תוצאות חיפוש - Dina Robaa
- Showing 1 - 17 results of 17
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Proteolysis targeting chimeras (PROTACs) for epigenetics research מאת Anja Vogelmann, Dina Robaa, Wolfgang Sippl, Manfred Jung
יצא לאור 2020Revisão -
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Ternary Complex Modeling, Induced Fit Docking and Molecular Dynamics Simulations as a Successful Approach for the Design of VHL‐Mediated PROTACs Targeting the Kinase FLT3 מאת Husam Nassar, Anne‐Christin Sarnow, İ. Çelik, Mohamed Abdelsalam, Dina Robaa, Wolfgang Sippl
יצא לאור 2025Artigo -
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Evolutionary relationships among protein lysine deacetylases of parasites causing neglected diseases מאת Larissa Scholte, Marina de Moraes Mourão, Fabiano Pais, Jelena Melesina, Dina Robaa, Ângela C. Volpini, Wolfgang Sippl, Raymond J. Pierce, Guilherme Oliveira, Laila Alves Nahum
יצא לאור 2017Artigo -
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A Novel Class of Schistosoma mansoni Histone Deacetylase 8 (HDAC8) Inhibitors Identified by Structure-Based Virtual Screening and In Vitro Testing מאת Conrad V. Simoben, Dina Robaa, Alokta Chakrabarti, Matthias Schmidt, Martin Marek, Julien Lancelot, Srinivasaraghavan Kannan, Jelena Melesina, T.B. Shaik, Raymond J. Pierce, Christophe Romier, Manfred Jung, Wolfgang Sippl
יצא לאור 2018Artigo -
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Design, Synthesis and Biological Characterization of Histone Deacetylase 8 (HDAC8) Proteolysis Targeting Chimeras (PROTACs) with Anti-Neuroblastoma Activity מאת Salma Darwish, Ehab Ghazy, Tino Heimburg, Daniel Herp, Patrik Zeyen, Rabia Salem-Altintas, Johannes Ridinger, Dina Robaa, Matthias Schmidt, Frank Erdmann, Matthias Schmidt, Christophe Romier, Manfred Jung, Ina Oehme, Wolfgang Sippl
יצא לאור 2022Artigo -
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Structure-Based Design and Synthesis of Novel Inhibitors Targeting HDAC8 from <i>Schistosoma mansoni</i> for the Treatment of Schistosomiasis מאת Tino Heimburg, Alokta Chakrabarti, Julien Lancelot, Martin Marek, Jelena Melesina, Alexander‐Thomas Hauser, T.B. Shaik, Sylvie Duclaud, Dina Robaa, Frank Erdmann, Matthias Schmidt, Christophe Romier, Raymond J. Pierce, Manfred Jung, Wolfgang Sippl
יצא לאור 2016Artigo -
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Synthesis and Biological Investigation of Phenothiazine-Based Benzhydroxamic Acids as Selective Histone Deacetylase 6 Inhibitors מאת Katharina Vögerl, Nghia Ong, Johanna Senger, Daniel Herp, Matthias Schmidt, Martin Marek, Martin Müller, Karin Bartel, T.B. Shaik, Nicholas J. Porter, Dina Robaa, D.W. Christianson, Christophe Romier, Wolfgang Sippl, Manfred Jung, Franz Bracher
יצא לאור 2019Artigo -
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Development of Alkylated Hydrazides as Highly Potent and Selective Class I Histone Deacetylase Inhibitors with T cell Modulatory Properties מאת Ping Sun, Jing Wang, Khadija Shahed Khan, Weiqin Yang, Wai‐Lung Ng, Nikita V. Ilment, Matthes Zessin, Emre F. Bülbül, Dina Robaa, Frank Erdmann, Matthias Schmidt, Christophe Romier, Mike Schutkowski, Alfred S.L. Cheng, Wolfgang Sippl
יצא לאור 2022Artigo -
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Identification of histone deacetylase 10 (HDAC10) inhibitors that modulate autophagy in transformed cells מאת Patrik Zeyen, Yanira Zeyn, Daniel Herp, Fereshteh Mahmoudi, Talha Z. Yesiloglu, Frank Erdmann, Matthias Schmidt, Dina Robaa, Christophe Romier, Johannes Ridinger, Corey J. Herbst‐Gervasoni, D.W. Christianson, Ina Oehme, Manfred Jung, Oliver H. Krämer, Wolfgang Sippl
