Kết quả tìm kiếm - David Smil
- Đang hiển thị 1 - 15 kết quả của 15
-
1
-
2
Discovery of a Dual PRMT5–PRMT7 Inhibitor Bằng David Smil, Mohammad S. Eram, Fengling Li, Sidney H. Kennedy, Magdalena M. Szewczyk, Peter J. Brown, Dalia Baršytė-Lovejoy, C.H. Arrowsmith, Masoud Vedadi, Matthieu Schapira
Được phát hành 2015Artigo -
3
Bromo-deaza-SAH: A potent and selective DOT1L inhibitor Bằng Wenyu Yu, David Smil, Fengling Li, W. Tempel, O. Fedorov, Kong T. Nguyen, Yuri Bolshan, Rima Al‐awar, Stefan Knapp, C.H. Arrowsmith, Masoud Vedadi, Peter J. Brown, Matthieu Schapira
Được phát hành 2013Artigo -
4
Exploiting an Allosteric Binding Site of PRMT3 Yields Potent and Selective Inhibitors Bằng Feng Liu, Fengling Li, Anqi Ma, E. Dobrovetsky, Aiping Dong, Cen Gao, Ilia Korboukh, Jing Liu, David Smil, Peter J. Brown, Stephen V. Frye, C.H. Arrowsmith, Matthieu Schapira, Masoud Vedadi, Jian Jin
Được phát hành 2013Artigo -
5
Discovery of a Potent, Selective, and Cell-Active Dual Inhibitor of Protein Arginine Methyltransferase 4 and Protein Arginine Methyltransferase 6 Bằng Yudao Shen, Magdalena M. Szewczyk, Mohammad S. Eram, David Smil, H. Ümit Kanıskan, Renato Ferreira de Freitas, Guillermo Senisterra, Fengling Li, Matthieu Schapira, Peter J. Brown, C.H. Arrowsmith, Dalia Baršytė-Lovejoy, Jing Liu, Masoud Vedadi, Jian Jin
Được phát hành 2016Artigo -
6
Synthesis, Optimization, and Evaluation of Novel Small Molecules as Antagonists of WDR5-MLL Interaction Bằng Yuri Bolshan, Matthäus Getlik, Ekaterina Kuznetsova, Gregory A. Wasney, Taraneh Hajian, Gennadiy Poda, Kong T. Nguyen, Hong Wu, L. Dombrovski, Aiping Dong, Guillermo Senisterra, Matthieu Schapira, C.H. Arrowsmith, Peter J. Brown, Rima Al‐awar, Masoud Vedadi, David Smil
Được phát hành 2013Artigo -
7
Probing the SAM Binding Site of SARS-CoV-2 Nsp14 In Vitro Using SAM Competitive Inhibitors Guides Developing Selective Bisubstrate Inhibitors Bằng Kanchan Devkota, Matthieu Schapira, Sumera Perveen, Aliakbar Khalili Yazdi, Fengling Li, Irene Chau, Pegah Ghiabi, Taraneh Hajian, P. Loppnau, Albina Bolotokova, K.J.F. Satchell, Ke Wang, Deyao Li, Jing Liu, David Smil, Minkui Luo, Jian Jin, Paul V. Fish, Peter J. Brown, Masoud Vedadi
Được phát hành 2021Artigo -
8
Small-molecule inhibition of MLL activity by disruption of its interaction with WDR5 Bằng Guillermo Senisterra, Hong Wu, Abdellah Allali‐Hassani, Gregory A. Wasney, Dalia Baršytė-Lovejoy, L. Dombrovski, Aiping Dong, Kong T. Nguyen, David Smil, Yuri Bolshan, Taraneh Hajian, Hao He, Alma Seitova, Irene Chau, Fengling Li, Gennadiy Poda, Jean‐François Couture, Peter J. Brown, Rima Al‐awar, Matthieu Schapira, C.H. Arrowsmith, Masoud Vedadi
Được phát hành 2012Artigo -
9
An Allosteric Inhibitor of Protein Arginine Methyltransferase 3 Bằng Alena Siarheyeva, Guillermo Senisterra, Abdellah Allali‐Hassani, Aiping Dong, E. Dobrovetsky, Gregory A. Wasney, Irene Chau, Richard Marcellus, Taraneh Hajian, Feng Liu, Ilia Korboukh, David Smil, Yuri Bolshan, Jinrong Min, Hong Wu, Hong Zeng, P. Loppnau, Gennadiy Poda, Carly Griffin, Ahmed Aman, Peter J. Brown, Jian Jin, Rima Al‐awar, C.H. Arrowsmith, Matthieu Schapira, Masoud Vedadi
Được phát hành 2012Artigo -
10
A chemical biology toolbox to study protein methyltransferases and epigenetic signaling Bằng Sebastian Scheer, Suzanne Ackloo, Tiago da Silva Medina, Matthieu Schapira, Fengling Li, Jennifer Ward, Andrew M. Lewis, Jeffrey P. Northrop, Paul L. Richardson, H. Ümit Kanıskan, Yudao Shen, Jing Liu, David Smil, David McLeod, Carlos Zepeda‐Velázquez, Minkui Luo, Jian Jin, Dalia Baršytė-Lovejoy, K. Huber, Daniel D. De Carvalho, Masoud Vedadi, Colby Zaph, Peter J. Brown, C.H. Arrowsmith
