检索结果 - Divyabharathi Chepyala
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The orally bioavailable GSPT1/2 degrader SJ6986 exhibits in vivo efficacy in acute lymphoblastic leukemia 由 Yunchao Chang, Fatemeh Keramatnia, Pankaj S. Ghate, Gisele Nishiguchi, Qingsong Gao, Ilaria Iacobucci, Lei Yang, Divyabharathi Chepyala, Ashutosh Mishra, Anthony A. High, Hiroaki Goto, Koshi Akahane, Junmin Peng, Jun J. Yang, Marcus Fischer, Zoran Ranković, Charles G. Mullighan
出版 2023Artigo -
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Identification of Potent, Selective, and Orally Bioavailable Small-Molecule GSPT1/2 Degraders from a Focused Library of Cereblon Modulators 由 Gisele Nishiguchi, Fatemeh Keramatnia, Jaeki Min, Yunchao Chang, Barbara Jonchère, Sourav Das, Marisa Actis, Jeanine E. Price, Divyabharathi Chepyala, Brandon Young, Kevin M. McGowan, P.J. Slavish, Anand Mayasundari, Jamie Jarusiewicz, Lei Yang, Yong Li, Xiang Fu, Shalandus H. Garrett, James B. Papizan, Kiran Kodali, Junmin Peng, Shondra Miller, Martine F. Roussel, Charles G. Mullighan, Marcus Fischer, Zoran Ranković
出版 2021Artigo -
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Degradation of Janus kinases in <i>CRLF2</i>-rearranged acute lymphoblastic leukemia 由 Yunchao Chang, Jaeki Min, Jamie Jarusiewicz, Marisa Actis, S.Y.C. Bradford, Anand Mayasundari, Lei Yang, Divyabharathi Chepyala, Lisa J. Alcock, Kathryn G. Roberts, Stanley Nithianantham, Dylan Maxwell, Lauren Rowland, Randolph K. Larsen, Aman Seth, Hiroaki Goto, Toshihiko Imamura, Koshi Akahane, Baranda S. Hansen, Shondra M. Pruett‐Miller, Elisabeth Paietta, Mark R. Litzow, Chunxu Qu, Jun J. Yang, Marcus Fischer, Zoran Ranković, Charles G. Mullighan
出版 2021Artigo
相关主题
Biology
Biochemistry
Cancer research
Cell biology
Genetics
Immunology
In vivo
Leukemia
Pharmacology
Apoptosis
Bioavailability
Bone marrow
Bruton's tyrosine kinase
Cell culture
Cell growth
Cereblon
Chemical library
Chemistry
Computational biology
Cytotoxicity
Drug discovery
Ex vivo
Gene
Haematopoiesis
In vitro
JAK-STAT signaling pathway
Janus kinase
Kinase
Medicine
Myelofibrosis