יצא לאור 2022Artigo -
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Characterization of Histone Deacetylase 8 (HDAC8) Selective Inhibition Reveals Specific Active Site Structural and Functional Determinants מאת Martin Marek, T.B. Shaik, Tino Heimburg, Alokta Chakrabarti, Julien Lancelot, Elizabeth Ramos‐Morales, Cyrielle da Veiga, Dmitrii V. Kalinin, Jelena Melesina, Dina Robaa, Matthias Schmidt, Takayoshi Suzuki, Ralph Holl, Eric Ennifar, Raymond J. Pierce, Manfred Jung, Wolfgang Sippl, Christophe Romier
יצא לאור 2018Artigo -
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Synthesis, Molecular Docking and Biological Characterization of Pyrazine Linked 2-Aminobenzamides as New Class I Selective Histone Deacetylase (HDAC) Inhibitors with Anti-Leukemic... מאת Hany S. Ibrahim, Mohamed Abdelsalam, Yanira Zeyn, Matthes Zessin, Al‐Hassan M. Mustafa, Marten A. Fischer, Patrik Zeyen, Ping Sun, Emre F. Bülbül, Anita Vecchio, Frank Erdmann, Matthias Schmidt, Dina Robaa, Cyril Bařinka, Christophe Romier, Mike Schutkowski, Oliver H. Krämer, Wolfgang Sippl
יצא לאור 2021Artigo -
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Selective agonist of TRPML2 reveals direct role in chemokine release from innate immune cells מאת Eva Plesch, Cheng‐Chang Chen, Elisabeth Butz, Anna Scotto Rosato, Einar Krogsaeter, Hua Yinan, Karin Bartel, Marco Keller, Dina Robaa, Daniel Teupser, Lesca M. Holdt, Angelika M. Vollmar, Wolfgang Sippl, Rosa Puertollano, Diego L. Medina, Martin Biel, Christian Wahl‐Schott, Franz Bracher, Christian Grimm
יצא לאור 2018Artigo -
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Pharmacological inhibition of lysine-specific demethylase 1 (LSD1) induces global transcriptional deregulation and ultrastructural alterations that impair viability in <i>Schistoso... מאת Vitor Coutinho Carneiro, Isabel Caetano de Abreu da Silva, Murilo Sena Amaral, Adriana S. A. Pereira, Gilbert O. Silveira, David da Silva Pires, Sérgio Verjovski-Almeida, Frank J. Dekker, Dante Rotili, Antonello Mai, Eduardo José Lopes Torres, Dina Robaa, Wolfgang Sippl, Raymond J. Pierce, María Teresa Borrello, A. Ganesan, Julien Lancelot, Silvana Carvalho Thiengo, Mônica Ammon Fernandez, Amanda Roberta Revoredo Vicentino, Marina de Moraes Mourão, Fernanda Sales Coelho, Marcelo Rosado Fantappíé
יצא לאור 2019Pré-impressão -
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Pharmacological inhibition of lysine-specific demethylase 1 (LSD1) induces global transcriptional deregulation and ultrastructural alterations that impair viability in Schistosoma... מאת Vitor Coutinho Carneiro, Isabel Caetano de Abreu da Silva, Murilo Sena Amaral, Adriana S. A. Pereira, Gilbert O. Silveira, David da Silva Pires, Sérgio Verjovski-Almeida, Frank J. Dekker, Dante Rotili, Antonello Mai, Eduardo José Lopes Torres, Dina Robaa, Wolfgang Sippl, Raymond J. Pierce, María Teresa Borrello, A. Ganesan, Julien Lancelot, Silvana Carvalho Thiengo, Mônica Ammon Fernandez, Amanda Roberta Revoredo Vicentino, Marina de Moraes Mourão, Fernanda Sales Coelho, Marcelo Rosado Fantappíé
יצא לאור 2020Artigo
כלי חיפוש:
נושאים קשורים
Biochemistry
Biology
Gene
Chemistry
Histone
Histone deacetylase
Cell biology
Enzyme
Computational biology
Epigenetics
HDAC8
Pharmacology
Drug discovery
Immunology
In vitro
Cancer research
DNA
Helminths
Medicine
Schistosoma mansoni
Schistosomiasis
Acetylation
Bioinformatics
Computer science
Docking (animal)
Gene knockdown
Genetics
Nursing
Schistosoma
Biotechnology