Resultats de la cerca - Duffy, Sandra
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Plasmodium falciparum in vitro continuous culture conditions: A comparison of parasite susceptibility and tolerance to anti-malarial drugs throughout the asexual intra-erythrocytic... per Duffy, Sandra, Avery, Vicky M.
Publicat 2017Text -
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Identification of MMV Malaria Box Inhibitors of Plasmodium falciparum Early-Stage Gametocytes Using a Luciferase-Based High-Throughput Assay per Lucantoni, Leonardo, Duffy, Sandra, Adjalley, Sophie H., Fidock, David A., Avery, Vicky M.
Publicat 2013Text -
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A Meroisoprenoid, Heptenolides, and C-Benzylated Flavonoids from Sphaerocoryne gracilis ssp. gracilis per Maeda, Gasper, Munissi, Joan J. E., Lindblad, Sofia, Duffy, Sandra, Pelletier, Jerry, Avery, Vicky M., Nyandoro, Stephen S., Erdélyi, Máté
Publicat 2020Text -
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Identification and In-Vitro ADME Assessment of a Series of Novel Anti-Malarial Agents Suitable for Hit-to-Lead Chemistry per Edlin, Chris D., Morgans, Garreth, Winks, Susan, Duffy, Sandra, Avery, Vicky M., Wittlin, Sergio, Waterson, David, Burrows, Jeremy, Bryans, Justin
Publicat 2012Text -
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An evaluation of Minor Groove Binders as anti-Trypanosoma brucei brucei therapeutics per Scott, Fraser J., Khalaf, Abedawn I., Giordani, Federica, Wong, Pui Ee, Duffy, Sandra, Barrett, Michael, Avery, Vicky M., Suckling, Colin J.
Publicat 2016Text -
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Prenylated Flavonoids from the Roots of Tephrosia rhodesica per Atilaw, Yoseph, Muiva-Mutisya, Lois, Bogaerts, Jonathan, Duffy, Sandra, Valkonen, Arto, Heydenreich, Matthias, Avery, Vicky M., Rissanen, Kari, Erdélyi, Máté, Yenesew, Abiy
Publicat 2020Text -
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Screening and hit evaluation of a chemical library against blood-stage Plasmodium falciparum per Avery, Vicky M, Bashyam, Sridevi, Burrows, Jeremy N, Duffy, Sandra, Papadatos, George, Puthukkuti, Shyni, Sambandan, Yuvaraj, Singh, Shivendra, Spangenberg, Thomas, Waterson, David, Willis, Paul
Publicat 2014Text -
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Screening the Medicines for Malaria Venture Pathogen Box across Multiple Pathogens Reclassifies Starting Points for Open-Source Drug Discovery per Duffy, Sandra, Sykes, Melissa L., Jones, Amy J., Shelper, Todd B., Simpson, Moana, Lang, Rebecca, Poulsen, Sally-Ann, Sleebs, Brad E., Avery, Vicky M.
Publicat 2017Text -
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Secoiridoids and Iridoids from Morinda asteroscepa per Zandi, Linda, Makungu, Marco, Munissi, Joan J. E., Duffy, Sandra, Puttreddy, Rakesh, von der Heiden, Daniel, Rissanen, Kari, Avery, Vicky M., Nyandoro, Stephen S., Erdélyi, Máté
Publicat 2020Text -
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A New Benzopyranyl Cadenane Sesquiterpene and Other Antiplasmodial and Cytotoxic Metabolites from Cleistochlamys kirkii per Nyandoro, Stephen S., Maeda, Gasper, Munissi, Joan J.E., Gruhonjic, Amra, Fitzpatrick, Paul A., Lindblad, Sofia, Duffy, Sandra, Pelletier, Jerry, Pan, Fangfang, Puttreddy, Rakesh, Avery, Vicky M., Erdélyi, Máté
Publicat 2019Text -
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One-pot, multi-component synthesis and structure-activity relationships of peptoid-based histone deacetylase (HDAC) inhibitors targeting malaria parasites per Diedrich, Daniela, Stenzel, Katharina, Hesping, Eva, Antonova-Koch, Yevgeniya, Gebru, Tamirat, Duffy, Sandra, Fisher, Gillian, Schöler, Andrea, Meister, Stephan, Kurz, Thomas, Avery, VickyM., Winzeler, Elizabeth A., Held, Jana, Andrews, Katherine T., Hansen, Finn K.
