檢索結果 - David Smil
- Showing 1 - 15 results of 15
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Exploiting an Allosteric Binding Site of PRMT3 Yields Potent and Selective Inhibitors 由 Feng Liu, Fengling Li, Anqi Ma, E. Dobrovetsky, Aiping Dong, Cen Gao, Ilia Korboukh, Jing Liu, David Smil, Peter J. Brown, Stephen V. Frye, C.H. Arrowsmith, Matthieu Schapira, Masoud Vedadi, Jian Jin
出版 2013Artigo -
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Discovery of a Potent, Selective, and Cell-Active Dual Inhibitor of Protein Arginine Methyltransferase 4 and Protein Arginine Methyltransferase 6 由 Yudao Shen, Magdalena M. Szewczyk, Mohammad S. Eram, David Smil, H. Ümit Kanıskan, Renato Ferreira de Freitas, Guillermo Senisterra, Fengling Li, Matthieu Schapira, Peter J. Brown, C.H. Arrowsmith, Dalia Baršytė-Lovejoy, Jing Liu, Masoud Vedadi, Jian Jin
出版 2016Artigo -
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Synthesis, Optimization, and Evaluation of Novel Small Molecules as Antagonists of WDR5-MLL Interaction 由 Yuri Bolshan, Matthäus Getlik, Ekaterina Kuznetsova, Gregory A. Wasney, Taraneh Hajian, Gennadiy Poda, Kong T. Nguyen, Hong Wu, L. Dombrovski, Aiping Dong, Guillermo Senisterra, Matthieu Schapira, C.H. Arrowsmith, Peter J. Brown, Rima Al‐awar, Masoud Vedadi, David Smil
出版 2013Artigo -
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Probing the SAM Binding Site of SARS-CoV-2 Nsp14 In Vitro Using SAM Competitive Inhibitors Guides Developing Selective Bisubstrate Inhibitors 由 Kanchan Devkota, Matthieu Schapira, Sumera Perveen, Aliakbar Khalili Yazdi, Fengling Li, Irene Chau, Pegah Ghiabi, Taraneh Hajian, P. Loppnau, Albina Bolotokova, K.J.F. Satchell, Ke Wang, Deyao Li, Jing Liu, David Smil, Minkui Luo, Jian Jin, Paul V. Fish, Peter J. Brown, Masoud Vedadi
出版 2021Artigo -
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Small-molecule inhibition of MLL activity by disruption of its interaction with WDR5 由 Guillermo Senisterra, Hong Wu, Abdellah Allali‐Hassani, Gregory A. Wasney, Dalia Baršytė-Lovejoy, L. Dombrovski, Aiping Dong, Kong T. Nguyen, David Smil, Yuri Bolshan, Taraneh Hajian, Hao He, Alma Seitova, Irene Chau, Fengling Li, Gennadiy Poda, Jean‐François Couture, Peter J. Brown, Rima Al‐awar, Matthieu Schapira, C.H. Arrowsmith, Masoud Vedadi
出版 2012Artigo -
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An Allosteric Inhibitor of Protein Arginine Methyltransferase 3 由 Alena Siarheyeva, Guillermo Senisterra, Abdellah Allali‐Hassani, Aiping Dong, E. Dobrovetsky, Gregory A. Wasney, Irene Chau, Richard Marcellus, Taraneh Hajian, Feng Liu, Ilia Korboukh, David Smil, Yuri Bolshan, Jinrong Min, Hong Wu, Hong Zeng, P. Loppnau, Gennadiy Poda, Carly Griffin, Ahmed Aman, Peter J. Brown, Jian Jin, Rima Al‐awar, C.H. Arrowsmith, Matthieu Schapira, Masoud Vedadi
出版 2012Artigo -
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A chemical biology toolbox to study protein methyltransferases and epigenetic signaling 由 Sebastian Scheer, Suzanne Ackloo, Tiago da Silva Medina, Matthieu Schapira, Fengling Li, Jennifer Ward, Andrew M. Lewis, Jeffrey P. Northrop, Paul L. Richardson, H. Ümit Kanıskan, Yudao Shen, Jing Liu, David Smil, David McLeod, Carlos Zepeda‐Velázquez, Minkui Luo, Jian Jin, Dalia Baršytė-Lovejoy, K. Huber, Daniel D. De Carvalho, Masoud Vedadi, Colby Zaph, Peter J. Brown, C.H. Arrowsmith
出版 2018Artigo -