Được phát hành 2018Artigo -
11
Erratum: Pharmacological targeting of the Wdr5-MLL interaction in C/EBPα N-terminal leukemia. Bằng Florian Grebien, Masoud Vedadi, Matthäus Getlik, Roberto Giambruno, Amit Grover, Roberto Avellino, Anna Skucha, Sarah Vittori, Ekaterina Kuznetsova, David Smil, Dalia Baršytė-Lovejoy, Fengling Li, Gennadiy Poda, Matthieu Schapira, Hong Wu, Aiping Dong, Guillermo Senisterra, Alexey Stukalov, K. Huber, Andreas Schönegger, Richard Marcellus, Martin Bilban, Christoph Bock, Peter J. Brown, Johannes Zuber, Keiryn L. Bennett, Rima Al‐awar, Ruud Delwel, Claus Nerlov, C.H. Arrowsmith, Giulio Superti‐Furga
Được phát hành 2015Errata/Corrigenda -
12
A Potent, Selective and Cell‐Active Allosteric Inhibitor of Protein Arginine Methyltransferase 3 (PRMT3) Bằng H. Ümit Kanıskan, Magdalena M. Szewczyk, Zhengtian Yu, Mohammad S. Eram, Xiaobao Yang, Keith T. Schmidt, Xiao Luo, Miao Dai, Feng He, Irene Zang, Ying Lin, Sidney H. Kennedy, Fengling Li, E. Dobrovetsky, Aiping Dong, David Smil, Sun‐Joon Min, Melissa Landon, Jennifer Lin‐Jones, Xi‐Ping Huang, Bryan L. Roth, Matthieu Schapira, Peter Atadja, Dalia Baršytė-Lovejoy, C.H. Arrowsmith, Peter J. Brown, Kehao Zhao, Jian Jin, Masoud Vedadi
Được phát hành 2015Artigo -
13
Pharmacological targeting of the Wdr5-MLL interaction in C/EBPα N-terminal leukemia Bằng Florian Grebien, Masoud Vedadi, Matthäus Getlik, Roberto Giambruno, Amit Grover, Roberto Avellino, Anna Skucha, Sarah Vittori, Ekaterina Kuznetsova, David Smil, Dalia Baršytė-Lovejoy, Fengling Li, Gennadiy Poda, Matthieu Schapira, Hong Wu, Aiping Dong, Guillermo Senisterra, Alexey Stukalov, K. Huber, Andreas Schönegger, Richard Marcellus, Martin Bilban, Christoph Bock, Peter J. Brown, Johannes Zuber, Keiryn L. Bennett, Rima Al‐awar, Ruud Delwel, Claus Nerlov, C.H. Arrowsmith, Giulio Superti‐Furga
Được phát hành 2015Artigo -
14
MLL5 Orchestrates a Cancer Self-Renewal State by Repressing the Histone Variant H3.3 and Globally Reorganizing Chromatin Bằng Marco Gallo, Fiona J. Coutinho, Robert J. Vanner, Tenzin Gayden, Stephen C. Mack, Alex Murison, Marc Remke, Li Ren, Naoya Takayama, Kinjal Desai, Lilian Lee, Xiaoyang Lan, Nicole I. Park, Dalia Baršytė-Lovejoy, David Smil, Dominik Sturm, Michelle Kushida, Renee Head, Michael D. Cusimano, Mark Bernstein, Ian D. Clarke, John E. Dick, Stefan M. Pfister, Jeremy N. Rich, C.H. Arrowsmith, Michael D. Taylor, Nada Jabado, David P. Bazett‐Jones, Mathieu Lupien, Peter B. Dirks
Được phát hành 2015Artigo -
15
Functional interdependence of BRD4 and DOT1L in MLL leukemia Bằng Omer Gilan, Enid Y.N. Lam, Isabelle Becher, Dave Lugo, Ester Cannizzaro, Gérard Joberty, Aoife Ward, Meike Wiese, Chun Yew Fong, Sarah Ftouni, Dean Tyler, Kym L. Stanley, Laura MacPherson, Chen-Fang Weng, Yih-Chih Chan, Margherita Ghisi, David Smil, Christopher Carpenter, Peter J. Brown, Neil Garton, Marnie E. Blewitt, Andrew J. Bannister, Tony Kouzarides, Brian J.P. Huntly, Ricky W. Johnstone, Gerard Drewes, Sarah‐Jane Dawson, C.H. Arrowsmith, Paola Grandi, Rab K. Prinjha, Mark A. Dawson
Được phát hành 2016Artigo
Công cụ tìm kiếm:
Các môn học liên quan
Biology
Chemistry
Gene
Biochemistry
Methylation
Methyltransferase
Cell biology
Enzyme
Epigenetics
Genetics
Amino acid
Cancer research
Chromatin
Computational biology
Histone
In vitro
RNA
Allosteric regulation
Arginine
Chemical biology
DNA
Histone H3
Leukemia
Binding site
Computer science
Gene expression
Histone methyltransferase
Lysine
Peptide
Pharmacology