Publicat 2018Text -
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Repositioning: the fast track to new anti-malarial medicines? per Lotharius, Julie, Gamo-Benito, Francisco Javier, Angulo-Barturen, Iñigo, Clark, Julie, Connelly, Michele, Ferrer-Bazaga, Santiago, Parkinson, Tanya, Viswanath, Pavithra, Bandodkar, Balachandra, Rautela, Nikhil, Bharath, Sowmya, Duffy, Sandra, Avery, Vicky M, Möhrle, Jörg J, Guy, R Kiplin, Wells, Timothy
Publicat 2014Text -
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Lysine Acetylation in Sexual Stage Malaria Parasites Is a Target for Antimalarial Small Molecules per Trenholme, Katharine, Marek, Linda, Duffy, Sandra, Pradel, Gabriele, Fisher, Gillian, Hansen, Finn K., Skinner-Adams, Tina S., Butterworth, Alice, Ngwa, Che Julius, Moecking, Jonas, Goodman, Christopher D., McFadden, Geoffrey I., Sumanadasa, Subathdrage D. M., Fairlie, David P., Avery, Vicky M., Kurz, Thomas, Andrews, Katherine T.
Publicat 2014Text -
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Target Validation and Identification of Novel Boronate Inhibitors of the Plasmodium falciparum Proteasome per Xie, Stanley C., Gillett, David L., Spillman, Natalie J., Tsu, Christopher, Luth, Madeline R., Ottilie, Sabine, Duffy, Sandra, Gould, Alexandra E., Hales, Paul, Seager, Benjamin A., Charron, Carlie L., Bruzzese, Frank, Yang, Xiaofeng, Zhao, Xiansi, Huang, Shih-Chung, Hutton, Craig A., Burrows, Jeremy N., Winzeler, Elizabeth A., Avery, Vicky M., Dick, Lawrence R., Tilley, Leann
Publicat 2018Text -
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Histone Methyltransferase Inhibitors Are Orally Bioavailable, Fast-Acting Molecules with Activity against Different Species Causing Malaria in Humans per Malmquist, Nicholas A., Sundriyal, Sandeep, Caron, Joachim, Chen, Patty, Witkowski, Benoit, Menard, Didier, Suwanarusk, Rossarin, Renia, Laurent, Nosten, Francois, Jiménez-Díaz, María Belén, Angulo-Barturen, Iñigo, Martínez, María Santos, Ferrer, Santiago, Sanz, Laura M., Gamo, Francisco-Javier, Wittlin, Sergio, Duffy, Sandra, Avery, Vicky M., Ruecker, Andrea, Delves, Michael J., Sinden, Robert E., Fuchter, Matthew J., Scherf, Artur
Publicat 2015Text -
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Discovery of a Quinoline-4-carboxamide Derivative with a Novel Mechanism of Action, Multistage Antimalarial Activity, and Potent in Vivo Efficacy per Baragaña, Beatriz, Norcross, Neil R., Wilson, Caroline, Porzelle, Achim, Hallyburton, Irene, Grimaldi, Raffaella, Osuna-Cabello, Maria, Norval, Suzanne, Riley, Jennifer, Stojanovski, Laste, Simeons, Frederick R. C., Wyatt, Paul G., Delves, Michael J., Meister, Stephan, Duffy, Sandra, Avery, Vicky M., Winzeler, Elizabeth A., Sinden, Robert E., Wittlin, Sergio, Frearson, Julie A., Gray, David W., Fairlamb, Alan H., Waterson, David, Campbell, Simon F., Willis, Paul, Read, Kevin D., Gilbert, Ian H.
Publicat 2016Text -
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Hexahydroquinolines are Antimalarial Candidates with Potent Blood Stage and Transmission-Blocking Activity per Vanaerschot, Manu, Lucantoni, Leonardo, Li, Tao, Combrinck, Jill M., Ruecker, Andrea, Kumar, T.R. Santha, Rubiano, Kelly, Ferreira, Pedro E., Siciliano, Giulia, Gulati, Sonia, Henrich, Philipp P., Ng, Caroline L., Murithi, James M., Corey, Victoria C., Duffy, Sandra, Lieberman, Ori J., Veiga, M. Isabel, Sinden, Robert E., Alano, Pietro, Delves, Michael J., Sim, Kim Lee, Winzeler, Elizabeth A., Egan, Timothy J., Hoffman, Stephen L., Avery, Vicky M., Fidock, David A.
Publicat 2017Text