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Erratum: Pharmacological targeting of the Wdr5-MLL interaction in C/EBPα N-terminal leukemia. 由 Florian Grebien, Masoud Vedadi, Matthäus Getlik, Roberto Giambruno, Amit Grover, Roberto Avellino, Anna Skucha, Sarah Vittori, Ekaterina Kuznetsova, David Smil, Dalia Baršytė-Lovejoy, Fengling Li, Gennadiy Poda, Matthieu Schapira, Hong Wu, Aiping Dong, Guillermo Senisterra, Alexey Stukalov, K. Huber, Andreas Schönegger, Richard Marcellus, Martin Bilban, Christoph Bock, Peter J. Brown, Johannes Zuber, Keiryn L. Bennett, Rima Al‐awar, Ruud Delwel, Claus Nerlov, C.H. Arrowsmith, Giulio Superti‐Furga
出版 2015Errata/Corrigenda -
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A Potent, Selective and Cell‐Active Allosteric Inhibitor of Protein Arginine Methyltransferase 3 (PRMT3) 由 H. Ümit Kanıskan, Magdalena M. Szewczyk, Zhengtian Yu, Mohammad S. Eram, Xiaobao Yang, Keith T. Schmidt, Xiao Luo, Miao Dai, Feng He, Irene Zang, Ying Lin, Sidney H. Kennedy, Fengling Li, E. Dobrovetsky, Aiping Dong, David Smil, Sun‐Joon Min, Melissa Landon, Jennifer Lin‐Jones, Xi‐Ping Huang, Bryan L. Roth, Matthieu Schapira, Peter Atadja, Dalia Baršytė-Lovejoy, C.H. Arrowsmith, Peter J. Brown, Kehao Zhao, Jian Jin, Masoud Vedadi
出版 2015Artigo -
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Pharmacological targeting of the Wdr5-MLL interaction in C/EBPα N-terminal leukemia 由 Florian Grebien, Masoud Vedadi, Matthäus Getlik, Roberto Giambruno, Amit Grover, Roberto Avellino, Anna Skucha, Sarah Vittori, Ekaterina Kuznetsova, David Smil, Dalia Baršytė-Lovejoy, Fengling Li, Gennadiy Poda, Matthieu Schapira, Hong Wu, Aiping Dong, Guillermo Senisterra, Alexey Stukalov, K. Huber, Andreas Schönegger, Richard Marcellus, Martin Bilban, Christoph Bock, Peter J. Brown, Johannes Zuber, Keiryn L. Bennett, Rima Al‐awar, Ruud Delwel, Claus Nerlov, C.H. Arrowsmith, Giulio Superti‐Furga
出版 2015Artigo -
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MLL5 Orchestrates a Cancer Self-Renewal State by Repressing the Histone Variant H3.3 and Globally Reorganizing Chromatin 由 Marco Gallo, Fiona J. Coutinho, Robert J. Vanner, Tenzin Gayden, Stephen C. Mack, Alex Murison, Marc Remke, Li Ren, Naoya Takayama, Kinjal Desai, Lilian Lee, Xiaoyang Lan, Nicole I. Park, Dalia Baršytė-Lovejoy, David Smil, Dominik Sturm, Michelle Kushida, Renee Head, Michael D. Cusimano, Mark Bernstein, Ian D. Clarke, John E. Dick, Stefan M. Pfister, Jeremy N. Rich, C.H. Arrowsmith, Michael D. Taylor, Nada Jabado, David P. Bazett‐Jones, Mathieu Lupien, Peter B. Dirks
出版 2015Artigo -
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Functional interdependence of BRD4 and DOT1L in MLL leukemia 由 Omer Gilan, Enid Y.N. Lam, Isabelle Becher, Dave Lugo, Ester Cannizzaro, Gérard Joberty, Aoife Ward, Meike Wiese, Chun Yew Fong, Sarah Ftouni, Dean Tyler, Kym L. Stanley, Laura MacPherson, Chen-Fang Weng, Yih-Chih Chan, Margherita Ghisi, David Smil, Christopher Carpenter, Peter J. Brown, Neil Garton, Marnie E. Blewitt, Andrew J. Bannister, Tony Kouzarides, Brian J.P. Huntly, Ricky W. Johnstone, Gerard Drewes, Sarah‐Jane Dawson, C.H. Arrowsmith, Paola Grandi, Rab K. Prinjha, Mark A. Dawson
出版 2016Artigo
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Biology
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Methyltransferase
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Computational biology
Histone
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Allosteric regulation
Arginine
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