-1-yl)-Biphenyl Derivatives as P2Y<sub>14</sub> Receptor Antagonists Autor Anna Junker, R. Balasubramanian, Antonella Ciancetta, Elisa Uliassi, Evgeny Kiselev, Chiara Martiriggiano, Kevin Trujillo, Giorgi Mtchedlidze, Leah Birdwell, Kyle A. Brown, T. Kendall Harden, Kenneth A. Jacobson
Vydáno 2016Artigo -
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Design, Synthesis and Structure—Activity Relationships of a Phenotypic Small Library against Protozoan Infections Autor Elisa Uliassi, Lorna Piazzi, Federica Belluti, Marcel Kaiser, Reto Brun, Sheraz Gul, Bernhard Ellinger, Carolina Borsoi Moraes, Lúcio H. Freitas-Júnior, Chiara Borsari, Maria Paola Costi, María Laura Bolognesi
Vydáno 2017Artigo -
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Turning Donepezil into a Multi‐Target‐Directed Ligand through a Merging Strategy Autor Rosaria Carmela Perone, Claudia Albertini, Elisa Uliassi, Flaminia Di Pietri, Pedro de Sena Murteira Pinheiro, Sabrina Petralla, Nicola Rizzardi, Romana Fato, Lenka Pulkrabkova, Ondřej Soukup, Anna Tramarin, Manuela Bartolini, María Laura Bolognesi
Vydáno 2020Artigo -
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PROTAC-Induced Glycogen Synthase Kinase 3β Degradation as a Potential Therapeutic Strategy for Alzheimer’s Disease Autor Melissa Guardigni, Letizia Pruccoli, Alan Santini, Angela De Simone, Matteo Bersani, Francesca Spyrakis, Flavia Frabetti, Elisa Uliassi, Vincenza Andrisano, Barbara Pagliarani, Paula Fernández-Gómez, Valle Palomo, María Laura Bolognesi, Andrea Tarozzi, Andrea Milelli
Vydáno 2023Artigo -
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Front Cover: Discovery of Sustainable Drugs for Neglected Tropical Diseases: Cashew Nut Shell Liquid (CNSL)‐Based Hybrids Target Mitochondrial Function and ATP Production in <i>Try... Autor Michela Cerone, Elisa Uliassi, Federica Prati, Godwin U. Ebiloma, Leandro Lemgruber, Christian Bergamini, David G. Watson, Thais de A. M. Ferreira, Gabriella Simões Heyn, Luiz Antônio Soares Romeiro, Harry P. de Koning, María Laura Bolognesi
Vydáno 2019Paratexto -
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Discovery of sustainable drugs for Alzheimer's disease: cardanol-derived cholinesterase inhibitors with antioxidant and anti-amyloid properties Autor Giselle de Andrade Ramos, Andressa Souza de Oliveira, Manuela Bartolini, Marina Naldi, Irene Liparulo, Christian Bergamini, Elisa Uliassi, Ling Wu, Paul E. Fraser, M.L. Abreu, Alessandra S. Kiametis, Ricardo Gargano, Edilberto R. Silveira, Guilherme D. Brand, Lukáš Prchal, Ondřej Soukup, Jan Korábečný, María Laura Bolognesi, Luiz Antônio Soares Romeiro
Vydáno 2021Artigo -
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Crassiflorone derivatives that inhibit Trypanosoma brucei glyceraldehyde-3-phosphate dehydrogenase ( Tb GAPDH) and Trypanosoma cruzi trypanothione reductase ( Tc TR) and display tr... Autor Elisa Uliassi, Giulia Fiorani, R. Luise Krauth‐Siegel, Christian Bergamini, Romana Fato, Giulia Bianchini, J. Carlos Menéndez, Marı́a Teresa Molina, Eulogio López-Montero, Federico Falchi, Andrea Cavalli, Sheraz Gul, Maria Kuzikov, Bernhard Ellinger, Gesa Witt, Carolina Borsoi Moraes, Lúcio H. Freitas-Júnior, Chiara Borsari, Maria Paola Costi, María Laura Bolognesi
Vydáno 2017Artigo -
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Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease Autor Katarina Chalupova, Jan Korábečný, Manuela Bartolini, Barbara Monti, Doriano Lamba, Rosanna Caliandro, Alessandro Pesaresi, Xavier Brazzolotto, Anne-Julie Gastellier, Florian Nachon, Jaroslav Pejchal, Michaela Jarosova, Vendula Hepnarová, Daniel Jun, Martina Hrabinová, Rafael Doležal, Jana Žďárová Karasová, Martin Mžik, Zdena Krištofíková, Jan Misík, Ľubica Múčková, Petr Jošt, Ondřej Soukup, Markéta Benková, Vladimı́r Setnička, Lucie Habartová, Markéta Chvojková, Lenka Kletečková, Karel Valeš, Eva Mezeiová, Elisa Uliassi, Martin Vališ, Eugenie Nepovimová, María Laura Bolognesi, Kamil Kuča
Vydáno 2019Artigo -
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Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform Autor Carolina Borsoi Moraes, Gesa Witt, Maria Kuzikov, Bernhard Ellinger, Theodora Calogeropoulou, Kyriakos C. Prousis, Stefano Mangani, F. Di Pisa, Giacomo Landi, Lucia Dello Iacono, Cecilia Pozzi, Lúcio H. Freitas-Júnior, Bruno dos Santos Pascoalino, Claudia P. Bertolacini, Birte Behrens, Oliver Keminer, Jennifer Leu, Markus Wolf, Jeanette Reinshagen, Anabela Cordeiro‐da‐Silva, Nuno Santarém, Alberto Venturelli, Stephen K. Wrigley, Deepa Karunakaran, Bethlehem Kebede, Ina Pöhner, Wolfgang G. Müller, Joanna Panecka-Hofman, Rebecca C. Wade, Martina Fenske, Joachim Clos, José María Alunda, María Jesús Corral, Elisa Uliassi, María Laura Bolognesi, Pasquale Linciano, Antonio Quotadamo, Stefania Ferrari, Matteo Santucci, Chiara Borsari, Maria Paola Costi, Sheraz Gul
Vydáno 2019Artigo
Vyhledávací nástroje:
Související témata
Medicine
Biology
Chemistry
Biochemistry
Enzyme
Pharmacology
Disease
Computer science
Drug discovery
Gene
Pathology
Bioinformatics
Combinatorial chemistry
Computational biology
Acetylcholinesterase
Alzheimer's disease
Biotechnology
Drug
Internal medicine
Neuroscience
Aché
Butyrylcholinesterase
Cashew nut
Genetics
Microbiology
Organic chemistry
Parasite hosting
Psychology
Receptor
Trypanosoma brucei